Synthesis, analgesic, anti-inflammatory and antibacterial activities of some novel 2-methylthio-3-substituted quinazolin-4-(3H)-ones

Biological and Pharmaceutical Bulletin

Volumn 27, Issue 5, 2004, Pages 652-656

  Alagarsamy, Veerachamy ^a   Rajesh, Ramadoss ^a   Ramaseshu, Meena ^b   Vijaykumar, Sukumaran ^b   Ramseshu, Kona Venkat ^b   Duraianandakumar, Thirumoorthy ^b  

^a JSS COLLEGE OF PHARMACY   (India)

^b K M COLLEGE OF PHARMACY   (India)

Author keywords

Analgesic; Anti inflammatory; Pyrimidine; Quinazoline; Thiourea

Indexed keywords

(2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)DITHIOCARBAMIC ACID METHYL ESTER; 1 (MORPHOLINYL) 3 (2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)THIOUREA; 1 (PYRROLIDINYL) 3 (2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)THIOUREA; 1 METHYL 3 (2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)THIOUREA; 1,1 DIETHYL 3 (2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)THIOUREA; 1,1 DIMETHYL 3 (2 METHYLTHIO 4 OXO 3 QUINAZOLIN 3 YL)THIOUREA; AMINE; CARBAMIC ACID DERIVATIVE; DICLOFENAC; QUINAZOLINONE DERIVATIVE; UNCLASSIFIED DRUG; ANALGESIC AGENT; ANTIINFECTIVE AGENT; NONSTEROID ANTIINFLAMMATORY AGENT; QUINAZOLINE DERIVATIVE;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBACTERIAL ACTIVITY; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; MOUSE; NONHUMAN; PAIN; PAW EDEMA; ANIMAL; DRUG EFFECT; METHODOLOGY; MICROBIOLOGICAL EXAMINATION; PAIN ASSESSMENT; SYNTHESIS;

ANALGESICS; ANIMALS; ANTI-BACTERIAL AGENTS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; MICE; MICROBIAL SENSITIVITY TESTS; PAIN MEASUREMENT; QUINAZOLINES;

EID: 16644386905     PISSN: 09186158     EISSN: 13475215     Source Type: Journal    
DOI: 10.1248/bpb.27.652     Document Type: Article

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