Difference in percutaneous absorption and intracutaneous distribution in guinea pigs among topical antifungal drugs (tioconazole solution, tioconazole cream, miconazole nitrate solution and bifonazole solution)

Biological and Pharmaceutical Bulletin

Volumn 27, Issue 9, 2004, Pages 1428-1432

  Sobue, Satoshi ^a   Sekiguchi, Kaneo ^a  

^a PFIZER INC   (United States)

Author keywords

Bifonazole; Guinea pig; Intracutaneous distribution; Miconazole; Percutaneous absorption; Tioconazole

Indexed keywords

ANTIFUNGAL AGENT; BIFONAZOLE; MICONAZOLE NITRATE; TIOCONAZOLE; IMIDAZOLE DERIVATIVE; MICONAZOLE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DERMATOMYCOSIS; DERMATOPHYTE; DRUG ABSORPTION; DRUG FORMULARY; EPIDERMIS; GUINEA PIG; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; SKIN; SKIN ABSORPTION; STRATUM CORNEUM; SUBCUTANEOUS TISSUE; YEAST; ANIMAL; AREA UNDER THE CURVE; COMPARATIVE STUDY; DRUG ADMINISTRATION; DRUG DOSAGE FORM; INTRADERMAL DRUG ADMINISTRATION; METABOLISM;

ADMINISTRATION, CUTANEOUS; ANIMALS; ANTIFUNGAL AGENTS; AREA UNDER CURVE; DOSAGE FORMS; DRUG ADMINISTRATION SCHEDULE; GUINEA PIGS; IMIDAZOLES; MICONAZOLE; SKIN;

EID: 16644385791     PISSN: 09186158     EISSN: 13475215     Source Type: Journal    
DOI: 10.1248/bpb.27.1428     Document Type: Article

References (31)

1. Clissold S. P., Heel R. C., Drugs, 31, 29-51 (1986).
2. Marriott M. S., Baird J. R., Brammer K. W., Faulkner J. K., Halliwell G., Jevons S., Tarbit M. H., Dermatologica, 166, 1S-7S (1983).
3. Kawasaki K., Niimi H., Oki T., Jpn. Pharmacol. Ther., 10, 3863-3877 (1982).
4. Lackner T. E., Clissold S. P., Drugs, 38, 204-225 (1989).
5. Odds F. C., Webster C. E., Abbott A. B., J. Antimicrob. Chemother., 14, 105-114 (1984).
6. Hiratani T., Nagata J., Yamaguchi H., Chemotherapy, 34, 125-136 (1986).
7. Beggs W. H., Andrews F. A., Sarosi G. A., Life Sci., 28, 111-118 (1981).
8. Beggs W. H., Antimicrob. Agents Chemother., 26, 699-701 (1984).
9. Yamaguchi H., Hiratani T., Nagata J., Uchida K., Chemotherapy, 34, 146-156 (1986).
10. Lefler E., Stevens D. A., Antimicrob. Agents Chemother., 25, 450-454 (1984).
11. Clayton Y. M., Hay R. J., McGibbon D. H., Pye R. J., Clin. Exp. Dermatol., 7, 543S-549S (1982).
12. Tioconazole Study Group, Nishinihon J. Dermatol. 44, 425-443 (1982).
13. Tioconazole Study Group, Nishinihon J. Dermatol. 44, 444-451 (1982).
14. O'Neill East M., Henderson J. T., Jevons S., Dermatologica, 166, 20S-33S (1983).
15. Matsuda T., Hori Y., Matsumoto T., Nishinihon J. Dermatol. 58, 138-143 (1996).
16. Haustein U. F., Seebacher C., Taube K. M., Dermatol. Monatsschr., 175, 751-756 (1989).
17. Alchorne M. M., Paschoalick R. C., Forjaz M. H., Clin. Ther., 9, 360-367 (1987).
18. del Palacio Hernanz A., Lopez Gomez S., Iglesias Diez L., Clin. Ther., 9, 333-338 (1987).
19. Enogaki K., Tatematsu H., Yoshida K., Ito M., Shimooka K., Oki T., Iyakuhin Kenkyu, 16, 759-768 (1985).
20. Lucker P. W., Beubler E., Kukovetz W. R., Ritter W., Dermatologica, 169, 51S-55S (1984).
21. Veronese M., Bertoncini A., Preti P. M., Mykosen, 30, 386-390 (1987).
22. Hood D. B., "Cutaneous Toxicology," eds. by Drill V. A., Lazar P., Academic, New York, 1977, p. 15.
23. Tregear R., "The permeability of skin to molecules of widely differing properties. Progress in Biological Science in Relation to Dermatology," eds. by Rock A. J., Cambridge Univ. Press, London, 1962.
24. Kashin P., Phyfferoen M. C., Gibbs D. L., J. Int. Med. Res., 13, 88-95 (1985).
25. Patzschke K., Ritter W., Siefert H. M., Weber H., Wegner L. A., Arzneimittelforschung, 33, 745-750 (1983).
26. Agut J., Moren M., Rego M., Sacristan A., Ortiz J. A., Arzneimittelforschung, 42, 748-751 (1992).
27. Ramis J., Conte L., Segado X., Forn J., Lauroba J., Calpena A., Escribano E., Domenech J., Arzneimittelforschung, 47, 1139-1144 (1997).
28. Tsai J., Chuang S., Hsu M., Sheu H., Int. J. Pharm., 188, 145-153 (1999).
29. Tokudome Y., Sugibayashi K., Biol. Pharm. Bull., 26, 1508-1510 (2003).
30. Rougier A., Rallis M., Krien P., Lotte C., Arch. Dermatol. Res., 282, 498-505 (1990).
31. Surber C., Wilhelm K. P., Hori M., Maibach H. I., Guy R. H., Pharm. Res., 7, 1320-1324 (1990).