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Volumn 77, Issue 2, 2004, Pages 337-343

Antagonism of anticholinesterase (DFP) toxicity by donepezil plus scopolamine: A preliminary study

Author keywords

Acetylcholine; Cholinesterase inhibitors; DFP; Diarrhea; Diisopropyl fluorophosphate; Donepezil; Flinders rats; Hypoactivity; Hypothermia; Sarin; Scopolamine; Soman

Indexed keywords

CHOLINESTERASE INHIBITOR; DONEPEZIL; DYFLOS; LONG ACTING DRUG; SCOPOLAMINE;

EID: 1642493734     PISSN: 00913057     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.pbb.2003.11.012     Document Type: Conference Paper
Times cited : (15)

References (53)
  • 1
    • 0025912177 scopus 로고
    • Effects of subacute pretreatment with carbamate together with adjunct pretreatment against nerve agent exposure
    • Anderson D.R., Harris L.W., Lennox W.J., Solana R.P. Effects of subacute pretreatment with carbamate together with adjunct pretreatment against nerve agent exposure. Drug Chem. Toxicol. 14(1-2):1991;1-19.
    • (1991) Drug Chem. Toxicol. , vol.14 , Issue.12 , pp. 1-19
    • Anderson, D.R.1    Harris, L.W.2    Lennox, W.J.3    Solana, R.P.4
  • 4
    • 0036622723 scopus 로고    scopus 로고
    • Clinical and cost-effectiveness of donepezil, rivastigmine and galantamine for Alzheimer's disease. a systematic review
    • Clegg A., Bryant J., Nicholson T., McIntyre L., De Broe S., Gerard K.et al. Clinical and cost-effectiveness of donepezil, rivastigmine and galantamine for Alzheimer's disease. A systematic review. Int. J. Technol. Assess Health Care. 18:2002;497-507.
    • (2002) Int. J. Technol. Assess Health Care , vol.18 , pp. 497-507
    • Clegg, A.1    Bryant, J.2    Nicholson, T.3    McIntyre, L.4    De Broe, S.5    Gerard, K.6
  • 6
    • 0032910699 scopus 로고    scopus 로고
    • Ontogeny of muscarinic cholinergic supersensitivity in the Flinders sensitive line rat
    • Daws L.C., Overstreet D.H. Ontogeny of muscarinic cholinergic supersensitivity in the Flinders sensitive line rat. Pharmacol. Biochem. Behav. 62:1999;367-380.
    • (1999) Pharmacol. Biochem. Behav. , vol.62 , pp. 367-380
    • Daws, L.C.1    Overstreet, D.H.2
  • 7
    • 0022637475 scopus 로고
    • Effectiveness of physostigmine as a pretreatment drug for protection of rats from organophosphate poisoning
    • Deshponde S.S., Viana G.G., Kauffman F.C., Rickett D.L., Albuquerque E.X. Effectiveness of physostigmine as a pretreatment drug for protection of rats from organophosphate poisoning. Fundam. Appl. Toxicol. 6:1986;566-577.
    • (1986) Fundam. Appl. Toxicol. , vol.6 , pp. 566-577
    • Deshponde, S.S.1    Viana, G.G.2    Kauffman, F.C.3    Rickett, D.L.4    Albuquerque, E.X.5
  • 9
    • 0018748169 scopus 로고
    • The reversal by pyridostigmine of neuromuscular block produced by soman
    • French M.C., Wetherell J.R., White P.D. The reversal by pyridostigmine of neuromuscular block produced by soman. J. Pharm. Pharmacol. 31:1979;290-294.
    • (1979) J. Pharm. Pharmacol. , vol.31 , pp. 290-294
    • French, M.C.1    Wetherell, J.R.2    White, P.D.3
  • 10
    • 0025761088 scopus 로고
    • Physostigmine (alone and together with adjunct) pretreatment against soman, sarin, tabun and VX intoxication
    • Harris L.W., Talbot B.G., Lennox W.J., Anderson D.R., Solana R.P. Physostigmine (alone and together with adjunct) pretreatment against soman, sarin, tabun and VX intoxication. Drug Chem. Toxicol. 14:1991;265-281.
    • (1991) Drug Chem. Toxicol. , vol.14 , pp. 265-281
    • Harris, L.W.1    Talbot, B.G.2    Lennox, W.J.3    Anderson, D.R.4    Solana, R.P.5
  • 12
    • 0036063785 scopus 로고    scopus 로고
    • The tolerability and safety of cholinesterase inhibitors in the treatment of dementia
    • Inglis F. The tolerability and safety of cholinesterase inhibitors in the treatment of dementia. Int. J. Clin. Pract. 127S:2002;45-63.
    • (2002) Int. J. Clin. Pract. , vol.127 , pp. 45-63
    • Inglis, F.1
  • 13
    • 0037132887 scopus 로고    scopus 로고
    • Central anticholinergics to treat nerve agent poisoning
    • Janowsky D.S. Central anticholinergics to treat nerve agent poisoning. Lancet. 359(9302):2002;265-266.
    • (2002) Lancet , vol.359 , Issue.9302 , pp. 265-266
    • Janowsky, D.S.1
  • 15
    • 0021947125 scopus 로고
    • Antagonism of physostigmine induced lethality by a combination of scopolamine and methscopolamine
    • Janowsky D.S., Berkowitz A., Turken A., Risch S.C. Antagonism of physostigmine induced lethality by a combination of scopolamine and methscopolamine. Acta Pharm. Toxicol. 56:1985;154-157.
    • (1985) Acta Pharm. Toxicol. , vol.56 , pp. 154-157
    • Janowsky, D.S.1    Berkowitz, A.2    Turken, A.3    Risch, S.C.4
  • 16
    • 1642551146 scopus 로고
    • Central versus peripheral antagonism of cholinesterase inhibitor induced lethality
    • I. Hanin. New York: Plenum Publishing
    • Janowsky D.S., Risch D.S., Berkowitz A., Turken A., Drennan M. Central versus peripheral antagonism of cholinesterase inhibitor induced lethality. Hanin I. Dynamics of cholinergic function. 1986;791-798 Plenum Publishing, New York.
    • (1986) Dynamics of Cholinergic Function , pp. 791-798
    • Janowsky, D.S.1    Risch, D.S.2    Berkowitz, A.3    Turken, A.4    Drennan, M.5
  • 17
    • 0023241530 scopus 로고
    • Antagonistic effects of scopolamine and atropine on the physostigmine response in man
    • Janowsky D., Risch S.C., Ziegler M., Gillin J.C. Antagonistic effects of scopolamine and atropine on the physostigmine response in man. Mil. Med. 152:1987;579-581.
    • (1987) Mil. Med. , vol.152 , pp. 579-581
    • Janowsky, D.1    Risch, S.C.2    Ziegler, M.3    Gillin, J.C.4
  • 18
    • 0025893153 scopus 로고
    • Pyridostigmine used as a nerve agent pretreatment under wartime conditions
    • Keeler J.F., Hurst G.G., Dunn A.L. Pyridostigmine used as a nerve agent pretreatment under wartime conditions. JAMA. 266:1991;693-695.
    • (1991) JAMA , vol.266 , pp. 693-695
    • Keeler, J.F.1    Hurst, G.G.2    Dunn, A.L.3
  • 19
    • 0032851864 scopus 로고    scopus 로고
    • Review of the value of gacyclidine (GK-11) as adjuvant medication to conventional treatments of organophosphate poisoning: Primate experiments mimicking various scenarios of military and terrorist attack by soman
    • Lallement G., Baubichon D., Clarencon D., Galnnier M., Peoc'h M., Carpentier P. Review of the value of gacyclidine (GK-11) as adjuvant medication to conventional treatments of organophosphate poisoning: primate experiments mimicking various scenarios of military and terrorist attack by soman. Neurotoxicology. 20:1999;675-684.
    • (1999) Neurotoxicology , vol.20 , pp. 675-684
    • Lallement, G.1    Baubichon, D.2    Clarencon, D.3    Galnnier, M.4    Peoc'H, M.5    Carpentier, P.6
  • 20
    • 0035003687 scopus 로고    scopus 로고
    • Subchronic administration of various pretreatments of nerve gas poisoning: II. Compared efficacy against soman toxicity
    • Lallement G., Foquin A., Dorandeu F., Baubichon D., Carpentier P. Subchronic administration of various pretreatments of nerve gas poisoning: II. Compared efficacy against soman toxicity. Drug Chem. Toxicol. 24:2001;165-180.
    • (2001) Drug Chem. Toxicol. , vol.24 , pp. 165-180
    • Lallement, G.1    Foquin, A.2    Dorandeu, F.3    Baubichon, D.4    Carpentier, P.5
  • 21
    • 0035990680 scopus 로고    scopus 로고
    • Subchronic administration of pyridostigmine or huperzine to primates: Compared efficacy against soman toxicity
    • Lallement G., Demoncheoux J.P., Foquin A., Baubichon D., Galonnier M., Clarencon D.et al. Subchronic administration of pyridostigmine or huperzine to primates: compared efficacy against soman toxicity. Drug Chem. Toxicol. 25:2002;309-320.
    • (2002) Drug Chem. Toxicol. , vol.25 , pp. 309-320
    • Lallement, G.1    Demoncheoux, J.P.2    Foquin, A.3    Baubichon, D.4    Galonnier, M.5    Clarencon, D.6
  • 25
    • 0024156788 scopus 로고
    • Prevention of soman toxicity after the continuous administration of physostigmine
    • Lim D.K., Ito Y., Yu H.J., Hoskins B., Ho I.K. Prevention of soman toxicity after the continuous administration of physostigmine. Pharmacol. Biochem. Behav. 31(3):1988;633-639.
    • (1988) Pharmacol. Biochem. Behav. , vol.31 , Issue.3 , pp. 633-639
    • Lim, D.K.1    Ito, Y.2    Yu, H.J.3    Hoskins, B.4    Ho, I.K.5
  • 26
    • 77957188346 scopus 로고
    • Trihexyphenidyl enhances physostigmine prophylaxis against poisoning in guinea pigs
    • Lim D.K., Hoskins B., Ho I.K. Trihexyphenidyl enhances physostigmine prophylaxis against poisoning in guinea pigs. Fundam. Appl. Toxicol. 16:1991;482-489.
    • (1991) Fundam. Appl. Toxicol. , vol.16 , pp. 482-489
    • Lim, D.K.1    Hoskins, B.2    Ho, I.K.3
  • 27
    • 0022458744 scopus 로고
    • Dissociation of locomotor depression and ChE activity after DFP, soman and sarin
    • Lynch M.R., Rice M.A., Robinson S.E. Dissociation of locomotor depression and ChE activity after DFP, soman and sarin. Pharmacol. Biochem. Behav. 24:1986;941-947.
    • (1986) Pharmacol. Biochem. Behav. , vol.24 , pp. 941-947
    • Lynch, M.R.1    Rice, M.A.2    Robinson, S.E.3
  • 28
    • 0023502249 scopus 로고
    • Direct microinjection of soman or VX into the amygdala produces repetitive limbic convulsions and neurophathology
    • McDonough J.H., McLeod C.G., Nipwoda M.T. Direct microinjection of soman or VX into the amygdala produces repetitive limbic convulsions and neurophathology. Brain Res. 435:1987;123-137.
    • (1987) Brain Res. , vol.435 , pp. 123-137
    • McDonough, J.H.1    McLeod, C.G.2    Nipwoda, M.T.3
  • 29
    • 0029096096 scopus 로고
    • Prophylactic transdermal treatment with physostigmine and scopolamine against soman intoxication in guinea-pigs
    • Meshulam Y., Davidovici R., Wengier A., Levy A. Prophylactic transdermal treatment with physostigmine and scopolamine against soman intoxication in guinea-pigs. J. Appl. Toxicol. 15:1995;263-266.
    • (1995) J. Appl. Toxicol. , vol.15 , pp. 263-266
    • Meshulam, Y.1    Davidovici, R.2    Wengier, A.3    Levy, A.4
  • 30
    • 0027459129 scopus 로고
    • Efficacy of physostigmine as a pretreatment for organophosphate poisoning
    • Miller S.A., Blick D.W., Kerenyi S.Z., Murphy M.R. Efficacy of physostigmine as a pretreatment for organophosphate poisoning. Pharmacol. Biochem. Behav. 44(2):1993;343-347.
    • (1993) Pharmacol. Biochem. Behav. , vol.44 , Issue.2 , pp. 343-347
    • Miller, S.A.1    Blick, D.W.2    Kerenyi, S.Z.3    Murphy, M.R.4
  • 31
    • 0031842293 scopus 로고    scopus 로고
    • Metrifonate benefits cognitive, behavioral, and global function in patients with Alzheimer's disease
    • Morris J.C., Cyrus P.A., Orazem J., Mas J., Bieber F., Rusicka B.B.et al. Metrifonate benefits cognitive, behavioral, and global function in patients with Alzheimer's disease. Neurology. 50:1998;1222-1230.
    • (1998) Neurology , vol.50 , pp. 1222-1230
    • Morris, J.C.1    Cyrus, P.A.2    Orazem, J.3    Mas, J.4    Bieber, F.5    Rusicka, B.B.6
  • 32
    • 0344643406 scopus 로고    scopus 로고
    • Assessment of a combination of physostigmine and scopolamine as pretreatment against the behavioural effects of organophosphates in the common marmoset (Callithrix jacchus)
    • Muggleton A.C., Bowditch A.F., Crofts H.S., Scott E.A.M., Pearce P.C. Assessment of a combination of physostigmine and scopolamine as pretreatment against the behavioural effects of organophosphates in the common marmoset (Callithrix jacchus). Psychopharmacology. 166:2003;212-220.
    • (2003) Psychopharmacology , vol.166 , pp. 212-220
    • Muggleton, A.C.1    Bowditch, A.F.2    Crofts, H.S.3    Scott, E.A.M.4    Pearce, P.C.5
  • 33
    • 0027513369 scopus 로고
    • The Flinders sensitive line rats: A genetic animal model of depression
    • Overstreet D.H. The Flinders sensitive line rats: a genetic animal model of depression. Neurosci. Biobehav. Rev. 17:1993;51-68.
    • (1993) Neurosci. Biobehav. Rev. , vol.17 , pp. 51-68
    • Overstreet, D.H.1
  • 35
    • 0021343462 scopus 로고
    • Selective breeding for differences in cholinergic function: Pre- and post-synaptic mechanisms involved in sensitivity to the anticholinesterase, DFP
    • Overstreet D.H., Russell R.W., Crocker A.D., Schiller G.D. Selective breeding for differences in cholinergic function: pre- and post-synaptic mechanisms involved in sensitivity to the anticholinesterase, DFP. Brain Res. 294:1984;327-332.
    • (1984) Brain Res. , vol.294 , pp. 327-332
    • Overstreet, D.H.1    Russell, R.W.2    Crocker, A.D.3    Schiller, G.D.4
  • 36
    • 0030037417 scopus 로고    scopus 로고
    • A potential animal model of multiple chemical sensitivity with cholinergic supersensitivity
    • Overstreet D.H., Miller C.M., Janowsky D.S., Russell R.W. A potential animal model of multiple chemical sensitivity with cholinergic supersensitivity. Toxicology. 111:1996;119-134.
    • (1996) Toxicology , vol.111 , pp. 119-134
    • Overstreet, D.H.1    Miller, C.M.2    Janowsky, D.S.3    Russell, R.W.4
  • 39
    • 0028228480 scopus 로고
    • Autonomic and behavioral responses of selectively bred hypercholinergic rats to oxotremorine and diisopropyl fluorophosphate
    • Rezvani A.H., Overstreet D.H., Ejantkar A., Gordon C.J. Autonomic and behavioral responses of selectively bred hypercholinergic rats to oxotremorine and diisopropyl fluorophosphate. Pharmacol. Biochem. Behav. 48:1994;703-707.
    • (1994) Pharmacol. Biochem. Behav. , vol.48 , pp. 703-707
    • Rezvani, A.H.1    Overstreet, D.H.2    Ejantkar, A.3    Gordon, C.J.4
  • 40
    • 0036063168 scopus 로고    scopus 로고
    • The efficacy of cholinesterase inhibitors in treating the behavioral symptoms of dementia
    • Rosler M. The efficacy of cholinesterase inhibitors in treating the behavioral symptoms of dementia. Int. J. Clin. Pract. 127S:2002;20-36.
    • (2002) Int. J. Clin. Pract. , vol.127 , pp. 20-36
    • Rosler, M.1
  • 41
    • 0020445075 scopus 로고
    • Selective breeding for sensitivity to DFP. Generalization of effects beyond criterion variables
    • Russell R.W., Overstreet D.H., Messenger M., Helps S.C. Selective breeding for sensitivity to DFP. Generalization of effects beyond criterion variables. Pharmacol. Biochem. Behav. l7:1982;885-891.
    • (1982) Pharmacol. Biochem. Behav. , vol.7 , pp. 885-891
    • Russell, R.W.1    Overstreet, D.H.2    Messenger, M.3    Helps, S.C.4
  • 42
    • 0033989732 scopus 로고    scopus 로고
    • Dose-response curves and time-course effects of selected anticholinergics on locomotor activity in rats
    • Sipos M.L., Burchnell V., Galbicka G. Dose-response curves and time-course effects of selected anticholinergics on locomotor activity in rats. Psychopharmacology. 147:1999;250-256.
    • (1999) Psychopharmacology , vol.147 , pp. 250-256
    • Sipos, M.L.1    Burchnell, V.2    Galbicka, G.3
  • 43
    • 0021192673 scopus 로고
    • An assessment of comparative acute toxicity of diisopropyl- fluorophosphate, tabun, sarin, and soman in relation to cholinergic and GABAergic enzyme activities in rats
    • Sivam S.P., Hoskins B., Ho I.K. An assessment of comparative acute toxicity of diisopropyl-fluorophosphate, tabun, sarin, and soman in relation to cholinergic and GABAergic enzyme activities in rats. Fundam. Appl. Toxicol. 4:1984;531-538.
    • (1984) Fundam. Appl. Toxicol. , vol.4 , pp. 531-538
    • Sivam, S.P.1    Hoskins, B.2    Ho, I.K.3
  • 44
    • 0025697241 scopus 로고
    • Evaluation of the efficacy of two carbamates, physostigmine and pyridostigmine, when used in conjunction for protection against organophosphate exposure
    • Solana R.P., Gennings D., Carter W.H.J., Anderson D., Lennox W.J., Carchman R.A.et al. Evaluation of the efficacy of two carbamates, physostigmine and pyridostigmine, when used in conjunction for protection against organophosphate exposure. Fundam. Appl. Toxicol. 15:1990;814-819.
    • (1990) Fundam. Appl. Toxicol. , vol.15 , pp. 814-819
    • Solana, R.P.1    Gennings, D.2    Carter, W.H.J.3    Anderson, D.4    Lennox, W.J.5    Carchman, R.A.6
  • 45
    • 0030849914 scopus 로고    scopus 로고
    • The role of excitotoxicity in organophosphorous nerve agents central poisoning
    • Solberg Y., Belkin M. The role of excitotoxicity in organophosphorous nerve agents central poisoning. TIPS. 18:1997;183-185.
    • (1997) TIPS , vol.18 , pp. 183-185
    • Solberg, Y.1    Belkin, M.2
  • 46
    • 0037622682 scopus 로고    scopus 로고
    • Nicotinic acetylcholine receptor-mediated neuroprotection by donepezil against glutamate neurotoxicity in rat cortical neurons
    • Takada Y., Yonezawa A., Kume T., Katsuki H., Kaneko S., Sugimoto H.et al. Nicotinic acetylcholine receptor-mediated neuroprotection by donepezil against glutamate neurotoxicity in rat cortical neurons. J. Pharmacol. Exp. Ther. 306:2003;772-777.
    • (2003) J. Pharmacol. Exp. Ther. , vol.306 , pp. 772-777
    • Takada, Y.1    Yonezawa, A.2    Kume, T.3    Katsuki, H.4    Kaneko, S.5    Sugimoto, H.6
  • 47
    • 0000605095 scopus 로고    scopus 로고
    • Anticholinesterase agents
    • J.G. Hardman, L.E. Limbird, P.B. Molinoff, R.W. Luddon, & A.G. Gilman. New York: McGraw-Hill
    • Taylor P. Anticholinesterase agents. Hardman J.G., Limbird L.E., Molinoff P.B., Luddon R.W., Gilman A.G. The pharmacological basis of therapeutics. 1996;131-149 McGraw-Hill, New York.
    • (1996) The Pharmacological Basis of Therapeutics , pp. 131-149
    • Taylor, P.1
  • 48
    • 0029951072 scopus 로고    scopus 로고
    • Sarin: Guidelines on the management of victims of a nerve gas attack
    • Volans A.P. Sarin: guidelines on the management of victims of a nerve gas attack. J. Accid. Emerg. Med. 13:1996;202-206.
    • (1996) J. Accid. Emerg. Med. , vol.13 , pp. 202-206
    • Volans, A.P.1
  • 49
    • 77957176766 scopus 로고
    • Efficacy evaluation of physostigmine and anticholinergic adjuncts as a pretreatment for nerve agent intoxication
    • Von Bredow J., Corcoran K., Maitland G., Kaminskis A., Adams N., Wade J. Efficacy evaluation of physostigmine and anticholinergic adjuncts as a pretreatment for nerve agent intoxication. Fundam. Appl. Toxicol. 17:1991;782-789.
    • (1991) Fundam. Appl. Toxicol. , vol.17 , pp. 782-789
    • Von Bredow, J.1    Corcoran, K.2    Maitland, G.3    Kaminskis, A.4    Adams, N.5    Wade, J.6
  • 50
    • 0027536883 scopus 로고
    • Effect of pyridostigmine pretreatment, HI-6 and toxogonin treatment on rat tracheal smooth muscle response to cholinergic stimulation after organophosphorus inhalation exposure
    • Walday P., Aas P., Haider T., Fonnum F. Effect of pyridostigmine pretreatment, HI-6 and toxogonin treatment on rat tracheal smooth muscle response to cholinergic stimulation after organophosphorus inhalation exposure. Arch. Toxicol. 67:1993;212-219.
    • (1993) Arch. Toxicol. , vol.67 , pp. 212-219
    • Walday, P.1    Aas, P.2    Haider, T.3    Fonnum, F.4
  • 51
    • 0028584225 scopus 로고
    • Continuous administration of low dose rates of physostigmine and hyoscine in guinea-pigs prevents the toxicity and reduces the incapacitation produced by soman poisoning
    • Wetherell J.R. Continuous administration of low dose rates of physostigmine and hyoscine in guinea-pigs prevents the toxicity and reduces the incapacitation produced by soman poisoning. J. Pharm. Pharmacol. 46:1994;1023-1028.
    • (1994) J. Pharm. Pharmacol. , vol.46 , pp. 1023-1028
    • Wetherell, J.R.1
  • 52
    • 0036302138 scopus 로고    scopus 로고
    • Donepezil and rivastigmine in the treatment of Alzheimer's disease: A best-evidence synthesis of the published data on the efficacy and cost-effectiveness
    • Wolfson C., Oremus M., Shukla V., Momoli F., Demers L., Perrault A.et al. Donepezil and rivastigmine in the treatment of Alzheimer's disease: a best-evidence synthesis of the published data on the efficacy and cost-effectiveness. Clin. Ther. 24:2002;862-886.
    • (2002) Clin. Ther. , vol.24 , pp. 862-886
    • Wolfson, C.1    Oremus, M.2    Shukla, V.3    Momoli, F.4    Demers, L.5    Perrault, A.6
  • 53
    • 0019540611 scopus 로고
    • The inhibition and protection of cholinesterase by physostigmine and pyridostigmine against soman poisoning in vivo
    • Xia D.Y., Wang L.X., Pei S.Q. The inhibition and protection of cholinesterase by physostigmine and pyridostigmine against soman poisoning in vivo. Fundam. Appl. Toxicol. 1:1981;217-221.
    • (1981) Fundam. Appl. Toxicol. , vol.1 , pp. 217-221
    • Xia, D.Y.1    Wang, L.X.2    Pei, S.Q.3


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