A facile one-pot microwave assisted conversion of 3′-5′- dibromo/diiodo-4′-hydroxy substituted chalcones to 2-substituted-4,6- diaryl pyrimidines using S-benzylisothiouronium chloride (SBT) and their antibacterial activities

Afinidad

Volumn 60, Issue 508, 2003, Pages 558-562

  Gahlot, Udaibhan S ^a   Rao, Surendra S ^a   Dulawat, Shiv S ^a   Ameta, K L ^a   Verma, B L ^a  

^a M L SUKHADIA UNIVERSITY   (India)

Author keywords

Antibacterial; Chalcones; Microwave; Pyrimidines; SBT

Indexed keywords

ACETOPHENONE DERIVATIVE; ALDEHYDE; ANTIINFECTIVE AGENT; BENZYL DERIVATIVE; CHALCONE DERIVATIVE; PYRIMIDINE DERIVATIVE; PYRROLIDINE DERIVATIVE; S BENZYLISOTHIOURONIUM CHLORIDE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MICROWAVE RADIATION; NONHUMAN; POLYMERIZATION; PROTON NUCLEAR MAGNETIC RESONANCE; REDUCTION; SEPARATION TECHNIQUE;

EID: 1642325807     PISSN: 00019704     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (23)

1. Caddick, S.: Tetrahedron, 1995, 51, 10403.
2. Galema, S.A.: Chem. Soc. Rev., 1997, 26, 233.
3. Bose, A.K.; Banik, B.K.; Lavlinskaia, N.; Jayaraman, M. and Manhas, M.S.: Chem. Tech., 1997, 27, 28.
4. Mogilaiah, K.; Vasudeva Reddy, N. and Babu Rao, R.: Indian J. Heterocyclic Chem., 2002, 11, 253.
5. Dandia, A.; Singh, R. and Arya, K.: Indian J. Heterocyclic Chem., 2002, 11, 269.
6. Paul, S. and Gupta, R.: Indian J. Chem., 1998, 37B, 1279.
7. Ameta, K.L. and Verma, B.L.: J. Indian Chem. Soc., 2002, 79, 840.
8. Vyas, R.: «Studies Related to Chalcones», Ph.D. Thesis M.L. Sukhadia University, Udaipur, Raj, India, 2000.
9. Gahlot, U.S.: «Synthesis and Reactions of Some Chalcones», Ph.D. Thesis M.L. Sukhadia University, Udaipur, Raj, India, 2002.
10. Rao, S.S.: «Synthesis and Chemical Reactions of Some Michael Acceptors», Ph.D. Thesis M.L. Sukhadia University, Udaipur, Raj, India, 2002.
11. Patil, V.D.; Wise, D.S. and Townsend, L.B.: J. Chem. Soc., Perkin Trans-I, 1980, 1853.
12. Russell, R.K.; Press, J.B.; Rampull, R.A.; Mc-Nally, J.J.; Falotico, R.; Keiser, J.A.; Bright, D.A. and Tobia, A.: J. Med. Chem., 1988, 31, 1786.
13. Narr, B. and Woitun, E.: German Offen., 2, 200, 767 (1973), Chem. Abstr., 1973, 79, 92279v.
14. Ishikawa, F.; Kossayama, A.; Yamaguchi, H.; Watanable, Y.; Saegusa, J.; Shibamura, S.; Sakuma, K.; Ashida, S. and Abiko, Y.: J. Med. Chem., 1981, 24, 376.
15. Fuchigami, T.; Yamanochi, A.; Tanaka, M.; Sakai, K. and Yamada, K.: Jpn Kokai, Tokyo Koho Jp., 61, 250, 261 (1986), Chem. Abstr., 1987, 106, 18608.
16. Janseens, F.E.; Kennis, L.E.J.; Hens, J.E.; Torremans, J.L.G. and Van, G.S.M.: European Patent Appl. Ep., 151, 826 (1985), Chem. Abstr., 1986, 104, 68861c.
17. Sukhwal, S. and Verma, B.L.: Indian J. Heterocyclic Chem., 1994, 4, 67.
18. Sharma, P.; Hussain, K.F.; Sukhwal, S.; Kothari, S.; Singhal, M. and Verma, B.L.: Indian J. Chem., 1999, 38B, 966.
19. Kothari, S.; Vyas, R. and Verma, B.L.: Indian J. Heterocyclic Chem., 1999, 8, 285.
20. Hussain, K.F.; Ashawa, A. and Verma, B.L.: Asian J. Chem., 1997, 9 (1), 86.
21. Kothari, S.; Sighal, M.; Vijayvergia, D.; Vyas, R. and Verma, B.L.: J. Indian Chem. Soc., 2000, 77, 329.
22. Rao, S.S.; Gahlot, U.S.; Dulawat, S.S.; Vyas, R.; Ameta, K.L. and Verma, B.L.: Afinidad J. Accepted, May-June, 2003, 60, N.503.
23. Baur, A.W.; Kirby, W.M.M.; Sherries, J.C. and Turk, M.: J. Clin. Pathol., 1966, 45, 493.