-
1
-
-
0037436160
-
A MurG assay which utilizes a synthetic analog of lipid I
-
Auger, G., J. van Heijenoort, D. Mengin-Lecreulx, and D. Blanot. 2003. A MurG assay which utilizes a synthetic analog of lipid I. FEMS Microbiol. Lett. 219:115-119.
-
(2003)
FEMS Microbiol. Lett.
, vol.219
, pp. 115-119
-
-
Auger, G.1
Van Heijenoort, J.2
Mengin-Lecreulx, D.3
Blanot, D.4
-
2
-
-
0036629192
-
A multitarget assay for inhibitors of membrane-associated steps of peptidoglycan biosynthesis
-
Barbosa, M. D. F. S., H. O. Ross, M. C. Hillman, R. P. Meade, M. G. Kurilla, and D. L. Pompliano. 2002. A multitarget assay for inhibitors of membrane-associated steps of peptidoglycan biosynthesis. Anal. Biochem. 306:17-22.
-
(2002)
Anal. Biochem.
, vol.306
, pp. 17-22
-
-
Barbosa, M.D.F.S.1
Ross, H.O.2
Hillman, M.C.3
Meade, R.P.4
Kurilla, M.G.5
Pompliano, D.L.6
-
3
-
-
0030004930
-
Slow binding inhibition of phospho-N-acetylmuramyl-pentapeptide- translocase (Escherichia coli) by mureidomycin A
-
Brandish, P. E., M. K. Burnham, J. T. Lonsdale, R. Southgate, M. Inukai, and T. D. H. Bugg. 1996. Slow binding inhibition of phospho-N-acetylmuramyl- pentapeptide-translocase (Escherichia coli) by mureidomycin A. J. Biol. Chem. 271:7609-7614.
-
(1996)
J. Biol. Chem.
, vol.271
, pp. 7609-7614
-
-
Brandish, P.E.1
Burnham, M.K.2
Lonsdale, J.T.3
Southgate, R.4
Inukai, M.5
Bugg, T.D.H.6
-
4
-
-
0034192601
-
Assay for identification of inhibitors for bacterial MraY translocase or MurG transferase
-
Branstrom, A. A., S. Midha, C. B. Longley, K. Han, E. R. Baizman, and H. R. Axelrod. 2000. Assay for identification of inhibitors for bacterial MraY translocase or MurG transferase. Anal. Biochem. 280:315-319.
-
(2000)
Anal. Biochem.
, vol.280
, pp. 315-319
-
-
Branstrom, A.A.1
Midha, S.2
Longley, C.B.3
Han, K.4
Baizman, E.R.5
Axelrod, H.R.6
-
5
-
-
0027405768
-
The final step of peptidoglycan subunit assembly in Escherichia coli occurs in the cytoplasm
-
Bupp, K., and J. van Heijenoort. 1993. The final step of peptidoglycan subunit assembly in Escherichia coli occurs in the cytoplasm. J. Bacteriol. 175:1841-1843.
-
(1993)
J. Bacteriol.
, vol.175
, pp. 1841-1843
-
-
Bupp, K.1
Van Heijenoort, J.2
-
6
-
-
0035115653
-
Novel scintillation proximity assay for measuring membrane-associated steps of peptidoglycan biosynthesis in Escherichia coli
-
Chandrakala, B., B. C. Elias, U. Mehra, N. S. Umapathy, P. Dwarakanath, T. S. Balganesh, and S. M. de Sousa. 2001. Novel scintillation proximity assay for measuring membrane-associated steps of peptidoglycan biosynthesis in Escherichia coli. Antimicrob. Agents Chemother. 45:768-775.
-
(2001)
Antimicrob. Agents Chemother.
, vol.45
, pp. 768-775
-
-
Chandrakala, B.1
Elias, B.C.2
Mehra, U.3
Umapathy, N.S.4
Dwarakanath, P.5
Balganesh, T.S.6
De Sousa, S.M.7
-
7
-
-
0346101458
-
High-throughput screen for inhibitors of transglycosylase and/or transpeptidase activities of Escherichia coli penicillin binding protein 1b
-
Chandrakala, B., R. K. Shandil, U. Mehra, S. Ravishankar, P. Kaur, V. Usha, B. Joe, and S. M. de Sousa. 2004. High-throughput screen for inhibitors of transglycosylase and/or transpeptidase activities of Escherichia coli penicillin binding protein 1b. Antimicrob. Agents Chemother. 48:30-40.
-
(2004)
Antimicrob. Agents Chemother.
, vol.48
, pp. 30-40
-
-
Chandrakala, B.1
Shandil, R.K.2
Mehra, U.3
Ravishankar, S.4
Kaur, P.5
Usha, V.6
Joe, B.7
De Sousa, S.M.8
-
8
-
-
0037188393
-
Intrinsic lipid preferences and kinetic mechanism of Escherichia coli MurG
-
Chen, L., H. Men, S. Ha, X. Y. Ye, L. Brunner, Y. Hu, and S. Walker. 2002. Intrinsic lipid preferences and kinetic mechanism of Escherichia coli MurG. Biochemistry 41:6824-6833.
-
(2002)
Biochemistry.
, vol.41
, pp. 6824-6833
-
-
Chen, L.1
Men, H.2
Ha, S.3
Ye, X.Y.4
Brunner, L.5
Hu, Y.6
Walker, S.7
-
9
-
-
0000885268
-
Scintillation proximity assay: A versatile high throughput screening technology
-
Cook, N. D. 1996. Scintillation proximity assay: a versatile high throughput screening technology. Drug Discov. Today 1:87-294.
-
(1996)
Drug Discov. Today
, vol.1
, pp. 87-294
-
-
Cook, N.D.1
-
10
-
-
0032930890
-
UDP-N-acetylglucosamine:N-acetylmuramoyl-(pentapeptide) pyrophosphoryl undecaprenol N-acetylglucosamine transferase from Escherichia coli: Overproduction, solubilization, and purification
-
Crouvoisier, M., D. Mengin-Lecreulx, and J. van Heijenoort. 1999. UDP-N-acetylglucosamine:N-acetylmuramoyl-(pentapeptide) pyrophosphoryl undecaprenol N-acetylglucosamine transferase from Escherichia coli: overproduction, solubilization, and purification. FEBS Lett. 449:289-292.
-
(1999)
FEBS Lett.
, vol.449
, pp. 289-292
-
-
Crouvoisier, M.1
Mengin-Lecreulx, D.2
Van Heijenoort, J.3
-
11
-
-
0035904887
-
Synthesis of P1-citronellyl-P2-a-D-pyranosyl pyrophosphates as potential substrates for the E. coli undecaprenyl-pyrophosphoryl-N-acetylglucosaminyl transferase MurG
-
Cudic, P., D. C. Behanna, M. K. Yu, R. G. Kruger, L. M. Szewczuk, and D. G. McCafferry. 2001. Synthesis of P1-citronellyl-P2-a-D-pyranosyl pyrophosphates as potential substrates for the E. coli undecaprenyl-pyrophosphoryl-N- acetylglucosaminyl transferase MurG. Bioorg. Med. Chem. Lett. 11:3107-3110.
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 3107-3110
-
-
Cudic, P.1
Behanna, D.C.2
Yu, M.K.3
Kruger, R.G.4
Szewczuk, L.M.5
McCafferry, D.G.6
-
12
-
-
0021363648
-
Stability of cefsulodin in aqueous buffered solutions and some intravenous admixtures
-
Das Gupta, V., and K. R. Stewart. 1981. Stability of cefsulodin in aqueous buffered solutions and some intravenous admixtures. J. Clin. Hosp. Pharm. 9:21-27.
-
(1981)
J. Clin. Hosp. Pharm.
, vol.9
, pp. 21-27
-
-
Das Gupta, V.1
Stewart, K.R.2
-
13
-
-
0036215198
-
Identification of compounds that inhibit the late stages of peptidoglycan synthesis in bacteria
-
deCenzo, M., M. Kuranda, S. Cohen, J. Babiak, Z.-D. Jiang, D. Sun, M. Hickey, P. Sanc, P. A. Bradford, P. Youngman, S. Projan, and D. M. Rothstein. 2002. Identification of compounds that inhibit the late stages of peptidoglycan synthesis in bacteria. J. Antibiot. (Tokyo) 55:288-295.
-
(2002)
J. Antibiot. (Tokyo)
, vol.55
, pp. 288-295
-
-
DeCenzo, M.1
Kuranda, M.2
Cohen, S.3
Babiak, J.4
Jiang, Z.-D.5
Sun, D.6
Hickey, M.7
Sanc, P.8
Bradford, P.A.9
Youngman, P.10
Projan, S.11
Rothstein, D.M.12
-
14
-
-
0025020741
-
Interaction of monoclonal antibodies with the enzymatic domains of penicillin-binding protein 1b of Escherichia coli
-
den Blaauwen, T., M. Aarsman, and N. Nanninga. 1990. Interaction of monoclonal antibodies with the enzymatic domains of penicillin-binding protein 1b of Escherichia coli. J. Bacteriol. 172:63-70.
-
(1990)
J. Bacteriol.
, vol.172
, pp. 63-70
-
-
Den Blaauwen, T.1
Aarsman, M.2
Nanninga, N.3
-
15
-
-
0021200835
-
Kinetics and mechanism of the degradation and epimerisation of sodium cefsulodin in aqueous solution
-
Fujita, T., and A. Koshiro. 1984. Kinetics and mechanism of the degradation and epimerisation of sodium cefsulodin in aqueous solution. Chem. Pharm. Bull. 32:3651-3661.
-
(1984)
Chem. Pharm. Bull.
, vol.32
, pp. 3651-3661
-
-
Fujita, T.1
Koshiro, A.2
-
16
-
-
0033574743
-
Vancomycin derivatives that inhibit peptidoglycan synthesis without binding D-ala-D-ala
-
Ge, M., Z. Chen, H. R. Onishi, J. Kohler, L. L. Silver, R. Kerns, S. Fukuzawa, S. Thompson, and D. Kahne. 1999. Vancomycin derivatives that inhibit peptidoglycan synthesis without binding D-ala-D-ala. Science 284:507-511.
-
(1999)
Science
, vol.284
, pp. 507-511
-
-
Ge, M.1
Chen, Z.2
Onishi, H.R.3
Kohler, J.4
Silver, L.L.5
Kerns, R.6
Fukuzawa, S.7
Thompson, S.8
Kahne, D.9
-
17
-
-
0033623762
-
The 1.9 A crystal structure of Escherichia coli MurG, a membrane-associated glycosyltransferase involved in peptidoglycan biosynthesis
-
Ha, S., D. Walker, Y. Shi, and S. Walker. 2000. The 1.9 A crystal structure of Escherichia coli MurG, a membrane-associated glycosyltransferase involved in peptidoglycan biosynthesis. Protein Sei. 9:1045-1052.
-
(2000)
Protein Sei.
, vol.9
, pp. 1045-1052
-
-
Ha, S.1
Walker, D.2
Shi, Y.3
Walker, S.4
-
18
-
-
0033595530
-
The kinetic characterization of Escherichia coli MurG using synthetic substrate analogues
-
Ha, S., E. Chang, M.-C. Lo, H. Men, P. Park, M. Ge, and S. Walker. 1999. The kinetic characterization of Escherichia coli MurG using synthetic substrate analogues. J. Am. Chem. Soc. 121:8415-8426.
-
(1999)
J. Am. Chem. Soc.
, vol.121
, pp. 8415-8426
-
-
Ha, S.1
Chang, E.2
Lo, M.-C.3
Men, H.4
Park, P.5
Ge, M.6
Walker, S.7
-
19
-
-
0021139196
-
Studies on the mechanism of action of imipenem (N-formimidoylthienamycin) in vitro: Binding to the penicillin-binding proteins (PBPs) in Escherichia coli and Pseudomonas aeruginosa, and inhibition of enzyme activities due to the PBPs in E. coli. 3
-
Hashizume, T., F. Ishino, J. Nakagawa, S. Tamaki, and M. Matsuhashi. 1984. Studies on the mechanism of action of imipenem (N-formimidoylthienamycin) in vitro: binding to the penicillin-binding proteins (PBPs) in Escherichia coli and Pseudomonas aeruginosa, and inhibition of enzyme activities due to the PBPs in E. coli. 3. Antibiot. (Tokyo) 37:394-400.
-
(1984)
Antibiot. (Tokyo)
, vol.37
, pp. 394-400
-
-
Hashizume, T.1
Ishino, F.2
Nakagawa, J.3
Tamaki, S.4
Matsuhashi, M.5
-
20
-
-
0041692300
-
Identification of active-site inhibitors of MurG using a generalizable, high-throughput glycosyltransferase screen
-
Helm, J. S., Y. Hu, L. Chen, B. Gross, and S. Walker. 2003. Identification of active-site inhibitors of MurG using a generalizable, high-throughput glycosyltransferase screen. J. Am. Chem. Soc. 125:11168-11169.
-
(2003)
J. Am. Chem. Soc.
, vol.125
, pp. 11168-11169
-
-
Helm, J.S.1
Hu, Y.2
Chen, L.3
Gross, B.4
Walker, S.5
-
21
-
-
0037417869
-
Crystal structure of the MurG:UDP-GlcNAc complex reveals common structural principles of a superfamily of glycosyltransferases
-
Hu, Y., L. Chen, S. Ha, B. Gross, B. Falcone, D. Walker, M. Mokhtarzadeh, and S. Walker. 2003. Crystal structure of the MurG:UDP-GlcNAc complex reveals common structural principles of a superfamily of glycosyltransferases. Proc. Natl. Acad. Sci. USA 100:845-849.
-
(2003)
Proc. Natl. Acad. Sci. USA
, vol.100
, pp. 845-849
-
-
Hu, Y.1
Chen, L.2
Ha, S.3
Gross, B.4
Falcone, B.5
Walker, D.6
Mokhtarzadeh, M.7
Walker, S.8
-
22
-
-
0038296043
-
A high-throughput solid-phase extraction assay capable of measuring diverse polyprenyl phosphate:sugar-1-phosphate transferases as exemplified by the WecA, MraY, and MurG proteins
-
Hyland, S. A., and M. S. Anderson. 2003. A high-throughput solid-phase extraction assay capable of measuring diverse polyprenyl phosphate:sugar-1- phosphate transferases as exemplified by the WecA, MraY, and MurG proteins. Anal. Biochem. 317:156-165.
-
(2003)
Anal. Biochem.
, vol.317
, pp. 156-165
-
-
Hyland, S.A.1
Anderson, M.S.2
-
23
-
-
0032542717
-
Substrate synthesis and activity assay for MurG
-
Men, H., P. Park, M. Ge, and S. Walker. 1998. Substrate synthesis and activity assay for MurG. J. Am. Chem. Soc. 120:2484-2485.
-
(1998)
J. Am. Chem. Soc.
, vol.120
, pp. 2484-2485
-
-
Men, H.1
Park, P.2
Ge, M.3
Walker, S.4
-
24
-
-
0025833399
-
The murG gene of Escherichia coli codes for the UDP-N-acetylglucosamine: N-acetylmuramyl-(pentapeptide) pyrophosphoryl-undecaprenol N-acetylglucosamine transferase involved in the membrane steps of peptidoglycan synthesis
-
Mengin-Lecreulx, D., L. Texier, M. Rousseau, and J. van Heijenoort. 1991. The murG gene of Escherichia coli codes for the UDP-N-acetylglucosamine: N-acetylmuramyl-(pentapeptide) pyrophosphoryl-undecaprenol N-acetylglucosamine transferase involved in the membrane steps of peptidoglycan synthesis. J. Bacteriol. 173:4625-4636.
-
(1991)
J. Bacteriol.
, vol.173
, pp. 4625-4636
-
-
Mengin-Lecreulx, D.1
Texier, L.2
Rousseau, M.3
Van Heijenoort, J.4
-
25
-
-
16244378628
-
Scintillation proximity assay for inhibitors of Escherichia coli MurG and, optionally, the MraY as well
-
poster F-1454
-
Ravishankar, S., V. P. Kumar, B. Chandrakala, S. M. Solapure, and S. M. de Sousa. 2003. Scintillation proximity assay for inhibitors of Escherichia coli MurG and, optionally, the MraY as well. 43rd Intersci. Conf. Antimicrob. Agents Chemother., poster F-1454.
-
(2003)
43rd Intersci. Conf. Antimicrob. Agents Chemother.
-
-
Ravishankar, S.1
Kumar, V.P.2
Chandrakala, B.3
Solapure, S.M.4
De Sousa, S.M.5
-
26
-
-
0034684788
-
Synthesis and biological evaluation of analogues of bacterial lipid I
-
Silva, D. J., C. L. Bowe, A. A. Branstrom, E, R. Baizman, and M. J. Sofia. 2000. Synthesis and biological evaluation of analogues of bacterial lipid I. Bioorg. Med. Chem. Lett. 10:2811-2813.
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 2811-2813
-
-
Silva, D.J.1
Bowe, C.L.2
Branstrom, A.A.3
Baizman, E.R.4
Sofia, M.J.5
-
27
-
-
16244369150
-
High-throughput screen for inhibitors of E. coli MraY
-
poster F-1455
-
Solapure, S. M., C. N. Gayathri, K. Das, B. Chandrakala, and S. M. de Sousa. 2003. High-throughput screen for inhibitors of E. coli MraY. 43rd Intersci. Conf. Antimicrob. Agents Chemother., poster F-1455.
-
(2003)
43rd Intersci. Conf. Antimicrob. Agents Chemother.
-
-
Solapure, S.M.1
Gayathri, C.N.2
Das, K.3
Chandrakala, B.4
De Sousa, S.M.5
-
28
-
-
0036215241
-
A pathway-specific cell based screening system to detect bacterial cell wall inhibitors
-
Sun, D., S. Cohen, N. Mani, C. Murphy, and D. M. Rothstein. 2002. A pathway-specific cell based screening system to detect bacterial cell wall inhibitors. J. Antibiot. 55:279-287.
-
(2002)
J. Antibiot.
, vol.55
, pp. 279-287
-
-
Sun, D.1
Cohen, S.2
Mani, N.3
Murphy, C.4
Rothstein, D.M.5
-
29
-
-
0022389693
-
Lysis of Escherichia coli by beta-lactam antibiotics: Deletion analysis of the role of penicillin-binding proteins 1A and 1B
-
Yonsif, S. Y., J. K. Broome-Smith, and B. G. Spratt. 1985. Lysis of Escherichia coli by beta-lactam antibiotics: deletion analysis of the role of penicillin-binding proteins 1A and 1B. J. Gen. Microbiol. 131:2839-2845.
-
(1985)
J. Gen. Microbiol.
, vol.131
, pp. 2839-2845
-
-
Yonsif, S.Y.1
Broome-Smith, J.K.2
Spratt, B.G.3
-
30
-
-
0037443830
-
Targeting the MraY and MurG bacterial enzymes for antimicrobial therapeutic intervention
-
Zawadzke, L. E., P. Wu, L. Cook, L. Fan, M. Casperson, M. Kishnani, D. Calambur, S. J. Hofstead, and R. Padmanabha. 2003. Targeting the MraY and MurG bacterial enzymes for antimicrobial therapeutic intervention. Anal. Biochem. 314:243-252.
-
(2003)
Anal. Biochem.
, vol.314
, pp. 243-252
-
-
Zawadzke, L.E.1
Wu, P.2
Cook, L.3
Fan, L.4
Casperson, M.5
Kishnani, M.6
Calambur, D.7
Hofstead, S.J.8
Padmanabha, R.9
-
31
-
-
0033003760
-
A simple statistical parameter for use in evaluation and validation of high throughput screening assays
-
Zhang, J.-H., T. D, Y. Chung, and K. R. Oldenburg. 1999. A simple statistical parameter for use in evaluation and validation of high throughput screening assays. J. Biomol. Screen. 4:67-73.
-
(1999)
J. Biomol. Screen
, vol.4
, pp. 67-73
-
-
Zhang, J.-H.1
Chung, Y.2
Oldenburg, K.R.3
|