Novel heterocyclic family of phenyl naphthothiazole carboxamides derived from naphthalimides: Synthesis, antitumor evaluation, and DNA photocleavage

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 9, 2005, Pages 3149-3155

  Li, Zhigang ^a   Yang, Qing ^a   Qian, Xuhong ^a,b  

^a DALIAN UNIVERSITY OF TECHNOLOGY   (China)

^b EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY   (China)

Author keywords

Antitumor; Cytotoxicity; DNA cleavage; Phenyl naphthothiazole carboxamides; Photocleavage; Synthesis

Indexed keywords

AMIDE; ANTINEOPLASTIC AGENT; IMIDE; N [2 (DIMETHYLAMINO)ETHYL] 2 (3 NITROPHENYL)NAPHTHO[2,1 D]THIAZOLE 5 CARBOXAMIDE; N [2 (DIMETHYLAMINO)ETHYL] 2 (4 METHOXYPHENYL)NAPHTHA[2,1 D]THIAZOLE 5 CARBOXAMIDE; N [2 (DIMETHYLAMINO)ETHYL] 2 (4 TOLYL)NAPHTHO[2,1 D]THIAZOLE 5 CARBOXAMIDE; N [2 (DIMETHYLAMINO)ETHYL] 2 PHENYLNAPHTHO[2,1 D]THIAZOLE 5 CARBOXAMIDE; SUPEROXIDE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL; CHEMICAL MODIFICATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYTOTOXICITY TEST; DNA CLEAVAGE; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MOUSE; NONHUMAN; QUANTITATIVE ANALYSIS;

EID: 16244367779     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.02.045     Document Type: Article

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