Cyclization of 1-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-acetyl} thiosemicarbazides to 1,2,4-triazole and 1,3,4-thiadiazole derivatives and their pharmacological properties

Collection of Czechoslovak Chemical Communications

Volumn 70, Issue 1, 2005, Pages 51-62

  Maliszewska Guz, Alicja ^a   Wujec, Monika ^a   Pitucha, Monika ^a   Dobosz, Maria ^a   Chodkowska, Anna ^a   Jagiełło Wójtowicz, Ewa ^a   Mazur, Liliana ^b   Kozioł, Anna E ^b  

^a MEDICAL UNIVERSITY OF LUBLIN   (Poland)

^b MARIA CURIE SK ODOWSKA UNIVERSITY   (Poland)

Author keywords

1,2,4 Triazoles; 1,3,4 Thiadiazoles; Antidepressives; Crystal structure determination; Cyclizations; Pharmacological screening; Thiosemicarbazides; X ray diffraction

Indexed keywords

4 ETHYL 5 [[(4 METHYL 4H 1,2,4 TRIAZOL 3 YL)SULFANYL]METHYL] 4H 1,2,4 TRIAZOLE 3(2H) THIONE; 5 [[(4 METHYL 4H 1,2,4 TRIAZOL 3 YL)SULFANYL]METHYL] 4 (4 TOLYL) 4H 1,2,4 TRIAZOLE 3(2H) THIONE; 5 [[(4 METHYL 4H 1,2,4 TRIAZOL 3 YL)SULFANYL]METHYL] 4 PHENYL 4H 1,2,4 TRIAZOLE 3(2H) THIONE; THIAZOLE DERIVATIVE; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONTROLLED STUDY; CYCLIZATION; MALE; MOUSE; NONHUMAN; REACTION ANALYSIS; STRUCTURE ANALYSIS; X RAY ANALYSIS;

EID: 15444365881     PISSN: 00100765     EISSN: None     Source Type: Journal    
DOI: 10.1135/cccc20050051     Document Type: Article

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