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Volumn 506, Issue 3, 2005, Pages 257-264

Comparative anticholinergic activities of 10 histamine H1 receptor antagonists in two functional models

Author keywords

Acetylcholine; Anticholinergic; Antihistamine; Carbachol; Histamine H1 antagonist

Indexed keywords

ATROPINE; CARBACHOL; CETIRIZINE; CHLORPHENIRAMINE MALEATE; CYPROHEPTADINE; DESLORATADINE; DIPHENHYDRAMINE; FEXOFENADINE; HISTAMINE H2 RECEPTOR ANTAGONIST; HYDROXYZINE; LORATADINE; MEPYRAMINE MALEATE; PROMETHAZINE; CHOLINERGIC RECEPTOR BLOCKING AGENT; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST;

EID: 14944341738     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2004.11.006     Document Type: Article
Times cited : (70)

References (27)
  • 2
  • 4
    • 0033028937 scopus 로고    scopus 로고
    • Anticholinergic effects of desloratadine, the major metabolite of loratadine, in rabbit and guinea-pig iris smooth muscle
    • I. Cardelús, F. Antón, J. Beleta, and J. Palacios Anticholinergic effects of desloratadine, the major metabolite of loratadine, in rabbit and guinea-pig iris smooth muscle Eur. J. Pharmacol. 374 1999 249 254
    • (1999) Eur. J. Pharmacol. , vol.374 , pp. 249-254
    • Cardelús, I.1    Antón, F.2    Beleta, J.3    Palacios, J.4
  • 5
    • 0034125545 scopus 로고    scopus 로고
    • Effects of H1 antagonists on cholinomimetics-induced tremulous jaw movements: Studies of diphenhydramine, doxepin, and mepyramine
    • B.B. Carlson, J.T. Trevitt, and J.D. Salamone Effects of H1 antagonists on cholinomimetics-induced tremulous jaw movements: studies of diphenhydramine, doxepin, and mepyramine Pharmacol. Biochem. Behav. 65 2000 683 689
    • (2000) Pharmacol. Biochem. Behav. , vol.65 , pp. 683-689
    • Carlson, B.B.1    Trevitt, J.T.2    Salamone, J.D.3
  • 6
    • 0030442725 scopus 로고    scopus 로고
    • Muscarinic receptor subtypes and smooth muscle function
    • R.M. Eglen, S.S. Hegde, and N. Watson Muscarinic receptor subtypes and smooth muscle function Pharmacol. Rev. 48 1996 531 565
    • (1996) Pharmacol. Rev. , vol.48 , pp. 531-565
    • Eglen, R.M.1    Hegde, S.S.2    Watson, N.3
  • 7
    • 4243512135 scopus 로고    scopus 로고
    • Desloratadine interacts with muscarinic acetylcholine receptors with high affinity and antagonizes the cyclic AMP response at the M2 subtype
    • J. Ellis, and M. Seidenberg Desloratadine interacts with muscarinic acetylcholine receptors with high affinity and antagonizes the cyclic AMP response at the M2 subtype J. Allergy Clin. Immunol. 107 2001 S160 (abstract 528)
    • (2001) J. Allergy Clin. Immunol. , vol.107 , pp. 160
    • Ellis, J.1    Seidenberg, M.2
  • 9
    • 0025944764 scopus 로고
    • Muscarinic receptor subtypes in guinea pig airways
    • E.B. Haddad, Y. Landry, and J.P. Gies Muscarinic receptor subtypes in guinea pig airways Am. J. Physiol. 261 1991 L327 L333
    • (1991) Am. J. Physiol. , vol.261
    • Haddad, E.B.1    Landry, Y.2    Gies, J.P.3
  • 10
    • 0026485735 scopus 로고
    • Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation
    • M.G. Hendriks, M. Pfaffendorf, and P.A. Van Zwieten Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation J. Auton. Pharmacol. 12 1992 411 420
    • (1992) J. Auton. Pharmacol. , vol.12 , pp. 411-420
    • Hendriks, M.G.1    Pfaffendorf, M.2    Van Zwieten, P.A.3
  • 11
    • 0019730409 scopus 로고
    • 3[H]mepyramine binding and from inhibition of a functional response
    • 3[H]mepyramine binding and from inhibition of a functional response J. Neurochem. 37 1981 1357 1360
    • (1981) J. Neurochem. , vol.37 , pp. 1357-1360
    • Hill, S.J.1    Daum, P.2    Young, J.M.3
  • 12
    • 0032807637 scopus 로고    scopus 로고
    • Antihistamines: Models to assess sedative properties, assessment of sedation, safety and other side-effects
    • I. Hindmarch, and Z. Shamsi Antihistamines: models to assess sedative properties, assessment of sedation, safety and other side-effects Clin. Exp. Allergy 29 1999 133 142
    • (1999) Clin. Exp. Allergy , vol.29 , pp. 133-142
    • Hindmarch, I.1    Shamsi, Z.2
  • 14
    • 0023096152 scopus 로고
    • Antimuscarinic effect of antihistamines: Quantitative evaluation by receptor binding assay
    • N. Kubo, O. Shirakawa, T. Kuno, and C. Tanaka Antimuscarinic effect of antihistamines: quantitative evaluation by receptor binding assay Jpn. J. Pharmacol. 43 1987 277 282
    • (1987) Jpn. J. Pharmacol. , vol.43 , pp. 277-282
    • Kubo, N.1    Shirakawa, O.2    Kuno, T.3    Tanaka, C.4
  • 16
    • 0024217607 scopus 로고
    • Muscarinic receptor subtypes mediating vasodilation in the pulmonary artery
    • D.G. McCormack, J.C. Mak, P. Minette, and P.J. Barnes Muscarinic receptor subtypes mediating vasodilation in the pulmonary artery Eur. J. Pharmacol. 158 1988 293 297
    • (1988) Eur. J. Pharmacol. , vol.158 , pp. 293-297
    • McCormack, D.G.1    Mak, J.C.2    Minette, P.3    Barnes, P.J.4
  • 17
    • 0020461127 scopus 로고
    • The in vivo pharmacologic profile of histamine (H1) antagonists in the rat
    • C.J.E. Niemegeers, F.H.L. Awouters, and P.A.J. Janssen The in vivo pharmacologic profile of histamine (H1) antagonists in the rat Drug Dev. Res. 2 1982 559 566
    • (1982) Drug Dev. Res. , vol.2 , pp. 559-566
    • Niemegeers, C.J.E.1    Awouters, F.H.L.2    Janssen, P.A.J.3
  • 20
    • 0017664338 scopus 로고
    • (+)- and (-)-3-methoxycyproheptadine. a comparative evaluation of the antiserotonin, antihistaminic, anticholinergic, and orexigenic properties with cyproheptadine
    • D.C. Remy, K.E. Rittle, C.A. Hunt, P.S. Anderson, E.L. Engelhardt, B.V. Clineschmidt, and A. Scriabine (+)- and (-)-3-methoxycyproheptadine. A comparative evaluation of the antiserotonin, antihistaminic, anticholinergic, and orexigenic properties with cyproheptadine J. Med. Chem. 20 1977 1681 1684
    • (1977) J. Med. Chem. , vol.20 , pp. 1681-1684
    • Remy, D.C.1    Rittle, K.E.2    Hunt, C.A.3    Anderson, P.S.4    Engelhardt, E.L.5    Clineschmidt, B.V.6    Scriabine, A.7
  • 21
    • 0011391436 scopus 로고
    • Comparisons of various histamine antagonists
    • J.J. Reuse Comparisons of various histamine antagonists Br. J. Pharmacol. 3 1948 174 179
    • (1948) Br. J. Pharmacol. , vol.3 , pp. 174-179
    • Reuse, J.J.1
  • 22
    • 0033746828 scopus 로고    scopus 로고
    • Sedation and antihistamines: A review of inter-drug differences using proportional impairment ratios
    • Z. Shamsi, and I. Hindmarch Sedation and antihistamines: a review of inter-drug differences using proportional impairment ratios Hum. Psychopharmacol. Clin. Exp. 15 2000 S3 S30
    • (2000) Hum. Psychopharmacol. Clin. Exp. , vol.15
    • Shamsi, Z.1    Hindmarch, I.2
  • 23
    • 33544455829 scopus 로고
    • Pharmacological properties of antihistamine drugs, benadryl, pyribenzamine, and neoantergan
    • T.R. Sherrod, E.R. Loew, and H.F. Schloemer Pharmacological properties of antihistamine drugs, benadryl, pyribenzamine, and neoantergan J. Pharmacol. Exp. Ther. 89 1947 247 255
    • (1947) J. Pharmacol. Exp. Ther. , vol.89 , pp. 247-255
    • Sherrod, T.R.1    Loew, E.R.2    Schloemer, H.F.3
  • 24
    • 0032810612 scopus 로고    scopus 로고
    • Non-cardiac adverse effects of antihistamines (H1-receptor antagonists)
    • F.E.R. Simons Non-cardiac adverse effects of antihistamines (H1-receptor antagonists) Clin. Exp. Allergy 29 Suppl. 3 1999 125 132
    • (1999) Clin. Exp. Allergy , vol.29 , Issue.SUPPL. 3 , pp. 125-132
    • Simons, F.E.R.1
  • 25
    • 0032919046 scopus 로고    scopus 로고
    • Second-generation antihistamines: A comparative review
    • J.W. Slater, A.D. Zechnich, and D.G. Haxby Second-generation antihistamines: a comparative review Drugs 57 1999 31 47
    • (1999) Drugs , vol.57 , pp. 31-47
    • Slater, J.W.1    Zechnich, A.D.2    Haxby, D.G.3
  • 26
    • 0027405484 scopus 로고
    • Is there a difference in the affinity of histamine H1 receptor antagonists for CNS and peripheral receptors? An in vitro study
    • A.M. Ter Laak, G.M. Donne-Op den Kelder, A. Bast, and H. Timmerman Is there a difference in the affinity of histamine H1 receptor antagonists for CNS and peripheral receptors? An in vitro study Eur. J. Pharmacol. 232 1993 199 205
    • (1993) Eur. J. Pharmacol. , vol.232 , pp. 199-205
    • Ter Laak, A.M.1    Donne-Op Den Kelder, G.M.2    Bast, A.3    Timmerman, H.4
  • 27
    • 0032970244 scopus 로고    scopus 로고
    • Cholinergic control of human and animal pulmonary vascular tone
    • L. Walch, X. Norel, B. Leconte, J.P. Gascard, and C. Brink Cholinergic control of human and animal pulmonary vascular tone Therapie 54 1999 99 102
    • (1999) Therapie , vol.54 , pp. 99-102
    • Walch, L.1    Norel, X.2    Leconte, B.3    Gascard, J.P.4    Brink, C.5


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