1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 6, 2005, Pages 1707-1711

  Lee, Mase ^a   Rangisetty, Jagadeesh B ^a   Pullagurla, Manik R ^a   Dukat, Małgorzata ^a   Setola, Vince ^b   Roth, Bryan L ^b   Glennon, Richard A ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

^b CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

5 HT6 Serotonin receptors

Indexed keywords

1 (1 NAPHTHYL)PIPERAZINE; 1 BENZENESULFONYL 5 METHOXY N,N DIMETHYLTRYPTAMINE; SEROTONIN 6 RECEPTOR; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR AFFECTING AGENT; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; STRUCTURE ACTIVITY RELATION;

EID: 14644433606     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.01.031     Document Type: Article

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