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Volumn 56, Issue 6, 2004, Pages 843-848

Introduction of a new complex imide system into the structure of LCAPs. The synthesis and a 5-HT1A, 5-HT2A and D2 receptor binding study

(4) Kossakowski, Jerzy a Raszkiewicz, Aldona a Bugno, Ryszard b Bojarski, Andrzej J b

a MEDICAL UNIVERSITY OF WARSAW (Poland)

b POLISH ACADEMY OF SCIENCES (Poland)

Author keywords

1 arylpiperazine derivatives; 5 HT1A and 5 HT2A receptor affinity; Structure activity relationship

Indexed keywords

1,3 DIPHENYLISOBENZOFURAN; 4,9 DIPHENYL 4,9 EPOXY 3A,4,9,9A 1H BENZ[F]ISOINDOLE 1,3(2H) DIONE; 5,8 DIMETHYL 3B,9 EPOXY(3A,4,5,6,7,8,9,9A)OCTAHYDRO 1H BENZ[E]ISOINDOLE 1,3 (2H) DIONE; DOPAMINE 2 RECEPTOR; IMIDE; ISOBENZOFURAN DERIVATIVE; MALEIMIDE DERIVATIVE; PIPERAZINE DERIVATIVE; RADIOLIGAND; SEROTONIN 1A RECEPTOR; SEROTONIN 2A RECEPTOR; SEROTONIN AGONIST; UNCLASSIFIED DRUG;

ALKYLATION; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING SITE; DOPAMINERGIC ACTIVITY; DRUG INHIBITION; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TOLERANCE; IN VITRO STUDY; NONHUMAN; RADIOASSAY; RAT; STRUCTURE ACTIVITY RELATION; TRANQUILIZING ACTIVITY;

IMIDES; MOLECULAR STRUCTURE; PIPERAZINES; PROTEIN BINDING; RECEPTOR, SEROTONIN, 5-HT1A; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, DOPAMINE D2;

EID: 14244262379 PISSN: 12306002 EISSN: None Source Type: Journal
DOI: None Document Type: Article

Times cited : (9)

References (10)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.