Synthetic applications of aryl radical building blocks for cyclisation onto azoles

Tetrahedron

Volumn 61, Issue 10, 2005, Pages 2689-2696

  Allin, Steven M ^a   Bowman, W Russell ^a   Elsegood, Mark R J ^a   McKee, Vickie ^a   Karim, Rehana ^a   Rahman, Shahzad S ^b  

^a LOUGHBOROUGH UNIVERSITY   (United Kingdom)

^b GLAXOSMITHKLINE   (United Kingdom)

Author keywords

Aryl radicals; Azoles; Building blocks; Heterocycles; Radical cyclisation

Indexed keywords

2 (2 BROMOPHENYL)ETHYLMETHANESULFONATE; CARBOXYLIC ACID DERIVATIVE; GERMANIUM DERIVATIVE; IMIDAZOLE DERIVATIVE; INDOLE DERIVATIVE; MESYLIC ACID DERIVATIVE; METHYL 5,6 DIHYDROIMIDAZO[2,1 A]ISOQUINOLINE 3 CARBOXYLATE; METHYL 5,6 DIHYDROIMIDAZO[5,1 A]ISOQUINOLINE 1 CARBOXYLATE; PYRAZOLE DERIVATIVE; PYRROLE DERIVATIVE; TRIBUTYLGERMANIUM; UNCLASSIFIED DRUG;

ARTICLE; CRYSTAL STRUCTURE; CYCLIZATION; PRIORITY JOURNAL; REACTION ANALYSIS; SUBSTITUTION REACTION; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

EID: 13944260490     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2005.01.064     Document Type: Article

References (33)

1. W.R. Bowman, C.F. Bridge, and P. Brookes J. Chem. Soc., Perkin Trans. 1 2000 1 14
2. W.R. Bowman, M.O. Cloonan;, and S.L. Krintel J. Chem. Soc., Perkin Trans. 1 2001 2885 2991
3. W.R. Bowman, A.J. Fletcher, and G.B.S. Potts J. Chem. Soc., Perkin Trans. 1 2002 2747 2762
4. F. Aldabbagh, W.R. Bowman, and E. Mann Tetrahedron Lett. 38 1997 7937 7940
5. F. Aldabbagh, W.R. Bowman, E. Mann, and A.M.Z. Slawin Tetrahedron 55 1999 8111 8128
6. S.M. Allin, W.R.S. Barton, W.R. Bowman, and T. McInally Tetrahedron Lett. 43 2002 4191 4193
7. Y. Antonio, E. De La Cruz, E. Galeazzi, A. Guzman, B.L. Bray, R. Greenhouse, L.J. Kurz, D.A. Lustig, M.L. Maddox, and J.M. Muchowski Can. J. Chem. 72 1994 15 22
8. F.E. Ziegler, and M. Belema J. Org. Chem. 62 1997 1083 7967
9. C.J. Moody, and C.L. Norton J. Chem. Soc., Perkin Trans. 1 1997 2639 2643
10. J.A. Murphy, and M.S. Sherburn Tetrahedron 47 1991 4077 4088
11. J. Marco-Contelles, and M. Rodríquez-Fernández Tetrahedron Lett. 41 2000 381 384
12. J. Marco-Contelles, and M. Rodríquez-Fernández J. Org. Chem. 66 2001 3717 3725
13. Y.Z. Osornio, L.D. Miranda, R. Cruz-Almaza, and J.D. Muchowski Tetrahedron Lett. 45 2004 2855 2858
14. S.M. Allin, W.R.S. Barton, W.R. Bowman, and T. McInally Tetrahedron Lett. 42 2001 7887 7890
15. W.R. Bowman, S.L. Krintel, and M.B. Schilling Org. Biomol. Chem. 2004 585 592
16. W. Zhang, and G. Pugh Tetrahedron 59 2003 3009 3018 and 4237-4247 and references therein
17. O. Tsuge, T. Hatta, and H. Tsuchiyama Chem. Lett. 1998 2003 155 156
18. S.R. Flannagan, D.C. Harrowven, and M. Bradley Tetrahedron Lett. 44 2003 1795 1798
19. T.C.T. Ho, and K. Jones Tetrahedron 53 1997 8287 8294
20. A. Nadin, and T. Harrison Tetrahedron Lett. 40 1999 4073 4076
21. K.C. Mujumbar, and P.P. Mukhopadhyay Synthesis 2003 920 924
22. K.C. Mujumbar, P.K. Basu, P.P. Mukhopadhyay, S. Sarkar, S.K. Ghosh, and P. Biswas Tetrahedron 59 2003 2151 2157
23. K. Orito, Y. Satoh, H. Nishizawa, R. Harada, and M. Tokuda Org. Lett. 2 2000 2535 2537
24. D.C. Harrowven, B.J. Sutton, and S. Coulton Tetrahedron 58 2002 3387 3400
25. D.C. Harrowven, B.J. Sutton, and S. Coulton Tetrahedron Lett. 42 2001 2907 2910
26. D.C. Harrowven, B.J. Sutton, and S. Coulton Tetrahedron Lett. 42 2001 9061 9064
27. D.C. Harrowven, B.J. Sutton, and S. Coulton Org. Biomol. Chem. 2003 4047 4057
28. B.P. Roberts Chem. Soc. Rev. 28 1999 25 35
29. A.L.J. Beckwith, W.R. Bowman, V.W. Bowry, E. Mann, J. Parr, and J.M.D. Storey Angew. Chem., Int. Ed. Engl. 43 2004 95 98
30. Review: A. Studer, and M. Bossart P. Renaud M.P. Sibi Radicals in Organic Synthesis Vol. 2 2001 Wiley-VCH Weinheim 62 80
31. Review: A. Ganesan P. Renaud M.P. Sibi Radicals in Organic Synthesis Vol. 2 2001 Wiley-VCH Weinheim 81 91
32. T.J. Colacot J. Organomet. Chem. 1999 378 381
33. Sheldrick, G.M., SHELXTL version 5.1, Bruker-AXS, Madison WI, 1998.