Claimed 2,1-benzisoxazoles are indazalones

Journal of Organic Chemistry

Volumn 70, Issue 3, 2005, Pages 1060-1062

  Kurth, Mark J ^a   Olmstead, Marilyn M ^a   Haddadin, Makhluf J ^b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b AMERICAN UNIVERSITY OF BEIRUT   (Lebanon)

Author keywords

[No Author keywords available]

Indexed keywords

DERIVATIVES; REACTION KINETICS; SUBSTITUTION REACTIONS;

2,1-BENZISOXAZOLES; INDAZALONES;

NITROGEN COMPOUNDS;

2 BENZYLINDAZALONE; 2,1 BENZISOXAZOLE; 3 METHOXY 2 BENZYL 2H INDAZOLE; INDAZALONE; INDAZOLE DERIVATIVE; ISOXAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CRYSTAL STRUCTURE; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

EID: 13244277640     PISSN: 00223263     EISSN: None     Source Type: Journal    
DOI: 10.1021/jo048153i     Document Type: Article

References (8)

1. Chen, L.-J.; Burka, L. T. Tetrahedron Lett. 1998, 39, 5351-5354.
2. Boduszek, B.; Halama, A.; Zón, J. Tetrahedron 1997, 53, 11399-11410. This reference includes more examples of alledged 2,1-benzisoxazoles prepared by the methods cited here in Scheme 2.
3. 13C NMR data of the desired product.
4. Haddadin, M. J.; Nazer, M. Z.; Olmstead, M. M.; Kurth, M. J. Unpublished results.
5. Ishikawa, F.; Watanabe, Y.; Saegusa, J. Chem. Pharm. Bull. 1980, 28, 1357-1364.
6. Bjørsvik, H,-R.; González, R. R.; Liguori, L. J. Org. Chem. 2004, 69, 7720-7727.
7. For a comprehensive review of the chemistry of indazoles, see: Stadlbauer, W. Product class 2: 1H- and 2H-indazoles. Sci. Synth. 2002, 12, 227-324.
8. Bamberger, E. Chem. Ber. 1918, 51, 606-12.