Use of a pharmacophore model for the design of EGFr tyrosine kinase inhibitors: 4-(Phenylamino)pyrazolo[3,4-d]pyrimidines

Chemtracts

Volumn 11, Issue 7, 1998, Pages 550-560

  Traxler, P ^a   Bold, G ^a   Frei, J ^a   Lang, M ^a   Lydon, N ^a   Mett, H ^a   Buchdunger, E ^a   Meyer, T ^a   Mueller, M ^a   Furet, P ^a  

^a NONE

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 BROMOANILINO) 6,7 DIMETHOXYQUINAZOLINE; 4 (PHENYLAMINO)PYRAZOLO[3,4 D]PYRIMIDINE; 4 (PHENYLAMINO)PYRROLOPYRIMIDINE; DRUG CARRIER; ENZYME INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE; PROTEIN TYROSINE KINASE INHIBITOR; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

COMPETITIVE INHIBITION; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME LINKED IMMUNOSORBENT ASSAY; REVIEW;

EID: 13144261724     PISSN: 14319268     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

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