1-(Phenyl)isoquinoline carboxamides: A novel class of subtype selective inhibitors of thyrotropin-releasing hormone (TRH) receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 3, 2005, Pages 733-736

  Jiang, Jian Kang ^a   Thomas, Craig J ^a   Neumann, Susanne ^a   Lu, Xinping ^a   Rice, Kenner C ^a   Gershengorn, Marvin C ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

PK 11195; TRH; TRH receptors

Indexed keywords

AMIDE; LIGAND; PROTIRELIN RECEPTOR; PROTIRELIN RECEPTOR 1; PROTIRELIN RECEPTOR 2; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS;

AMIDES; ANIMALS; BINDING, COMPETITIVE; ISOQUINOLINES; LIGANDS; MICE; RADIOLIGAND ASSAY; RECEPTORS, THYROTROPIN-RELEASING HORMONE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 12444299951     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.017     Document Type: Article

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