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Volumn 137, Issue 8, 2002, Pages 1217-1224

Smooth muscle 5-HT 2A receptors mediating contraction of porcine isolated proximal stomach strips

Author keywords

5 HT 2A receptors; Fundus; Ketanserin; Pig; Proximal stomach

Indexed keywords

1 (1 METHYL 5 INDOLYL) 3 (3 METHYL 5 ISOTHIAZOLYL)UREA; 1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; ALPHA METHYLSEROTONIN; ATROPINE; FLUOXETINE; GRANISETRON; KETANSERIN; MESULERGINE; METHYSERGIDE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; OMEGA CONOTOXIN; PARGYLINE; RITANSERIN; SEROTONIN 2A RECEPTOR; SEROTONIN 3 RECEPTOR; SEROTONIN 4 RECEPTOR; SEROTONIN ANTAGONIST; TETRODOTOXIN; UNCLASSIFIED DRUG;

EID: 12244308529     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704992     Document Type: Article
Times cited : (16)

References (28)
  • 1
    • 0028300802 scopus 로고
    • Further characterization of 5-hydroxytryptamine receptors (putative 5-HT2B) in rat stomach fundus longitudinal muscle
    • Baxter, G.S., Murphy, O.E. & Blackburn, T.P. (1994). Further characterization of 5-hydroxytryptamine receptors (putative 5-HT2B) in rat stomach fundus longitudinal muscle. Br. J. Pharmacol., 112, 323-331.
    • (1994) Br. J. Pharmacol. , vol.112 , pp. 323-331
    • Baxter, G.S.1    Murphy, O.E.2    Blackburn, T.P.3
  • 2
    • 0022271882 scopus 로고
    • Further analysis of anomalous pKB values for histamine H2-receptor antagonists on the mouse isolated stomach assay
    • Black, J.W., Leff, P. & Shankley, N.P. (1985). Further analysis of anomalous pKB values for histamine H2-receptor antagonists on the mouse isolated stomach assay. Br. J. Pharmacol., 86, 581-587.
    • (1985) Br. J. Pharmacol. , vol.86 , pp. 581-587
    • Black, J.W.1    Leff, P.2    Shankley, N.P.3
  • 3
    • 0023912384 scopus 로고
    • In vitro studies with ICI 169,369, a chemically novel 5-HT antagonist
    • Blackburn, T.P., Thornber, C.W., Pearce, R.J. & Cox, B. (1988). In vitro studies with ICI 169,369, a chemically novel 5-HT antagonist. Eur. J. Pharmacol., 150, 247-256.
    • (1988) Eur. J. Pharmacol. , vol.150 , pp. 247-256
    • Blackburn, T.P.1    Thornber, C.W.2    Pearce, R.J.3    Cox, B.4
  • 4
    • 0028107979 scopus 로고
    • Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro
    • Buchheit, K.H. & Buhl, T. (1994). Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro. Eur. J. Pharmacol., 262, 91-97.
    • (1994) Eur. J. Pharmacol. , vol.262 , pp. 91-97
    • Buchheit, K.H.1    Buhl, T.2
  • 5
    • 0030609834 scopus 로고    scopus 로고
    • Influence of 5-HT1A receptor antagonism on plus-maze behaviour in mice. II. WAY 100635, SDZ 216-525 and NAN-190
    • Cao, B.J. & Rodgers, R.J. (1997). Influence of 5-HT1A receptor antagonism on plus-maze behaviour in mice. II. WAY 100635, SDZ 216-525 and NAN-190. Pharm. Biochem. Behav., 58, 593-603.
    • (1997) Pharm. Biochem. Behav. , vol.58 , pp. 593-603
    • Cao, B.J.1    Rodgers, R.J.2
  • 6
    • 0032914788 scopus 로고    scopus 로고
    • Role of nitric oxide in fasting gastric fundus tone and in 5-HT1 receptor-mediated relaxation of gastric fundus
    • Coulie, B., Tack, J., Sifrim, D., Andrioli, A. & Janssens, J. (1999). Role of nitric oxide in fasting gastric fundus tone and in 5-HT1 receptor-mediated relaxation of gastric fundus. Am. J. Physiol., 276, G373-G377.
    • (1999) Am. J. Physiol. , vol.276
    • Coulie, B.1    Tack, J.2    Sifrim, D.3    Andrioli, A.4    Janssens, J.5
  • 7
    • 0029646696 scopus 로고
    • N-(1-Methyl-5-indolyl)-N′-(3-methyl-5-isothiazolyl) urea: A novel, high-affinity 5-HT2B receptor antagonist
    • Forbes, I.T., Jones, G.E., Murphy, O.E., Holland, V. & Baxter, G.S. (1995). N-(1-Methyl-5-indolyl)-N′-(3-methyl-5-isothiazolyl) urea: A novel, high-affinity 5-HT2B receptor antagonist. J. Med. Chem., 38, 855-857.
    • (1995) J. Med. Chem. , vol.38 , pp. 855-857
    • Forbes, I.T.1    Jones, G.E.2    Murphy, O.E.3    Holland, V.4    Baxter, G.S.5
  • 9
    • 0000009439 scopus 로고    scopus 로고
    • Extensive pharmacological study of the G-protein coupled fraction of human 5-HT receptors using agonist radioligand binding
    • Gommeren, W., Renders, J., van Gompel, P., Lesage, A., Leysen, J.E. & Jurzak, M. (1998). Extensive pharmacological study of the G-protein coupled fraction of human 5-HT receptors using agonist radioligand binding. Naunyn-Schmiedeberg's Arch. Pharmacol., 358, 8.42.
    • (1998) Naunyn-Schmiedeberg's Arch. Pharmacol. , vol.358 , pp. 842
    • Gommeren, W.1    Renders, J.2    Van Gompel, P.3    Lesage, A.4    Leysen, J.E.5    Jurzak, M.6
  • 10
    • 0030265544 scopus 로고    scopus 로고
    • Peripheral 5-HT4 receptors
    • Hegde, S.S. & Eglen, R.M. (1996). Peripheral 5-HT4 receptors. FASEB J., 10, 1398-1407.
    • (1996) FASEB J. , vol.10 , pp. 1398-1407
    • Hegde, S.S.1    Eglen, R.M.2
  • 12
    • 0026004944 scopus 로고
    • 5-HT receptors: Subtypes and second messengers
    • Hoyer, D. & Schoeffter, P. (1991). 5-HT receptors: Subtypes and second messengers. J. Recept. Res., 11, 197-214.
    • (1991) J. Recept. Res. , vol.11 , pp. 197-214
    • Hoyer, D.1    Schoeffter, P.2
  • 13
    • 0036267564 scopus 로고    scopus 로고
    • Pharmacological characterization of the 5-HT receptors mediating contraction and relaxation of canine isolated proximal stomach smooth muscle
    • Janssen, P., Prins, N.H., Meulemans, A.L. & Lefebvre, R.A. (2002). Pharmacological characterization of the 5-HT receptors mediating contraction and relaxation of canine isolated proximal stomach smooth muscle. Br. J. Pharmacol., 136, 321-329.
    • (2002) Br. J. Pharmacol. , vol.136 , pp. 321-329
    • Janssen, P.1    Prins, N.H.2    Meulemans, A.L.3    Lefebvre, R.A.4
  • 14
    • 0030854356 scopus 로고    scopus 로고
    • Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b)
    • Jasper, J.R., Kosaka, A., To, Z.P., Chang, D.J. & Eglen, R.M. (1997). Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b). Br. J. Pharmacol., 122, 126-132.
    • (1997) Br. J. Pharmacol. , vol.122 , pp. 126-132
    • Jasper, J.R.1    Kosaka, A.2    To, Z.P.3    Chang, D.J.4    Eglen, R.M.5
  • 15
    • 0026499745 scopus 로고
    • Investigation into the 5-hydroxytryptamine-induced relaxation of the circular smooth muscle of guinea-pig stomach fundus
    • Kojima, S., Ishizaki, R. & Shimo, Y. (1992). Investigation into the 5-hydroxytryptamine-induced relaxation of the circular smooth muscle of guinea-pig stomach fundus. Eur. J. Pharmacol., 224, 45-49.
    • (1992) Eur. J. Pharmacol. , vol.224 , pp. 45-49
    • Kojima, S.1    Ishizaki, R.2    Shimo, Y.3
  • 16
    • 0031984424 scopus 로고    scopus 로고
    • Effect of nitroglycerin and long-term electrical stimulation on nitrergic relaxation in the pig gastric fundus
    • Lefebvre, R.A. & Vandekerckhove, K. (1998). Effect of nitroglycerin and long-term electrical stimulation on nitrergic relaxation in the pig gastric fundus. Br. J. Pharmacol., 123, 143-149.
    • (1998) Br. J. Pharmacol. , vol.123 , pp. 143-149
    • Lefebvre, R.A.1    Vandekerckhove, K.2
  • 17
    • 0023879569 scopus 로고
    • The classification of 5-Hydroxytryptamine Receptors
    • Leff, P. & Martin, G.R. (1988). The classification of 5-Hydroxytryptamine Receptors. Med. Res. Rev., 8, 187-202.
    • (1988) Med. Res. Rev. , vol.8 , pp. 187-202
    • Leff, P.1    Martin, G.R.2
  • 18
    • 0027374438 scopus 로고
    • The role of nitric oxide (NO) in 5-HT-induced relaxations of the guinea-pig stomach
    • Meulemans, A.L., Helsen, L.F. & Schuurkes, J.A. (1993). The role of nitric oxide (NO) in 5-HT-induced relaxations of the guinea-pig stomach. Naunyn Schmiedebergs Arch. Pharmacol., 348, 424-430.
    • (1993) Naunyn Schmiedebergs Arch. Pharmacol. , vol.348 , pp. 424-430
    • Meulemans, A.L.1    Helsen, L.F.2    Schuurkes, J.A.3
  • 19
    • 0023081945 scopus 로고
    • The pig as a model for human nutrition
    • Miller, E.R. & Ullrey, D.E. (1987). The pig as a model for human nutrition. Annu. Rev. Nutr., 7, 361-382.
    • (1987) Annu. Rev. Nutr. , vol.7 , pp. 361-382
    • Miller, E.R.1    Ullrey, D.E.2
  • 20
    • 0030981178 scopus 로고    scopus 로고
    • Effect of a selective 5-HT3 receptor agonist on gastric motility in fasted and fed dogs
    • Nagakura, Y., Ito, H., Kamato, T., Nishida, A. & Miyata, K. (1997). Effect of a selective 5-HT3 receptor agonist on gastric motility in fasted and fed dogs. Eur. J. Pharmacol., 327, 189-193.
    • (1997) Eur. J. Pharmacol. , vol.327 , pp. 189-193
    • Nagakura, Y.1    Ito, H.2    Kamato, T.3    Nishida, A.4    Miyata, K.5
  • 21
    • 0035197085 scopus 로고    scopus 로고
    • Characterization of the receptors involved in the 5-HT-induced excitation of canine antral longitudinal muscle
    • Prins, N.H., Akkermans, L.M., Lefebvre, R.A. & Schuurkes, J.A. (2001a). Characterization of the receptors involved in the 5-HT-induced excitation of canine antral longitudinal muscle. Br. J. Pharmacol., 134, 1351-1359.
    • (2001) Br. J. Pharmacol. , vol.134 , pp. 1351-1359
    • Prins, N.H.1    Akkermans, L.M.2    Lefebvre, R.A.3    Schuurkes, J.A.4
  • 22
    • 0035041126 scopus 로고    scopus 로고
    • 5-HT4 receptors mediating enhancement of contractility in canine stomach; an in vitro and in vivo study
    • Prins, N.H., van der Grijn, A., Lefebvre, R.A., Akkermans, L.M.A. & Schuurkes, J.A.J. (2001b). 5-HT4 receptors mediating enhancement of contractility in canine stomach; an in vitro and in vivo study. Br. J. Pharmacol., 132, 1941-1947.
    • (2001) Br. J. Pharmacol. , vol.132 , pp. 1941-1947
    • Prins, N.H.1    Van der Grijn, A.2    Lefebvre, R.A.3    Akkermans, L.M.A.4    Schuurkes, J.A.J.5
  • 23
    • 0031039753 scopus 로고    scopus 로고
    • Characterization of the contraction to 5-HT in the canine colon longitudinal muscle
    • Prins, N.H., Briejer, M.R. & Schuurkes, J.A. (1997). Characterization of the contraction to 5-HT in the canine colon longitudinal muscle. Br. J. Pharmacol., 120, 714-720.
    • (1997) Br. J. Pharmacol. , vol.120 , pp. 714-720
    • Prins, N.H.1    Briejer, M.R.2    Schuurkes, J.A.3
  • 24
    • 0024587689 scopus 로고
    • Selective and functional 5-hydroxytryptamine 3 receptor antagonism by BRL 43694 (granisetron)
    • Sanger, G.J. & Nelson, D.R. (1989). Selective and functional 5-hydroxytryptamine 3 receptor antagonism by BRL 43694 (granisetron). Eur. J. Pharmacol., 159, 113-124.
    • (1989) Eur. J. Pharmacol. , vol.159 , pp. 113-124
    • Sanger, G.J.1    Nelson, D.R.2
  • 25
    • 0034070874 scopus 로고    scopus 로고
    • Influence of sumatriptan on gastric fundus tone and on the perception of gastric distension in man
    • Tack, J., Coulie, B., Wilmer, A., Andrioli, A. & Janssens, J. (2000). Influence of sumatriptan on gastric fundus tone and on the perception of gastric distension in man. Gut, 46, 468-473.
    • (2000) Gut , vol.46 , pp. 468-473
    • Tack, J.1    Coulie, B.2    Wilmer, A.3    Andrioli, A.4    Janssens, J.5
  • 26
    • 0033045313 scopus 로고    scopus 로고
    • Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach
    • Takemura, K., Takada, K., Mameya, S., Kaibara, M. & Taniyama, K. (1999). Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach. Jap. J. Pharm., 79, 41-49.
    • (1999) Jap. J. Pharm. , vol.79 , pp. 41-49
    • Takemura, K.1    Takada, K.2    Mameya, S.3    Kaibara, M.4    Taniyama, K.5
  • 27
    • 0029922424 scopus 로고    scopus 로고
    • GR127935 is a potent antagonist of the 5-HT1-like receptor mediating contraction in the canine coronary artery
    • Terron, J.A. (1996). GR127935 is a potent antagonist of the 5-HT1-like receptor mediating contraction in the canine coronary artery. Eur. J. Pharmacol., 300, 109-112.
    • (1996) Eur. J. Pharmacol. , vol.300 , pp. 109-112
    • Terron, J.A.1
  • 28
    • 0032993173 scopus 로고    scopus 로고
    • Pharmacological evidence for the 5-HT7 receptor mediating smooth muscle relaxation in canine cerebral arteries
    • Terron, J.A. & Falcon-Neri, A. (1999). Pharmacological evidence for the 5-HT7 receptor mediating smooth muscle relaxation in canine cerebral arteries. Br. J. Pharmacol., 127, 609-616.
    • (1999) Br. J. Pharmacol. , vol.127 , pp. 609-616
    • Terron, J.A.1    Falcon-Neri, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.