Immediate drug release from solid oral dosage forms

Journal of Pharmaceutical Sciences

Volumn 94, Issue 1, 2005, Pages 120-133

  Schreiner, Thomas ^a   Schaefer, Ulrich F ^a   Loth, Helmut ^a  

^a SAARLAND UNIVERSITY   (Germany)

Author keywords

Dissolution; Excipients; Formulation; Kinetics; Mathematical model; Unit operations

Indexed keywords

CELLULOSE; EXCIPIENT; KETOPROFEN; SOLVENT; STARCH;

ARTICLE; CHEMICAL MODIFICATION; COMPUTER PROGRAM; DRUG DOSAGE FORM; DRUG FORMULATION; DRUG GRANULATION; DRUG RELEASE; DRUG SOLUBILITY; IMMEDIATE DRUG RELEASE; MATHEMATICAL MODEL; ORAL DRUG ADMINISTRATION; POROSITY; STOCHASTIC MODEL; SURFACE PROPERTY; TABLET; TABLET DISINTEGRATION; WATER TRANSPORT; WETTABILITY;

EID: 12244270370     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/jps.20226     Document Type: Article

References (40)

1. Marrer S, Häusler H. 2002. Excipients' functionality impact on product quality and process performance. Pharm Ind 64:1083-1086.
2. Lippold BC, Ohm A. 1986. Correlation between wettability and dissolution rate of pharmaceutical powders. Int J Pharm 28:67-74.
3. Lerk CF, Bolhuis GK. 1977. Interaction of lubricants and colloidal silica during mixing with excipients. II. Its effect on wettability and dissolution velocity. Pharm Acta Helv 52:39-44.
4. Hersey JA, Krycer I. 1980. Biopharmaceutical implications of technological change. Int J Pharm Tech Prod Manuf 1:18-21.
5. Loth H, Schaefer U. 1985. Messungen der korngrößenabhä ngigen Lösungsgeschwindigkeiten schlecht benetzbarer Substanzen und ihre mathematische Auswertung. Act Pharm Technol 31:160-166.
6. Hemgesberg EM. 1986. Untersuchungen zum Benetzungs- und Auflösungsverhalten schlecht benetzbarer Arzneistoffe [PhD thesis]. Saarbruecken, Germany: Saarland University.
7. Ishizaka T, Honda H, Ikawa K, Kizu N, Yano K, Koishi M. 1988. Complexation of aspirin with potato starch and improvement of dissolution rate by dry mixing. Chem Pharm Bull 36:2562-2569.
8. Te Wierik GHP, Bolhuis GK, Zuurman K, Lerk CF. 1992. Improvement of dissolution of poorly soluble drugs by solid deposition on a super disintegrant. I. Physical mixtures. Acta Pharm Nord 4:239-244.
9. Liversidge GG. 1981. Ketoprofen. In: Florey K, editor. Analytical profiles of drug substances. Vol. 10. New York: Academic Press, pp 443-471.
10. Freundlich H, Enslin O, Lindau G. 1933. Über den Einfluß von Fremdstoffen auf die Flüssigkeitsaufnahme von nicht quellbaren Pulvern. Kolloid-Beihefte 37:242-280.
11. Enslin O. 1933. Über einen Apparat zur Messung der Flüssigkeitsaufnahme von quellbaren und porösen Stoffen und zur Charakterisierung der Benetzbarkeit. Die Chemische Fabrik 13:147-148.
12. Mühlemann H, Vegezzi G. 1954. Einfluß der Qualität von Bolus alba auf seine Verwendbarkeit als Grundlage für Umschlagspasten und als orales Adsorbens. Pharm Acta Helv 29:111-117.
13. USP 23. 1995. Dissolution, apparatus 2. Rockville, MD: United States Pharmacopeial Convention, pp 1791-1793.
14. Schittkowski K. 1988. Solving nonlinear least squares problems by a general purpose SQP-method. In: Hoffmann KH, Hiriart-Urruty JB, Lemarechal C, Zowe J, editors. Trends in mathematical optimization, International Series of Numerical Mathematics. Vol. 84. Basel: Birkhauser, pp 295-309.
15. Schittkowski K. 2002. EASY-FIT: A software system for data fitting in dynamic systems. Struct Multidisciplinary Optimization 23:153-169.
16. Schittkowski K. 2003. Numerical data fitting in dynamical systems. Dordrecht: Kluwer Academic Publishers.
17. Hairer E, Wanner G. 1991. Solving ordinary differential equations. II. Stiff and differential-algebraic problems. Series computational mathematics. Berlin: Springer.
18. Washburn EW. 1921. The dynamics of capillary flow. Phys Rev 17:273-283.
19. Allen T. 1975. Particle size measurement. 2nd ed. London: Chapman & Hall, p 180.
20. Cassie ABD. 1948. Contact angles. Discuss Faraday Soc 3:11-16.
21. Schreiner Th. 1995. Mechanistische und kinetische Parameter der Arzneistoffauflösung aus festen Zubereitungen als Kriterien der galenischen Qualitätssicherung [PhD thesis]. Saarhruecken, Germany: Saarland University.
22. Noyes AA, Whitney WR. 1897. The rate of solution of solid substances in their own solutions. J Am Chem Soc 19:930-934.
23. Nernst W. 1904. Theorie der Reaktionsgeschwindigkeit in heterogenen Systemen. Z Phys Chem 47:52-55.
24. Brunner E. 1904. Reaktionsgeschwindigkeit in heterogenen Systemen. Z Phys Chem 47:56-102.
25. Carstensen JT, Musa MN. 1972. Dissolution rate patterns of log-normally distributed powders. J Pharm Sci 61:223-227.
26. Brooke D. 1974. Dissolution profile of log-normal powders. II. Dissolution before critical time. J Pharm Sci 63:344-347.
27. Veng Pedersen P, Myrick JW. 1978. Versatile kinetic approach to analysis of dissolution data. J Pharm Sci 67:1450-1455.
28. Sunada H, Yamamoto A, Otsuka A, Yonezawa Y. 1988. Changes of surface area in the dissolution process of crystalline substances. Chem Pharm Bull 36:2557-2561.
29. Yonezawa Y, Shinohara I, Otsuka A, Sunada H. 1990. Dissolution and simulation curves for log-normal particle-size-distributed model systems. Chem Pharm Bull 38:3107-3111.
30. Leary JR, Ross SD. 1983. Mathematical expression of tablet dissolution profiles. Int J Pharm 17:193-201.
31. Kervinen L, Yliruusi J. 1993. Modelling S-shaped dissolution curves. Int J Pharm 92:115-122.
32. Costa FO, Sousa JJS, Pais AACC, Formosinho SJ. 2003. Comparison of dissolution profiles of ibuprofen pellets. J Control Release 89:199-212.
33. Dressman JB, Amidon GL, Reppas C, Shah VP. 1998. Dissolution testing as a prognostic tool for oral drug absorption: Immediate release dosage forms. Pharm Res 15:11-22.
34. Costa P, Lobo JMS. 2001. Modeling and comparison of dissolution profiles. Eur J Pharm Sci 13:123-133.
35. Dokoumetzidis A, Macheras P. 1997. A population growth model of dissolution. Pharm Res 14:1122-1126.
36. Elkoshi Z. 1997. On the variability of dissolution data. Pharm Res 14:1355-1362.
37. Lansky P, Weiss M. 2001. Modeling heterogeneity of particles and random effects in drug dissolution. Pharm Res 18:1061-1067.
38. Lansky P, Weiss M. 2003. Classification of dissolution profiles in terms of fractional dissolution rate and a novel measure of heterogeneity. J Pharm Sci 92:1632-1647.
39. Langenbucher F. 1972. Linearization of dissolution rate curves by the Weibull distribution. J Pharm Pharmacol 24:979-981.
40. Sachs L. 1997. Angewandte Statistik. 8th ed. Berlin: Springer, pp 174, 355.