Microwave-assisted synthesis of novel thiazolocarbozoles and evaluation as potential anticancer agents. Part III

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 19, Issue 6, 2004, Pages 467-473

  Testard, Alexandra ^a   Picot, Laurent ^a   Fruitier Arnaudin, Ingrid ^a   Piot, Jean Marie ^a   Chabane, Hadjila ^a   Domon, Lisianne ^a   Thiery, Valerie ^a   Besson, Thierry ^a  

^a FRE CNRS 2766   (France)

Author keywords

Appel salt; Carbazoles; Cytotoxic and antiproliferative activities; Imino 1,2,3 dithiazoles; Microwave chemistry; Thiazoles

Indexed keywords

(6 BROMO 1,4 DIMETHYL 9H CARBAZOL 3 YL) (4 CHLORO[1,2,3]DITHIAZOL 5 YLIDENE)AMINE; (6 CHLORO 1,4 DIMETHYL 9H CARBAZOL 3 YL) (4 CHLORO[1,2,3]DITHIAZOL 5 YLIDENE)AMINE; 2 (4,5 DIHYDRO 1H IMIDAZOL 2 YL) 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE; 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE 2 CARBONITRILE; 6 BROMO 2 (4,5 DIHYDRO 1H IMIDAZOL 2 YL) 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUOREN 6 OL; 6 BROMO 2 (4,5 DIHYDRO 1H IMIDAZOL 2 YL) 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE; 6 BROMO 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE 2 CARBONITRILE; 6 CHLORO 4,10 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE 2 CARBONITRILE; 9 ETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUORENE 2 CARBONITRILE; ANTINEOPLASTIC AGENT; CARBAZOLE DERIVATIVE; CYTOTOXIC AGENT; DERCITINE; ELLIPTICINE; ETHYL [2 CYANO 4,5 DIMETHYL 9H 1 THIA 3,9 DIAZACYCLOPENTA[B]FLUOREN 6 YL]CARBONATE; ETHYL [6 (4 CHLORO[1,2,3]DITHIAZOL 5 YLIDENEAMINO) 5,8 DIMETHYL 9H CARBAZOL 3 YL]; KUANONIAMINE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; BREAST CARCINOMA; CANCER CELL CULTURE; CANCER INHIBITION; CELL VIABILITY; CHEMICAL PROCEDURES; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; MICROWAVE RADIATION; PRIORITY JOURNAL;

ANTINEOPLASTIC AGENTS; CARBAZOLES; CELL LINE; CELL LINE, TUMOR; CELL PROLIFERATION; CELL SURVIVAL; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; MICROWAVES; MOLECULAR STRUCTURE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 11244286080     PISSN: 14756366     EISSN: None     Source Type: Journal    
DOI: 10.1080/14756360412331280491     Document Type: Article

References (13)

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