Synthesis and radioiodination of some daunorubicin and doxorubicin derivatives

Carbohydrate Research

Volumn 340, Issue 1, 2005, Pages 15-24

  Ghirmai, Senait ^a   Mume, Eskender ^a   Tolmachev, Vladimir ^a,b   Sjöberg, Stefan ^a  

^a UPPSALA UNIVERSITY   (Sweden)

^b UPPSALA UNIVERSITY   (Sweden)

Author keywords

125I; Chloramine T; Daunorubicin; Doxorubicin; Radioiodination

Indexed keywords

AUGER ELECTRON EMITTERS; CLINICAL EFFICACY; DAUNORUBICIN; DOXORUBICIN; RADIOIODINATION;

ALDEHYDES; AMINATION; AMINES; AROMATIC COMPOUNDS; CARBOXYLIC ACIDS; CELLS; DERIVATIVES; DRUG PRODUCTS; ESTERIFICATION; ESTERS; TOXICITY; TUMORS;

SYNTHESIS (CHEMICAL);

ALDEHYDE; AMIDE; AMINE; BENZOIC ACID; BENZOIC ACID DERIVATIVE; DAUNORUBICIN DERIVATIVE; DOXORUBICIN DERIVATIVE; ESTER DERIVATIVE; IODINE 125; NICOTINIC ACID; OXIDIZING AGENT; PHENYL GROUP; POTASSIUM SALT; TOSYLCHLORAMIDE SODIUM;

AMINATION; ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ESTERIFICATION; ISOTOPE LABELING; PRIORITY JOURNAL; RADIOCHEMISTRY; RADIOIODINATION;

CHROMATOGRAPHY, THIN LAYER; DAUNORUBICIN; DOXORUBICIN; IODINE RADIOISOTOPES; MOLECULAR STRUCTURE;

EID: 11144322752     PISSN: 00086215     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.carres.2004.10.014     Document Type: Article

References (19)

1. T. Woodcock, J. Allegro, and S. Richman Semin. Oncol. 11 1984 28 32
2. D. Von Hoff Semin. Oncol. 11 1984 23 27
3. J.W. Lown J. Med. Chem. 29 1986 2235 2241
4. M. Berettoni, A. Cipollone, L. Olivieri, D. Palomba, F. Arcamone, A. Maggi, and F. Animati Tetrahedron Lett. 43 2002 2867 2871
5. Y.S. Rho, W. Kim, S. Park, D.J. Yoo, H. Kang, and S. Chung Bull. Korean Chem. Soc. 22 2001 581 586
6. K. Ok, Y. Takagi, T. Tsuchiya, S. Umezawa, and H. Umezawa Carbohydr. Res. 169 1987 69 81
7. Y.S. Rho, G. Kim, W. Kim, S. Park, D.J. Yoo, H. Kang, and S. Chung Bull. Korean Chem. Soc. 22 2001 587 592
8. F. Arcamone, G. Franceschi, A. Minghetti, S. Penco, and S. Redaelli J. Med. Chem. 17 1974 335 337
9. R. Seshadri, M. Israel, and W.J. Pegg J. Med. Chem. 26 1983 11 15
10. R. Seshadri, J.M. Idriss, and M. Israel J. Med. Chem. 29 1986 1269 1273 and references cited therein
11. D. Murali, and O.T. DeJesus Bioorg. Med. Chem. Lett. 8 1998 3419 3422 and references cited therein
12. J.W. Lown Chem. Soc. Rev. 1992 165 176
13. R.G.G. Leenders, and H.W. Scheeren Bioorg. Med. Chem. Lett. 5 24 1995 2975 2980
14. J. Carlsson, E.B. Kullberg, J. Capala, S. Sjöberg, K. Edwards, and L. Gedda J. Neuro-Oncol. 62 2003 47 59
15. Y.S. Rho, S. Park, W. Kim, G. Kim, D.J. Yoo, H. Kang, and S. Chung Synth. Commun. 32 2002 1961 1975
16. J. Koziorowski, C. Henssen, and R. Weinreich Appl. Radiat. Isot. 49 1998 955 959
17. S. Garg, P.K. Garg, and M.R. Zalutsky Bioconj. Chem. 2 1991 50 56
18. A.R. Hajpour, M. Arbabian, and A.E. Ruoho J. Org. Chem. 67 2002 8622 8624
19. D.D. Perrin, and W.L.F. Armarego Purification of Laboratory Chemicals 3rd ed. 1988 Pergamon