메뉴 건너뛰기




Volumn 42, Issue 4-5, 2004, Pages 367-373

Synthesis, analysis and biological evaluation of novel steroidal estrogenic prodrugs for the treatment of breast cancer

Author keywords

Breast cancer; Cancer chemotherapy; Doxorubicin; Drug targeting; Estrogen receptor; Estrogenic prodrugs; K562; MCF 7; MCF 7ADR; MT 1; Spacer group; Steroids

Indexed keywords

17 AMINOXYESTRONE DOXORUBICIN PRODRUG; 3 ESTRONE DODECANEDIOYL ESTER DOXORUBICIN PRODRUG; DOXORUBICIN; DOXORUBICIN DODECANEDIOYL ESTER; ESTROGEN RECEPTOR; ESTRONE 17 AMINODODECANE DOXORUBICIN PRODRUG; ESTRONE ADIPOYL ESTER DOXORUBICIN PRODRUG; PRODRUG; UNCLASSIFIED DRUG;

EID: 10344250434     PISSN: 13880209     EISSN: None     Source Type: Journal    
DOI: 10.1080/13880200490519686     Document Type: Article
Times cited : (7)

References (15)
  • 2
    • 0025869917 scopus 로고
    • Prospects for the chemoprevention of breast cancer
    • Baum M, Ziv Y, Colletta A (1991): Prospects for the chemoprevention of breast cancer. Br Med Bull 47: 493-503.
    • (1991) Br Med Bull , vol.47 , pp. 493-503
    • Baum, M.1    Ziv, Y.2    Colletta, A.3
  • 3
    • 0024343537 scopus 로고
    • Doxorubicin-effect of different schedules on toxicity and anti-tumor efficacy
    • Bielack SS, Erttmann R, Winkler K, Landbeck G (1989): Doxorubicin-effect of different schedules on toxicity and anti-tumor efficacy. Eur J Cancer Clin Oncol 25: 873-882.
    • (1989) Eur J Cancer Clin Oncol , vol.25 , pp. 873-882
    • Bielack, S.S.1    Erttmann, R.2    Winkler, K.3    Landbeck, G.4
  • 4
    • 0003882361 scopus 로고
    • London, Jones and Bartlett Publishers International
    • Cooper GM (1992): Elements of Human Cancer. London, Jones and Bartlett Publishers International, pp. 4-61.
    • (1992) Elements of Human Cancer , pp. 4-61
    • Cooper, G.M.1
  • 6
    • 0027483443 scopus 로고
    • High dose, dose-intensive chemotherapy with doxorubicin and cyclophosphamide for the treatment of advanced breast cancer
    • Ferguson JE, Dodwell DJ, Seymoure AM, Richards MA, Howell A (1993): High dose, dose-intensive chemotherapy with doxorubicin and cyclophosphamide for the treatment of advanced breast cancer. Br J Cancer 67: 825-829.
    • (1993) Br J Cancer , vol.67 , pp. 825-829
    • Ferguson, J.E.1    Dodwell, D.J.2    Seymoure, A.M.3    Richards, M.A.4    Howell, A.5
  • 7
    • 84970050234 scopus 로고
    • Establishment and characterisation of three new human breast cancer cell lines for anticancer drug evaluation in vitro
    • Hambly RJ, Bibby MC, Double JA (1994): Establishment and characterisation of three new human breast cancer cell lines for anticancer drug evaluation in vitro. Br J Cancer 69(Supp. 21): 31.
    • (1994) Br J Cancer , vol.69 , Issue.SUPPL. 21 , pp. 31
    • Hambly, R.J.1    Bibby, M.C.2    Double, J.A.3
  • 8
    • 10344226996 scopus 로고    scopus 로고
    • (1988): United Kingdom Patent GB 2201419 A (Application Number 8704236)
    • Hartman NG, Angelucci F, Suarato A (1988): United Kingdom Patent GB 2201419 A (Application Number 8704236).
    • Hartman, N.G.1    Angelucci, F.2    Suarato, A.3
  • 9
    • 0024426375 scopus 로고
    • The MTT assay underestimates the growth inhibitory effects of Interferon
    • Jabbar SAB, Twentyman PR, Watson JV (1989): The MTT assay underestimates the growth inhibitory effects of Interferon. Br J Cancer 60: 523-528.
    • (1989) Br J Cancer , vol.60 , pp. 523-528
    • Jabbar, S.A.B.1    Twentyman, P.R.2    Watson, J.V.3
  • 10
    • 0028788985 scopus 로고
    • Gynecological effects of tamoxifen
    • Kuo DYS, Runowicz CD (1995): Gynecological effects of tamoxifen. Med Oncol 12: 87-94.
    • (1995) Med Oncol , vol.12 , pp. 87-94
    • Kuo, D.Y.S.1    Runowicz, C.D.2
  • 11
    • 84986725681 scopus 로고
    • Cell uptake and estrogen receptor binding affinities of novel triphenylethylene compounds
    • Manns JE, Double JA, Brown JE (1993): Cell uptake and estrogen receptor binding affinities of novel triphenylethylene compounds. J Pharm Pharmacol 45: 1127.
    • (1993) J Pharm Pharmacol , vol.45 , pp. 1127
    • Manns, J.E.1    Double, J.A.2    Brown, J.E.3
  • 12
    • 0019287522 scopus 로고
    • Amino acid and dipeptide derivatives of daunorubicin. 1. Synthesis, physicochemical properties, and lysosomal digestion
    • Masquelier M, Baurain R, Trouet A (1980): Amino acid and dipeptide derivatives of daunorubicin. 1. Synthesis, physicochemical properties, and lysosomal digestion. J Med Chem 23: 1166-1170.
    • (1980) J Med Chem , vol.23 , pp. 1166-1170
    • Masquelier, M.1    Baurain, R.2    Trouet, A.3
  • 13
    • 0021958425 scopus 로고
    • Effect of estrogens and antiestrogens on growth of human breast cancer cells in athymic nude mice
    • Osborne CK, Hobbs K, Clark GM (1995): Effect of estrogens and antiestrogens on growth of human breast cancer cells in athymic nude mice. Cancer Res 45: 584-590.
    • (1995) Cancer Res , vol.45 , pp. 584-590
    • Osborne, C.K.1    Hobbs, K.2    Clark, G.M.3
  • 14
    • 0027259151 scopus 로고
    • Multidrug-resistance mediated by P-glycoprotein in hematological malignancies
    • Pasman PC, Schouten HC (1993): Multidrug-resistance mediated by P-glycoprotein in hematological malignancies. Netherlands J. Med 42: 218-231.
    • (1993) Netherlands J Med , vol.42 , pp. 218-231
    • Pasman, P.C.1    Schouten, H.C.2
  • 15
    • 0021348486 scopus 로고
    • Steroid-hormone receptors in breast cancer
    • Wittliff JL (1984): Steroid-hormone receptors in breast cancer. Cancer 53: 630-643.
    • (1984) Cancer , vol.53 , pp. 630-643
    • Wittliff, J.L.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.