A novel synthetic inhibitor of endopeptidase-24.15

Journal of Enzyme Inhibition

Volumn 11, Issue 1, 1996, Pages 39-49

  Ukai, Yuko ^a   Li, Qiulin ^a   Ito, Susumu ^a   Mita, Shiro ^a  

^a SANTEN PHARMACEUTICAL CO LTD   (Japan)

Author keywords

Endopeptidase 24.15; Inhibition; Metalloendopeptidase; SA898

Indexed keywords

DIPEPTIDYL CARBOXYPEPTIDASE; MEMBRANE METALLOENDOPEPTIDASE; PROTEINASE; PROTEINASE INHIBITOR; SA 898; THIMET OLIGOPEPTIDASE; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG STRUCTURE; ENZYME INHIBITION; INHIBITION KINETICS; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEINASE INHIBITION; RAT; REACTION ANALYSIS;

EID: 10244247859     PISSN: 87555093     EISSN: None     Source Type: Journal    
DOI: 10.3109/14756369609038221     Document Type: Article

References (14)

1. Schwartz, J.-C., Malftoy, B. and La Baume, S.D. (1981). Life Sci., 29, 1715-1740.
2. Black, R.A., Kronheim, S.R., Cantrell, M., Deeley, M.C., March, C.J., Prickett, K.S., Wignall, J., Conlon, P.J., Cosman, D., Hopp, T.P. and Mochizuki, D.Y. (1988). J. Biol. Chem., 263, 9437-9442.
3. Orlowski, M., Michaud, C. and Chu, T.G. (1983). Eur. J. Biochem., 135, 81-88.
4. Chu, T.G. and Orlowski, M. (1985). Endocrinology, 116, 1418-1425.
5. Orlowski, M., Reznik, S., Alaya, J. and Pierotti, A.R, (1989). Biochem. J., 261, 951-958.
6. Orlowski, M., Michaud, C. and Molineaux, C.J. (1988) Biochemistry, 27, 597-602.
7. Malfroy, B. and Schwartz, J.-C. (1984). J. Biol. Chem., 259, 14365-14370.
8. Oya, M., Kato, E., Iwao, J. and Yasuoka, N. (1982). Chem. Pharm. Bull., 30, 484-493.
9. Bratton, A.C. and Marshall, E.K., Jr. (1939). J. Biol. Chem., 128, 537-550.
10. Horiuchi, M., Fujimura, K., Terashima, T. and Iso, T. (1982). J. Chromatogr., 233, 123-130.
11. Orlowski, M. and Wilk, S. (1981). Biochemistry. 20, 4942-4950.
12. Barrett, A.J. (1972). Anal. Biochem., 47, 280-293.
13. Almenoff, J. and Orlowski, M. (1983). Biochemistry. 22, 590-599.
14. Malineaux, C.J., Lasdon, A., Michaud, C. and Orlowski, M. (1988). J. Neurochem. 51, 624-633.