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Volumn 37, Issue 7, 1996, Pages 1207-1214

Iodine-123-5-iodo-6-nitroquipazine: SPECT radiotracer to image the serotonin transporter

Author keywords

iodine 123 5 iodo 6 nitroquipazine; serotonin transporter

Indexed keywords

3,4 METHYLENEDIOXYMETHAMPHETAMINE; 5 IODO 6 NITROQUIPAZINE I 123; 5 IODO 6 NITROQUIPAZINE I 125; NEUROTOXIN; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

EID: 10144229103     PISSN: 01615505     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (58)

References (40)
  • 1
    • 0023234129 scopus 로고
    • Aminergic systems in Alzheimer's disease and Parkinson's disease
    • D'Amato RJ, Zweig RM, Whitehouse PJ, et al. Aminergic systems in Alzheimer's disease and Parkinson's disease. Ann Neurol 1987;22:229-236.
    • (1987) Ann Neurol , vol.22 , pp. 229-236
    • D'Amato, R.J.1    Zweig, R.M.2    Whitehouse, P.J.3
  • 2
    • 84950170900 scopus 로고
    • Neuropathology of immunohistochemically identified brainstem neurons in Parkinson's disease
    • Halliday GM, Li YW, Blumbergs PC, et al. Neuropathology of immunohistochemically identified brainstem neurons in Parkinson's disease. Ann Neurol 1990;27:373-385.
    • (1990) Ann Neurol , vol.27 , pp. 373-385
    • Halliday, G.M.1    Li, Y.W.2    Blumbergs, P.C.3
  • 3
    • 0021357276 scopus 로고
    • Altered serotonin metabolism in depressed patients with Parkinson's disease
    • Mayeux R, Stern Y, Cote L, Williams JBW. Altered serotonin metabolism in depressed patients with Parkinson's disease. Neurology 1984;34:642-646.
    • (1984) Neurology , vol.34 , pp. 642-646
    • Mayeux, R.1    Stern, Y.2    Cote, L.3    Williams, J.B.W.4
  • 4
    • 0025782754 scopus 로고
    • Neuropathologic and neurochemical correlates of psychosis in primary dementia
    • Zubenko GS, Moossy J, Martinez AJ, et al. Neuropathologic and neurochemical correlates of psychosis in primary dementia. Arch Neurol 1991;48:619-624.
    • (1991) Arch Neurol , vol.48 , pp. 619-624
    • Zubenko, G.S.1    Moossy, J.2    Martinez, A.J.3
  • 6
    • 0015842566 scopus 로고
    • Selective accumulation of 3H-serotonin by nerve terminals of raphe neurones: An autoradiographic study
    • Kuhar MJ, Aghajanian GK. Selective accumulation of 3H-serotonin by nerve terminals of raphe neurones: an autoradiographic study. Nature 1973;241:187-189.
    • (1973) Nature , vol.241 , pp. 187-189
    • Kuhar, M.J.1    Aghajanian, G.K.2
  • 7
    • 0015320153 scopus 로고
    • Synaptosomes from forebrains of rats with midbrain raphe lesions: Selective reduction of serotonin uptake
    • Kuhar MJ, Roth RH, Aghajanian GK. Synaptosomes from forebrains of rats with midbrain raphe lesions: selective reduction of serotonin uptake. J Pharmacol Exp Ther 1972;181:36-45.
    • (1972) J Pharmacol Exp Ther , vol.181 , pp. 36-45
    • Kuhar, M.J.1    Roth, R.H.2    Aghajanian, G.K.3
  • 8
    • 0015510739 scopus 로고
    • Tryptophan hydroxylase activity and synaptosomal uptake of serotonin in discrete brain regions after midbrain raphe lesion: Correlation with serotonin levels and histochemical fluorescence
    • Kuhar MJ, Aghajanian GK, Roth RH. Tryptophan hydroxylase activity and synaptosomal uptake of serotonin in discrete brain regions after midbrain raphe lesion: correlation with serotonin levels and histochemical fluorescence. Brain Res 1972;44: 165-176.
    • (1972) Brain Res , vol.44 , pp. 165-176
    • Kuhar, M.J.1    Aghajanian, G.K.2    Roth, R.H.3
  • 9
    • 0027390785 scopus 로고
    • A PET radiotracer for studying serotonin uptake sites: Carbon-11-McN-5652Z
    • Suehiro M, Scheffel U, Dannals RF, et al. A PET radiotracer for studying serotonin uptake sites: carbon-11-McN-5652Z. J Nucl Med 1993;34:120-127.
    • (1993) J Nucl Med , vol.34 , pp. 120-127
    • Suehiro, M.1    Scheffel, U.2    Dannals, R.F.3
  • 10
    • 0025180948 scopus 로고
    • Paroxetine as an in vivo indicator of 3,4-methyl-enedioxymethamphetamine neurotoxicity: A presynaptic serotonergic positron emission tomography ligand?
    • Scheffel U, Ricaurte GA. Paroxetine as an in vivo indicator of 3,4-methyl-enedioxymethamphetamine neurotoxicity: a presynaptic serotonergic positron emission tomography ligand? Brain Res 1990;527:89-95.
    • (1990) Brain Res , vol.527 , pp. 89-95
    • Scheffel, U.1    Ricaurte, G.A.2
  • 11
    • 10144242797 scopus 로고
    • Radioiodinated analogs of fluoxetine: Potential agents for imaging serotonin reuptake sites with SPECT
    • Kung MP, Chumpradit S, Panyachotipun C, et al. Radioiodinated analogs of fluoxetine: potential agents for imaging serotonin reuptake sites with SPECT. J Nucl Med 1991;32:964.
    • (1991) J Nucl Med , vol.32 , pp. 964
    • Kung, M.P.1    Chumpradit, S.2    Panyachotipun, C.3
  • 12
    • 0026478714 scopus 로고
    • Iodinated tomoxetine derivatives as selective ligands for serotonin and norepinephrine uptake sites
    • Chumpradit S, Kung MP, Panyachotipun C, et al. Iodinated tomoxetine derivatives as selective ligands for serotonin and norepinephrine uptake sites. J Med Chem 1992;35: 4492-4497.
    • (1992) J Med Chem , vol.35 , pp. 4492-4497
    • Chumpradit, S.1    Kung, M.P.2    Panyachotipun, C.3
  • 13
    • 0028063106 scopus 로고
    • Validation of the transporter ligand cyanoimipramine as a marker of serotonin innervation density in brain
    • Soucy JP, Lafaille F, Lemoine P, et al. Validation of the transporter ligand cyanoimipramine as a marker of serotonin innervation density in brain. J Nucl Med 1994;35: 1822-1830.
    • (1994) J Nucl Med , vol.35 , pp. 1822-1830
    • Soucy, J.P.1    Lafaille, F.2    Lemoine, P.3
  • 14
    • 0028178856 scopus 로고
    • PET study of [11C]beta-CIT binding to monoamine transporters in the monkey and human brain
    • Farde L, Halldin C, Muller L, et al. PET study of [11C]beta-CIT binding to monoamine transporters in the monkey and human brain. Synapse 1994;16:93-103.
    • (1994) Synapse , vol.16 , pp. 93-103
    • Farde, L.1    Halldin, C.2    Muller, L.3
  • 15
    • 44049119282 scopus 로고
    • Synthesis and biodistribution of a new radiotracer for in vivo labeling of serotonin uptake sites by PET, cis-N,N-[11C]dimethyl-3-(2′,4′-dichlorophenyl)-indanamine (cis-[11C]DDP1)
    • Suehiro M, Scheffel U, Dannals RF, et al. Synthesis and biodistribution of a new radiotracer for in vivo labeling of serotonin uptake sites by PET, cis-N,N-[11C]dimethyl-3-(2′,4′-dichlorophenyl)-indanamine (cis-[11C]DDP1). Nucl Med Biol 1992;19: 549-553.
    • (1992) Nucl Med Biol , vol.19 , pp. 549-553
    • Suehiro, M.1    Scheffel, U.2    Dannals, R.F.3
  • 16
    • 0027168674 scopus 로고
    • Evaluation of the monoamine uptake site ligand [123I]methyl 3beta-(4-iodophenyl)-tropane-2 beta-carboxylate ([123I]beta-CIT) in non-human primates: Pharmacokinetics, biodistribution and SPECT brain imaging coregistered with MRI
    • Baldwin RM, Zea-Ponce Y, Zoghbi SS, et al. Evaluation of the monoamine uptake site ligand [123I]methyl 3beta-(4-iodophenyl)-tropane-2 beta-carboxylate ([123I]beta-CIT) in non-human primates: pharmacokinetics, biodistribution and SPECT brain imaging coregistered with MRI. Nucl Med Biol 1993;20:597-606.
    • (1993) Nucl Med Biol , vol.20 , pp. 597-606
    • Baldwin, R.M.1    Zea-Ponce, Y.2    Zoghbi, S.S.3
  • 17
    • 0026753156 scopus 로고
    • 4-Iodotomoxetine: A novel ligand for serotonin uptake sites
    • Kung MP, Chumpradit S, Billings J, Kung H. 4-Iodotomoxetine: a novel ligand for serotonin uptake sites. Life Sci 1992;51:95-106.
    • (1992) Life Sci , vol.51 , pp. 95-106
    • Kung, M.P.1    Chumpradit, S.2    Billings, J.3    Kung, H.4
  • 19
    • 0026612598 scopus 로고
    • 125I]5-iodo-6-nitro-2-piperazinylquinoline - A potent and selective ligand for the serotonin uptake complex
    • 125I]5-iodo-6-nitro-2-piperazinylquinoline - a potent and selective ligand for the serotonin uptake complex. Eur J Pharmacol 1992;210:103-104.
    • (1992) Eur J Pharmacol , vol.210 , pp. 103-104
    • Mathis, C.A.1    Biegon, A.2    Taylor, S.E.3
  • 20
    • 0027337038 scopus 로고
    • 125I]5-iodo-6-nitroquipazine: A potent and selective ligand for the 5-hydroxytryptamine uptake complex I. in vitro studies
    • 125I]5-iodo-6-nitroquipazine: a potent and selective ligand for the 5-hydroxytryptamine uptake complex I. In vitro studies. Brain Res 1993;619:229-235.
    • (1993) Brain Res , vol.619 , pp. 229-235
    • Mathis, C.A.1    Taylor, S.E.2    Biegon, A.3    Enas, J.D.4
  • 21
    • 0027337040 scopus 로고
    • 125I]5-Iodo-6-nitroquipazine: A potent and selective ligand for the 5-hydroxytryptamine uptake complex II. in vivo studies in rats
    • 125I]5-Iodo-6-nitroquipazine: a potent and selective ligand for the 5-hydroxytryptamine uptake complex II. In vivo studies in rats Brain Res 1993;619:236-246
    • (1993) Brain Res , vol.619 , pp. 236-246
    • Biegon, A.1    Mathis, C.A.2    Hanrahan, S.M.3    Jagust, W.J.4
  • 23
    • 0025921971 scopus 로고
    • Synthesis and resolution of (±)-7-chloro-8-hydroxy-1-(3′-iodophenyl)-3-methyl-2,3,4,5- tetrahydro-1H-3-benzazepine (TISCH): A high affinity and selective iodinated ligand for CNS D1 dopamine receptor
    • Chumpradit S, Kung M-P, Billings JJ, Kung HF. Synthesis and resolution of (±)-7-chloro-8-hydroxy-1-(3′-iodophenyl)-3-methyl-2,3,4,5- tetrahydro-1H-3-benzazepine (TISCH): a high affinity and selective iodinated ligand for CNS D1 dopamine receptor. J Med Chem 1991;34:877.
    • (1991) J Med Chem , vol.34 , pp. 877
    • Chumpradit, S.1    Kung, M.-P.2    Billings, J.J.3    Kung, H.F.4
  • 24
    • 0025318248 scopus 로고
    • Inhibition of neuronal 5-HT uptake by ketamine, but not halothane, involves disruption of substrate recognition by the transporter
    • Martin DC, Introna RP, Aronstam RS. Inhibition of neuronal 5-HT uptake by ketamine, but not halothane, involves disruption of substrate recognition by the transporter. Neurosci Lett 1990;112:99-103.
    • (1990) Neurosci Lett , vol.112 , pp. 99-103
    • Martin, D.C.1    Introna, R.P.2    Aronstam, R.S.3
  • 27
    • 0026515597 scopus 로고
    • Structure and function of the brain serotonin system
    • Jacobs BL, Azmitia EC. Structure and function of the brain serotonin system. Physiol Rev 1992;72:165-229.
    • (1992) Physiol Rev , vol.72 , pp. 165-229
    • Jacobs, B.L.1    Azmitia, E.C.2
  • 29
    • 0020054344 scopus 로고
    • Noradrenergic and serotonergic fibers innervate complementary layers in monkey primary visual cortex: An immunohistochemical study
    • Morrison JH, Foote SL, Molliver ME, et al. Noradrenergic and serotonergic fibers innervate complementary layers in monkey primary visual cortex: an immunohistochemical study. Proc Natl Acad Sci 1982;79:2401-2405.
    • (1982) Proc Natl Acad Sci , vol.79 , pp. 2401-2405
    • Morrison, J.H.1    Foote, S.L.2    Molliver, M.E.3
  • 30
    • 0025936538 scopus 로고
    • Serotonergic innervation of the thalamus in the primate: An immunohistochemical study
    • Lavoie B, Parent A. Serotonergic innervation of the thalamus in the primate: an immunohistochemical study. J Comp Neurol 1991;312:1-18.
    • (1991) J Comp Neurol , vol.312 , pp. 1-18
    • Lavoie, B.1    Parent, A.2
  • 31
    • 0022584974 scopus 로고
    • The primate serotonergic system: A review of human and animal studies and a report on macaca fascicularis
    • Fahn S, ed. New York, NY: Raven Press
    • Azmitia EC, Gannon PJ. The primate serotonergic system: a review of human and animal studies and a report on macaca fascicularis. In: Fahn S, ed. Advances in neurology, vol. 43: myoclonus. New York, NY: Raven Press; 1986:407-468.
    • (1986) Advances in Neurology, Vol. 43: Myoclonus , vol.43 , pp. 407-468
    • Azmitia, E.C.1    Gannon, P.J.2
  • 32
    • 0023902232 scopus 로고
    • Toxic effects of MDMA on central serotonergic neurons in the primate: Importance of route and frequency of drug administration
    • Ricaurte GA, DeLanney LE, Irwin I, Langston JW. Toxic effects of MDMA on central serotonergic neurons in the primate: importance of route and frequency of drug administration. Brain Res 1988;446:165-168.
    • (1988) Brain Res , vol.446 , pp. 165-168
    • Ricaurte, G.A.1    DeLanney, L.E.2    Irwin, I.3    Langston, J.W.4
  • 33
    • 0026612759 scopus 로고
    • Lasting effects of (±)-3,4-methylenedioxymethamphetamine (MDMA) on central serotonergic neurons in nonhuman primates: Neurochemical observations
    • Ricaurte GA, Martello AL, Katz JL, Martello MB. Lasting effects of (±)-3,4-methylenedioxymethamphetamine (MDMA) on central serotonergic neurons in nonhuman primates: neurochemical observations. J Pharm Exp Ther 1992;261:616-622.
    • (1992) J Pharm Exp Ther , vol.261 , pp. 616-622
    • Ricaurte, G.A.1    Martello, A.L.2    Katz, J.L.3    Martello, M.B.4
  • 34
    • 0024541227 scopus 로고
    • Distinct morphologic classes of serotonergic axons in primates exhibit differential vulnerability to the psychotropic drug 3,4-methylenedioxymethamphetamine
    • Wilson MA, Ricaurte GA, Molliver ME. Distinct morphologic classes of serotonergic axons in primates exhibit differential vulnerability to the psychotropic drug 3,4-methylenedioxymethamphetamine. Neuroscience 1989;28:121-137.
    • (1989) Neuroscience , vol.28 , pp. 121-137
    • Wilson, M.A.1    Ricaurte, G.A.2    Molliver, M.E.3
  • 35
    • 0027157108 scopus 로고
    • Oral administration of 3,4-methylenedioxymethamphetamine (MDMA) produces selective serotonergic depletion in the nonhuman primate
    • Ali SF, Newport GD, Scallet AC, et al. Oral administration of 3,4-methylenedioxymethamphetamine (MDMA) produces selective serotonergic depletion in the nonhuman primate. Neurotoxicol Teratol 1993;15:91-96.
    • (1993) Neurotoxicol Teratol , vol.15 , pp. 91-96
    • Ali, S.F.1    Newport, G.D.2    Scallet, A.C.3
  • 37
    • 0026616797 scopus 로고
    • In vivo binding of [125I]RTI-55 to dopamine transporters: Pharmacology and regional distribution with autoradiography
    • Cline EJ, Scheffel U, Boja JW, et al. In vivo binding of [125I]RTI-55 to dopamine transporters: pharmacology and regional distribution with autoradiography. Synapse 1992;12:37-46.
    • (1992) Synapse , vol.12 , pp. 37-46
    • Cline, E.J.1    Scheffel, U.2    Boja, J.W.3
  • 39
    • 0027131948 scopus 로고
    • Single photon emission computed tomographic imaging demonstrates loss of striatal dopamine transporters in Parkinson's disease
    • Innis RB, Seibyl JP, Scanley BE, et al. Single photon emission computed tomographic imaging demonstrates loss of striatal dopamine transporters in Parkinson's disease. Proc Nat Acad Sci 1993;90:11965-11969.
    • (1993) Proc Nat Acad Sci , vol.90 , pp. 11965-11969
    • Innis, R.B.1    Seibyl, J.P.2    Scanley, B.E.3
  • 40
    • 17144434961 scopus 로고
    • 123I]beta-CIT: Pharmacological characterization of brain uptake in nonhuman primates
    • 123I]beta-CIT: pharmacological characterization of brain uptake in nonhuman primates. Synapse 1993;13:295-309.
    • (1993) Synapse , vol.13 , pp. 295-309
    • Laruelle, M.1    Baldwin, R.M.2    Malison, R.T.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.