A novel nonpeptide antagonist of the kinin B1 receptor: Effects at the rabbit receptor

Journal of Pharmacology and Experimental Therapeutics

Volumn 311, Issue 3, 2004, Pages 1121-1130

  Morissette, Guillaume ^a   Fortin, Jean Philippe ^a   Otis, Sophie ^a   Bouthillier, Johanne ^a   Marceau, François ^a,b  

^a Université Laval   (Canada)

^b LAVAL UNIVERSITY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

2 [1 [(3,4 DICHLOROPHENYL)SULFONYL] 3 OXO 1,2,3,4 TETRAHYDROQUINOXALIN 2 YL] N [2 [4 (4,5 DIHYDRO 1H IMIDAZOL 2 YL)PHENYL]ETHYL]ACETAMIDE; ANGIOTENSIN; ANTIINFLAMMATORY AGENT; BRADYKININ; G PROTEIN COUPLED RECEPTOR; HISTAMINE; HYBRID PROTEIN; KININ B1 RECEPTOR; MITOGEN ACTIVATED PROTEIN KINASE 1; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; AORTA CONSTRICTION; AORTA MEDIA; ARTICLE; CELL STRAIN COS1; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; EMBRYO; ENZYME PHOSPHORYLATION; HUMAN; HUMAN CELL; INFLAMMATION; JUGULAR VEIN; MESENTERIC ARTERY; NONHUMAN; PAIN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN TRANSPORT; RABBIT; RAT; SEPSIS;

ANIMALS; AORTA, THORACIC; BLOTTING, WESTERN; CELL LINE; CERCOPITHECUS AETHIOPS; COS CELLS; EPITOPES; GENES, MYC; IMAGE CYTOMETRY; MICROSCOPY, CONFOCAL; MUSCLE CONTRACTION; MUSCLE, SMOOTH, VASCULAR; PROTEIN FOLDING; QUINOXALINES; RABBITS; RECEPTOR, BRADYKININ B1; RECEPTORS, CELL SURFACE; RECEPTORS, G-PROTEIN-COUPLED; SULFONES;

EID: 10044280370     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.104.071266     Document Type: Article

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