Stereoselective synthesis of (±)-rocaglaol analogues

Organic Letters

Volumn 6, Issue 24, 2004, Pages 4595-4597

  Thede, Kai ^a   Diedrichs, Nicole ^a   Ragot, Jacques P ^a  

^a BAYER PHARMA AG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOFURAN DERIVATIVE; CYCLOPENTA[B]BENZOFURAN; CYCLOPENTANE DERIVATIVE; ROCAGLAOL DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DERIVATIZATION; DRUG SYNTHESIS; ENANTIOSELECTIVITY; MOLECULAR INTERACTION; ORGANIC CHEMISTRY; PROCESS DEVELOPMENT; REACTION ANALYSIS; STEREOCHEMISTRY;

EID: 10044253262     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol0479904     Document Type: Article

References (13)

1. King, M. L.; Chiang, C. C.; Ling, H. C.; Fujita, E.; Ochiai, M.; McPhail, A. T. J. Chem. Soc., Chem. Commun. 1982, 1150.
2. Proksch, P.; Edrada, R.; Ebel, R.; Bohnenstengel, F. I.; Nugroho, B. W. Curr. Org. Chem. 2001, 5, 923.
3. (a) Trost, B. M.; Greenspan, P. D.; Yang, B. V.; Saulnier, M. G. J. Am. Chem. Soc. 1990, 112, 9022.
4. (b) Kraus, G. A.; Sy, J. O. J. Org. Chem. 1989, 54, 77.
5. (c) Davey, A. E.; Schaeffer, M. J.; Taylor, R. J. K. J. Chem. Soc., Chem. Commun. 1991, 1137. Davey, A. E.; Schaeffer, M. J.; Taylor, R. J. K. J. Chem. Soc., Perkin Trans. 1 1992, 2657.
6. (c) Davey, A. E.; Schaeffer, M. J.; Taylor, R. J. K. J. Chem. Soc., Chem. Commun. 1991, 1137. Davey, A. E.; Schaeffer, M. J.; Taylor, R. J. K. J. Chem. Soc., Perkin Trans. 1 1992, 2657.
7. (d) Watanabe, T.; Shiraga, Y.; Takeuchi, T.; Otsuka, M.; Umezawa, K. Heterocycles 2000, 53, 1051.
8. (e) Dobler, M. R.; Brune, I.; Cederbaum, F.; Cooke, N. G.; Diorazio, L. J.; Hall, R. G.; Irving, E. Tetrahedron Lett. 2001, 42, 8281.
9. All compounds prepared are racemic. The relative stereochemistry is shown.
10. Polo, E.; Barbieri, A.; Traverse, O. Eur. J. Inorg. Chem. 2003, 2, 324.
11. Schoop, A.; Greiving, A.; Goehrt, A. Tetrahedron Lett. 2000, 41, 12, 1913.
12. Spectra of NOESY experiments are included in Supporting Information.
13. Henbest, H. B.; Wilson, R. A. J. Chem. Soc. 1957, 1958.