In vitro antiplasmodial activities of semisynthetic N,N′-spacer- linked oligomeric ergolines

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 4, 2004, Pages 817-824

  Jenett Siems, Kristina ^a   Köhler, Inga ^a   Kraft, Carola ^a   Pertz, Heinz H ^a   Křen, Vladimír ^b   Fišerová, Anna ^b   Kuzma, Marek ^b   Ulrichová, Jitka ^c   Bienzle, Ulrich ^d   Eich, Eckart ^a  

^a FREIE UNIVERSITÄT BERLIN   (Germany)

^b INSTITUTE OF MICROBIOLOGY   (Czech Republic)

^c PALACKÝ UNIVERSITY   (Czech Republic)

^d HUMBOLDT UNIVERSITY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

1,2 BIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL]BENZENE; 1,2,4,5 TETRAKIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL]BENZENE; 1,3 BIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL]BENZENE; 1,3,5 TRIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL] 2,4,6 TRIMETHYLBENZENE; 1,4 BIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL]BENZENE; 1,6 BIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YL]HEXANE; ALIPHATIC COMPOUND; ANTIMALARIAL AGENT; CHLOROQUINE; ERGOLINE DERIVATIVE; FESTUCLAVINE; HEXAKIS[6' METHYL 8BETA' (METHYL)ERGOLIN 1' YLMETHYL]BENZENE; PERGOLIDE; TERGURIDE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL STRAIN 3T3; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYTOTOXICITY; DIMERIZATION; DRUG ACTIVITY; DRUG EFFECT; DRUG SCREENING; DRUG SYNTHESIS; FIBROBLAST; IC 50; IN VITRO STUDY; LIVER CELL; NONHUMAN; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION;

PLASMODIUM FALCIPARUM;

EID: 0842326701     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2003.10.035     Document Type: Article

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