Utility of 1-(2,4-dimethoxyphenyl)-3-aryl-prop-2-ene-1-ones as ring transformer in preparing heterocyclic compounds and their potential biological activities

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 179, Issue 1, 2004, Pages 61-76

  Salem, M A I ^a,c   Soliman, E A ^a   Smith, M B ^b   Mahmoud, M R ^a   Azab, M E ^a  

^a AIN SHAMS UNIVERSITY   (Egypt)

^b Central   (United States)

^c Ain Shams University   (Egypt)

Author keywords

2 Cyanomethylthiazolidin 4 one; 4 oxo 4H pyrano 2,3 d tetrahydropyrimidin 2 thiones; Azo disperse dyes; Diazapinone pyrazolin 5 one; Thiobarbituric acid

Indexed keywords

2 (4 OXOTHIAZOLIDIN 2 YL) 5 OXOPENTANOCARBONITRILE; 2 AMINOPYRIDINE; 2 CYANOMETHYLTHIAZOLIDIN 4 ONE; ALKALINE EARTH METAL; CYANIDE; CYCLOHEXANO[B] 4H PYRAN; CYCLOHEXANONE; CYCLOPROPANE DERIVATIVE; ETHYL 5 OXOPENTANOATE; ETHYLCYANOACETATE; HETEROCYCLIC COMPOUND; HYDRAZINE DERIVATIVE; KETONE DERIVATIVE; PHENOL DERIVATIVE; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; PROPYLENE; PYRAN DERIVATIVE; PYRAZOLIN 5 ONE; PYRIDINE DERIVATIVE; THIOBARBITURIC ACID; UNCLASSIFIED DRUG;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL STRUCTURE; DIAZOTIZATION; DRUG ACTIVITY; DRUG POTENTIATION; DRUG SYNTHESIS; HYDROLYSIS; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MICHAEL ADDITION; PROTON NUCLEAR MAGNETIC RESONANCE; SCREENING TEST; THIN LAYER CHROMATOGRAPHY;

EID: 0742304850     PISSN: 10426507     EISSN: None     Source Type: Journal    
DOI: 10.1080/10426500490257041     Document Type: Article

References (33)

1. V. Sastry and T. Seshardi, Proc. Indian. Acad, Sci., 16A, 29 (1942); C.A., 37, 880 (1943).
2. V. Sastry and T. Seshardi, Proc. Indian. Acad, Sci., 16A, 29 (1942); C.A., 37, 880 (1943).
3. A. Tantawy, H. Eisa, A. Ismail, and M. El-Kerdawy, Alexandria, J. Pharm. Sci., 2, (2) 113 (1988); C.A., 111, 57616 (1989).
4. A. Tantawy, H. Eisa, A. Ismail, and M. El-Kerdawy, Alexandria, J. Pharm. Sci., 2, (2) 113 (1988); C.A., 111, 57616 (1989).
5. Ishihara and S. Kaisha, Ltd. Japan Kokai Tokkyo Koho, Jpn. 81, 127, 223; 06 Oct. 1981, Appl. 80/29, 11 May 829 (1980).
6. M. Takao, Takashi, and T. Juzo, (Sankyo Co. Ltd) Ger. Offen., 2, 627, 223, 30 Dec. 1976, Japan. Appl. 75/74, 19 Jun. 962 (1975).
7. Ishihara and S. Kaisha, Ltd. Jpn. Kokai Tokkyo Koho, 80, 85, 570, 27 Jun. 1980, Appl. 78/160, 25 Dec. 522 (1978).
8. S. Joerg, G. Reinhold, S. Otto, S. Hans Joachim, S. Robert, and L. Klaus, (Bayer A.G.) Ger. Offen., DE 3, 625, 686, 04 Feb. (1988); C.A., 108, 167465 (1988).
9. S. Joerg, G. Reinhold, S. Otto, S. Hans Joachim, S. Robert, and L. Klaus, (Bayer A.G.) Ger. Offen., DE 3, 625, 686, 04 Feb. (1988); C.A., 108, 167465 (1988).
10. P. N. Dhol, T. E. Achary, and A. Nayak, J. Ind. Chem. Soc., 152, 1196 (1975).
11. P. Mitra and A. Mittra, J. Ind. Chem. Soc., 58, 695 (1981).
12. A. Nayak and A. Mittra, J. Ind. Chem. Soc., 57, 643 (1980).
13. Kumiai, Chem. Industries Co. Ltd., Kokai Tokkyo Koho, Jpn. 81, 63, 964 30 May 1981, Appl. 79/139 29 Oct. (1979).
14. M. A. Hassan, A. Afifi, and S. El-Tamany, Pak. J. Sci., Ind. Res., 20, 79 (1977).
15. H. M. F. Madkour, M. A. I. Salem, E. A. Soliman, and N. F. H. Mahmoud, J. Phosphorus, Sulfur, and Silicon, 170, 15, (2001).
16. a) L. Kaplan and D. Glover, J. Am. Chem. Soc., 88, 84 (1966);
17. b) E. Afsah, F. Amer, and M. Soafan, Z. Naturforsch., B. Anorg. Chem. Org. Chem. 35B, 1313 (1980).
18. X. Liuli, Y. Wang, B. Tian, T. Matsuura, and Meng, J., J. Heterocyclic. Chem., 35, 129 (1998).
19. G. A. Newman and P. J. Pauwels, Tetrahedron, 25, 4605 (1969).
20. L. J. Bellamy, The Infra-red Spectrum of Complex Molecules (John Wiley and Sons, New York, 1958), 2nd ed.;
21. b) E. Pretsch, Th. Clerc, J. Seibl, and W. Simon, Tables of Spectral Data for Structures Determination of Organic Compounds, (Springer-Verlag, 1983), 2nd ed.
22. M. El-Deek, M. A. I. Salem, A. A. Hamed, and M. Saman, Revue Roumaine De Chimie, 26, 647 (1981).
23. H. M. F. Madkour, M. A. I. Salem, T. M. Abdel-Rahman, and M. E. Azab, Heterocycles, 38, 57 (1994).
24. V. Ahluwelia, K. Kumar, M. Alauddin, C. Khanduri, and N. Mallika, Synth. Commun., 20, 1265 (1990).
25. A. Sammour, A. Rauf, M. El-Kassaby, and M. A. I. Salem, Acta Chimica Acad. Hungarica, Tomus, 78, 399 (1973).
26. W. M. Abdou, M. A. I. Salem, and R. F. Barghash, J. Phosphorus, Sulfur, and Silicon, 178, 125 (2003).
27. M. Al-Arab, B. Ghanem, and A. Fitton, Tetrahedron, 45, 654 (1987).
28. a) M. Al-Arab and A. Issa, Collect. Czech. Chem. Commun., 52, 1021 (1987);
29. b) M. Al-Arab, B. Ghanem, and M. Olmstead, Synthesis, (10), 1003 (1992).
30. A. Sammour, M. Elzimaity, and A. Abd El-Maksoud, J. Chem., U.A.R., 12, 481 (1969).
31. J. G. Vincent and A. W. Vincent, Proc. Soc. Exptal. Biol. Med., 55, 162 (1944).
32. S. A. Waksman, Proc. Nat. Acad. Sci., USA, 45, 1043 (1959).
33. National Committee for Clinical Laboratory Standards, Methods for dilution Antimicrobial Susceptibility Tests for Bacteria Grow Aerobically, Approved Standard M2-A5, Villianova, PA (1993).