β-Enaminoesters as Building Blocks in Heterocyclic Synthesis. A Novel Synthesis of Fused Azines by Using Blaise Reaction as a Key Step

Advanced Synthesis and Catalysis

Volumn 341, Issue 2, 1999, Pages 147-151

  Erian, Ayman W ^a  

^a CAIRO UNIVERSITY   (Egypt)

Author keywords

Antimalarial agents; Bioorganic chemistry; Heterocycles; Pyrimethamine; enaminoesters

Indexed keywords

EID: 0347713516     PISSN: 16154150     EISSN: None     Source Type: Journal    
DOI: 10.1002/(sici)1521-3897(199902)341:2<147::aid-prac147>3.0.co;2-i     Document Type: Article

References (10)

1. A. W. Erian, Chem. Rev. 1993, 93, 1991
2. E. F. Elslager, J. Davoll, P. Jacob, J. Johnson, L. M. Werbel, J. Med. Chem. 1978, 21, 639
3. The antimalarial-antibacterial effect of quinazolines was supported by US Army Medical Research and Development Command Contract DA-49-193-MD-2754. This is contribution No. 1484 to the Army Research Program on Malaria.
4. J. Davoll, A. M. Johnson, H. J. Davies, O. D. Bird, J. Clarke, E. F. Elslager, J. Med. Chem. 1972, 15, 812
5. P. E. Thompson, A. Bayles, B. Olszewski, Am. J. Trop. Med. Hyg. 1970, 19, 12
6. B. Loev, M. M. Goodman, K. M. Snader, R. Tedeshi, E. Macko, J. Med. Chem. 1974, 17, 956
7. T. McInally, C. J. Tinker, J. Chem. Soc., Perkin Trans. 1, 1988, 1837
8. J. R. Pfister, Synthesis, 1990, 689
9. Biosynthesis of Some Heterocyclic Natural Product. In Comprehensive Heterocyclic Chemistry, Ed. A. R. Katritzky and C. W. Rees, Pergamon Press, Oxford, 1984, 1, p. 95, 96
10. A. Fürstner, Synthesis, 1989, 571 and references cited therein