Allosteric Enhancers of A1 Adenosine Receptors Increase Receptor-G Protein Coupling and Counteract Guanine Nucleotide Effects on Agonist Binding

Molecular Pharmacology

Volumn 64, Issue 6, 2003, Pages 1557-1564

  Figler, Heidi ^a   Olsson, Ray A ^b   Linden, Joel ^a  

^a UNIVERSITY OF VIRGINIA   (United States)

^b UNIVERSITY OF SOUTH FLORIDA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 4,5 DIMETHYL 3 (3 TRIFLUOROMETHYLBENZOYL)THIOPHENE; 2 AMINO 4,5,6,7 TETRAHYDROBENZO[B]THIOPHEN 3 YL BIPHENYL 4 YLMETHANONE; 6 N AMINOBENZYLADENOSINE I 125; 8 CYCLOPENTYLTHEOPHYLLINE; ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR AGONIST; ADENOSINE DERIVATIVE; ATL 525; FORSKOLIN; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); ROLIPRAM; THIOPHENE DERIVATIVE; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; BINDING SITE; CHO CELL; DRUG RECEPTOR BINDING; PRIORITY JOURNAL;

EID: 0346996805     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.64.6.1557     Document Type: Article

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