Synthesis and Antifilarial Evaluation of 7-O-Acetamidyl-4-alkyl-2H-1- benzopyran-2-ones

Arzneimittel-Forschung/Drug Research

Volumn 53, Issue 12, 2003, Pages 857-863

  Katiyar, Diksha ^a   Tiwari, Vinod Kumar ^a   Tripathi, Rama Pati ^a   Reddy, Velurijagan Mohan ^a   Bhattacharya, Shailza Mishra ^a   Saxena, Jitendra Kumar ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

7 O Acetamidyl 4 alkyl 2H 1 benzopyran 2 ones, antifilarial activity, in vitro and in vivo studies; Antifilarial agents; Brugia malayi; Coumarins; DNA topoisomerase II; Steria cervi

Indexed keywords

7 O (CARBETHOXYMETHYL) 2H 1 BENZOPYRAN 2 ONE; 7 O ACETAMIDYL 2H 1 BENZOPYRAN 2 ONE; ANTIFILARIAL AGENT; BENZOPYRAN DERIVATIVE; COUMARIN DERIVATIVE; DNA TOPOISOMERASE (ATP HYDROLYSING); DNA TOPOISOMERASE INHIBITOR; UNCLASSIFIED DRUG;

AMIDATION; ANTIFILARIAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; BRUGIA MALAYI; CARBON NUCLEAR MAGNETIC RESONANCE; DRUG EFFICACY; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; FILARIA; IN VITRO STUDY; IN VIVO STUDY; SETARIA CERVI;

EID: 0346733233     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1299841     Document Type: Article

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