Development of a photoaffinity label for respiratory syncytial virus inhibitors

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 46, Issue 12, 2003, Pages 1105-1116

  Dischino, Douglas D ^a   Cianci, Christopher W ^a   Civiello, Rita ^a   Krystal, Mark ^a   Meanwell, Nicholas A ^a   Morimoto, Hiromi ^b   Williams, Philip G ^b   Yu, Kuo Long ^a,c  

^a BRISTOL MYERS SQUIBB   (United States)

^b LAWRENCE BERKELEY NATIONAL LABORATORY   (United States)

^c ELI LILLY AND COMPANY   (United States)

Author keywords

Photoaffinity label; Radioiodination; RSV inhibitor

Indexed keywords

BENZOIMIDAZOLE; CHLOROMETHYL; IMIDAZOL; IODINATED DERIVATIVES; PHOTOAFFINITY; PHOTOAFFINITY LABEL; RADIOIODINATION; RESPIRATORY SYNCYTIAL VIRUS; RSV INHIBITOR; TRITIATION;

VIRUSES;

1 (4 HYDROXY 3 IODOBENZYL) 3 [1 [2 (3 METHYL 3H DIAZIRIN 3 YL)ETHYL] 2,3 DIHYDRO 1H BENZOIMIDAZOL 2 YLMETHYL] 1,3 DIHYDROBENZOIMIDAZOL 2 ONE I 123; 1 (4 HYDROXY 3 IODOBENZYL) 3 [1 [2 (3 METHYL 3H DIAZIRIN 3 YL)ETHYL] 2,3 DIHYDRO 1H BENZOIMIDAZOL 2 YLMETHYL] 1,3 DIHYDROBENZOIMIDAZOL 2 ONE I 125; 1 ISOPROPYL 3 [1 [2 (3 METHYL 3H DIAZIRIN 3 YL)ETHYL] 1H BENZOIMIDAZOL 2 YL]METHYL 1,3 DIHYDROBENZOIMIDAZOL 2 ONE H 3; 2 CHLOROMETHYL 1 [2 (3 METHYL 3H DIAZIRIN 3 YL)ETHYL] 1H BENZOIMIDAZOLE; BENZIMIDAZOLE DERIVATIVE; N ISOPROPENYL 2 BENZIMIDAZOLONE; RADIOACTIVE IODINE; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; PHOTOAFFINITY LABELING; RESPIRATORY SYNCYTIAL PNEUMOVIRUS;

RESPIRATORY SYNCYTIAL VIRUS; RICE STRIPE VIRUS;

EID: 0345686528     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.743     Document Type: Article

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