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Volumn 55, Issue 4, 2003, Pages 597-606

International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on Terms and Symbols in Quantitative Pharmacology

Author keywords

[No Author keywords available]

Indexed keywords

CONCENTRATION RESPONSE; DRUG CLASSIFICATION; DRUG MECHANISM; DRUG RECEPTOR BINDING; EQUILIBRIUM CONSTANT; NOMENCLATURE; PRIORITY JOURNAL; REVIEW;

EID: 0345490945     PISSN: 00316997     EISSN: None     Source Type: Journal    
DOI: 10.1124/pr.55.4.4     Document Type: Review
Times cited : (517)

References (27)
  • 1
    • 0009644628 scopus 로고
    • Some quantitative uses of drug antagonists
    • Arunlakshana O and Schild HO (1959) Some quantitative uses of drug antagonists. Br J Pharmacol 14:48-58.
    • (1959) Br J Pharmacol , vol.14 , pp. 48-58
    • Arunlakshana, O.1    Schild, H.O.2
  • 2
    • 0031815337 scopus 로고    scopus 로고
    • Effector pathway-dependent relative efficacy at serotonin type 2A and 2C receptors: Evidence for agonist-directed trafficking of receptor stimulus
    • Berg KA, Maayani S, Goldfarb J, Scaramellini C, Leff P, Clarke WP (1998) Effector pathway-dependent relative efficacy at serotonin type 2A and 2C receptors: evidence for agonist-directed trafficking of receptor stimulus. Mol Pharmacol 54:94-104.
    • (1998) Mol Pharmacol , vol.54 , pp. 94-104
    • Berg, K.A.1    Maayani, S.2    Goldfarb, J.3    Scaramellini, C.4    Leff, P.5    Clarke, W.P.6
  • 3
    • 0021058380 scopus 로고
    • Operational models of pharmacological agonism
    • Black JW and Leff P (1983) Operational models of pharmacological agonism. Proc R Soc Lond B Biol Sci 220:141-162.
    • (1983) Proc R Soc Lond B Biol Sci , vol.220 , pp. 141-162
    • Black, J.W.1    Leff, P.2
  • 5
    • 0033929371 scopus 로고    scopus 로고
    • Agonist-directed trafficking of porcine α2A-adrenergic receptor signaling in Chinese hamster ovary cells: 1-Isoproterenol selectively activates Gs
    • Brink CB, Wade SM, and Neubig RR (2000) Agonist-directed trafficking of porcine α2A-adrenergic receptor signaling in Chinese hamster ovary cells: 1-isoproterenol selectively activates Gs. J Pharmacol Exp Ther 294:539-547.
    • (2000) J Pharmacol Exp Ther , vol.294 , pp. 539-547
    • Brink, C.B.1    Wade, S.M.2    Neubig, R.R.3
  • 6
    • 0032436491 scopus 로고    scopus 로고
    • Assessing the distribution of parameters in models of ligand-receptor interaction: To log or not to log
    • Christopoulos A (1998) Assessing the distribution of parameters in models of ligand-receptor interaction: to log or not to log. Trends Pharmacol Sci 19:351-357.
    • (1998) Trends Pharmacol Sci , vol.19 , pp. 351-357
    • Christopoulos, A.1
  • 7
    • 0036258990 scopus 로고    scopus 로고
    • G protein-coupled receptor allosterism and complexing
    • Christopoulos A and Kenakin T (2002) G protein-coupled receptor allosterism and complexing. Pharmacol Rev 54:323-374.
    • (2002) Pharmacol Rev , vol.54 , pp. 323-374
    • Christopoulos, A.1    Kenakin, T.2
  • 8
    • 0002134457 scopus 로고
    • Affinity, efficacy and receptor classification: Is the classical theory still useful?
    • (Black JW, Jenkinson DH, and P. Gerskowitch V, eds), Alan R. Liss, New York
    • Colquhoun D (1987) Affinity, efficacy and receptor classification: is the classical theory still useful? in Perspectives on Receptor Classification: Receptor Biochemisty and Methodology (Black JW, Jenkinson DH, and P. Gerskowitch V, eds) vol. 6, pp. 103-114, Alan R. Liss, New York.
    • (1987) Perspectives on Receptor Classification: Receptor Biochemisty and Methodology , vol.6 , pp. 103-114
    • Colquhoun, D.1
  • 9
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (150) of an enzymatic reaction
    • Cheng Y and Prusoff W (1973) Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (150) of an enzymatic reaction. Biochem Pharmacol 22:3099-3108.
    • (1973) Biochem Pharmacol , vol.22 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.2
  • 10
    • 70449143838 scopus 로고
    • Interaction at end-plate receptors between different choline derivatives
    • Del Castillo J and Katz B (1957) Interaction at end-plate receptors between different choline derivatives. Proc R Soc Lond B Biol Sci 146:369-381.
    • (1957) Proc R Soc Lond B Biol Sci , vol.146 , pp. 369-381
    • Del Castillo, J.1    Katz, B.2
  • 11
    • 0019137579 scopus 로고
    • A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor
    • Delean A, Stadel JM, and Lefkowitz RJ (1980) A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor. J Biol Chem 255:7108-7117.
    • (1980) J Biol Chem , vol.255 , pp. 7108-7117
    • Delean, A.1    Stadel, J.M.2    Lefkowitz, R.J.3
  • 12
    • 0002355204 scopus 로고
    • The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes
    • Furchgott RF (1966) The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes. Adv Drug Res 3:21-55.
    • (1966) Adv Drug Res , vol.3 , pp. 21-55
    • Furchgott, R.F.1
  • 13
    • 0000911106 scopus 로고    scopus 로고
    • Introductory address. Part I. Biological aspects: The antagonism of drugs
    • 1043
    • Gaddum JH (1043) Introductory address. Part I. Biological aspects: the antagonism of drugs. Trans Faraday Soc 39:323-332.
    • Trans Faraday Soc , vol.39 , pp. 323-332
    • Gaddum, J.H.1
  • 14
    • 0029054965 scopus 로고
    • Agonist-receptor efficacy. II. Agonist trafficking of receptor signals
    • Kenakin T (1995) Agonist-receptor efficacy. II. Agonist trafficking of receptor signals. Trends Pharmacol Sci 16:232-238.
    • (1995) Trends Pharmacol Sci , vol.16 , pp. 232-238
    • Kenakin, T.1
  • 16
    • 0036591660 scopus 로고    scopus 로고
    • The ligand paradox between affinity and efficacy: Can you be there and not make a difference?
    • Kenakin T and Onaran O (2002) The ligand paradox between affinity and efficacy: can you be there and not make a difference? Trends Pharmacol Sci 23:275-280.
    • (2002) Trends Pharmacol Sci , vol.23 , pp. 275-280
    • Kenakin, T.1    Onaran, O.2
  • 17
    • 0027170155 scopus 로고
    • Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng-Prusoff equations
    • Lazareno S and Birdsall NJM (1993) Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng-Prusoff equations. Br J Pharmacol 109:1110-1119.
    • (1993) Br J Pharmacol , vol.109 , pp. 1110-1119
    • Lazareno, S.1    Birdsall, N.J.M.2
  • 18
    • 0029094516 scopus 로고
    • Analysis of competitive agonist-antagonist interactions by nonlinear regression
    • Lew MJ and Angus JA (1995) Analysis of competitive agonist-antagonist interactions by nonlinear regression. Trends Pharmacol Sci 16:328-337.
    • (1995) Trends Pharmacol Sci , vol.16 , pp. 328-337
    • Lew, M.J.1    Angus, J.A.2
  • 22
    • 84982328496 scopus 로고
    • pA, a new scale for the measurement of drug antagonism
    • Schild HO (1947) pA, a new scale for the measurement of drug antagonism. Br J Pharmacol 2:189-206.
    • (1947) Br J Pharmacol , vol.2 , pp. 189-206
    • Schild, H.O.1
  • 23
    • 78651007352 scopus 로고
    • x and competitive drug antagonism
    • x and competitive drug antagonism. Br J Pharmacol 4:277-280.
    • (1949) Br J Pharmacol , vol.4 , pp. 277-280
    • Schild, H.O.1
  • 24
    • 0036265931 scopus 로고    scopus 로고
    • International Union of Pharmacology. XXXI. Recommendations for the nomenclature of multimeric G protein-coupled Receptors
    • Spedding M, Bonner TI, and Watson SP (2002) International Union of Pharmacology. XXXI. Recommendations for the nomenclature of multimeric G protein-coupled Receptors. Pharmacol Rev 54:232-232.
    • (2002) Pharmacol Rev , vol.54 , pp. 232-232
    • Spedding, M.1    Bonner, T.I.2    Watson, S.P.3
  • 25
    • 0010673662 scopus 로고
    • A modification of receptor theory
    • Stephenson RP (1956) A modification of receptor theory. Br J Pharmacol 11:379-393.
    • (1956) Br J Pharmacol , vol.11 , pp. 379-393
    • Stephenson, R.P.1
  • 26
    • 0000921501 scopus 로고
    • Analysis of dose-response curves
    • (Daniel and Paton, ed), Plenum Press, New York
    • Waud DR (1975) Analysis of dose-response curves, in Methods in Pharmacology: Smooth Muscle (Daniel and Paton, ed) vol 3, pp 471-506, Plenum Press, New York.
    • (1975) Methods in Pharmacology: Smooth Muscle , vol.3 , pp. 471-506
    • Waud, D.R.1
  • 27
    • 0018143518 scopus 로고
    • Kinetic and empirical analysis of dose-response curves illustrated with a cardiac example
    • Waud DR, Son SL, and Waud BE (1978) Kinetic and empirical analysis of dose-response curves illustrated with a cardiac example. Life Sci 22:1275-1286.
    • (1978) Life Sci , vol.22 , pp. 1275-1286
    • Waud, D.R.1    Son, S.L.2    Waud, B.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.