Synthesis and antimicrobial activity of {2-[2-(N,N-disubstituted thiocarbamoyl-sulfanyl)-acylamino]thiazol-4-yl}acetic acid ethyl esters

Archiv der Pharmazie

Volumn 336, Issue 1, 2003, Pages 39-46

  Ateş, Öznur ^b   Gürsoy, Aysel ^b   Altintaş, Handan ^a   Ötük, Gülten ^a   Birteksöz, Seher ^a  

^a ISTANBUL UNIVERSITY   (Turkey)

^b NONE

Author keywords

2 (Thiocarbamoyl sulfanyl)acylamino 1,3 thiazoles; Anti bacterial; Antifungal; Antituberculosis activities; Synthesis

Indexed keywords

2 [(THIOCARBAMOYLSULFANYL)ACYLAMINO] 1,3 THIAZOLE; 2 [[2 (N,N DITHIOCARBAMOYLSULFANYL)ACYLAMINO]THIAZOL 4 YL]ACETIC ACID ETHYL ESTER; 2 AMINO 1,3 THIAZOLE DERIVATIVE; ANTIBIOTIC AGENT; CEFUROXIME; COTRIMOXAZOLE; DITHIOCARBAMIC ACID DERIVATIVE; THIAZOLE DERIVATIVE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; DRUG STRUCTURE; DRUG SYNTHESIS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; INFRARED SPECTROSCOPY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; ULTRAVIOLET SPECTROSCOPY;

ANTI-BACTERIAL AGENTS; ANTITUBERCULAR AGENTS; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0345270000     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.200390002     Document Type: Article

References (33)

1. F. Gagiu, G. Csavassy, E. Bebesel, Farmacia 1968, 16, 171-176 [Chem. Abstr. 1968, 69. 77155m].
2. F. Gagiu, G. Csavassy, E. Bebesel, Farmacia 1968, 16, 171-176 [Chem. Abstr. 1968, 69. 77155m].
3. R. Heymes, Ger. Offen. 2,700,552 1977 [Chem. Abstr. 1977, 87. 152245t].
4. M. Vignau, A. Lutz, Ger. Offen. 2,700,712, 1977 [Chem. Abstr. 1977, 87. 152252t]
5. S. N. Sawhney, S. K. Arora, S. P. Singh, Indian J. Chem. 1978, Sect. B, 16B, 523-524 [Chem. Abstr. 1978, 89. 215300w].
6. S. N. Sawhney, S. K. Arora, S. P. Singh, Indian J. Chem. 1978, Sect. B, 16B, 523-524 [Chem. Abstr. 1978, 89. 215300w].
7. S. S. Tiwari, R. K. Satsang, S. M. M. Zaidi, Indian Drugs 1979, 16, 292-294 [Chem. Abstr. 1980. 92. 94312c].
8. S. S. Tiwari, R. K. Satsang, S. M. M. Zaidi, Indian Drugs 1979, 16, 292-294 [Chem. Abstr. 1980. 92. 94312c].
9. M. Ochiai, A. Morimoto, Y. Matsushita, U.S. Patent 4,182,868 1980 [Chem. Abstr. 1980 92. 163985p].
10. M. Ochiai, A. Morimoto, Y. Matsushita, J. Antibiot. 1980, 33, 1014-1021 [Chem. Abstr. 1981, 94. 103270h].
11. M. Ochiai, A. Morimoto, Y. Matsushita, J. Antibiot. 1980, 33, 1014-1021 [Chem. Abstr. 1981, 94. 103270h].
12. M. Sendai, T. Iwahi, Y. Ishibashi, Jpn. Kokai Tokkyo Koho JP 08,151,386 1994 [Chem. Abstr. 1996, 125. 167689t].
13. H. Schönenberger, P. Lippert, Pharmazie 1972, 27, 139-145.
14. C. H. Fuchsmann, W. H. Meek, US 3,557 174 1971 [Chem. Abstr. 1971, 74.87636m].
15. R. R. Dalvi, D. P. Deores, Acta Pharmacol. Toxicol. (Copenh.) 1986, 58, 38.
16. N. Kh. Maksudov, M. A. Safaev, Uzb. Khim. Zh. 1981, 26-29 [Chem. Abstr. 1982, 96. 85383g].
17. N. Kh. Maksudov, M. A. Safaev, Uzb. Khim. Zh. 1981, 26-29 [Chem. Abstr. 1982, 96. 85383g].
18. R. J. Topping, M. M. Jones, Med. Hypotheses 1988, 27, 55.
19. C. Şafak, H. Erdoǧan, Arzneim.-Forsch./Drug Res. 1992, 42, 123-126.
20. Ö. Ateş, H. Altintaş, Arzneim.-Forsch./Drug Res. 2000, 50, 569-575.
21. N. Cesur, Ö. Ateş, Acta Pharm. Turc. 1994, 36, 74-79 [Chem. Abstr. 1995, 123. 198684a].
22. N. Cesur, Ö. Ateş, Acta Pharm. Turc. 1994, 36, 74-79 [Chem. Abstr. 1995, 123. 198684a].
23. Ö. Ateş, N. Cesur, Farmaco 1995, 50, 361-364.
24. A. Gürsoy, Ö. Ateş, Eur. J. Med. Chem. 1996, 31, 643-646.
25. G. Çapan, N. Ergenç. Sci. Pharm. 1993, 61, 243-250.
26. N. Karali, I. Apak, Arch. Pharm. Pharm. Med. Chem. 1999, 332, 422-426.
27. D. V. Naik, G. J. Palanik, Acta Crystallogr. 1974, 30, B2396 [Chem. Abstr. 1974, 81. 160506v].
28. D. V. Naik, G. J. Palanik, Acta Crystallogr. 1974, 30, B2396 [Chem. Abstr. 1974, 81. 160506v].
29. F. Beaulieu, V. Snieckus, Synthesis 1992, 112-118.
30. M. Oki, Recent Advances in Atropisomerism, Eds. N. L. Allinger, E. L. Eliel, S. H. Wilen, Topics in Stereochemistry 14, John Wiley & Sons, New York-Chichester-Brisbane-Toronto-Singapore, 1983, pp. 10-28.
31. K. R. Gayathri, D. N. Sathyanarayana, Spectrochim. Acta 1981, 37A, 31-36.
32. R. K. Bansal, G. Bhagchandani, J. Indian Chem. Soc. 1982, 59, 277.
33. C. B. Inderleid, Antibiotics in Laboratory Medicine, 3rd ed., V. Lorian (Ed.), William and Wilkins, Baltimore 1991, 134-197.