Thrombin inhibitors and thrombin receptor agonists/antagonists

Pharmacochemistry Library

Volumn 24, Issue C, 1996, Pages 271-289

  DiMaio, J ^a   Winocour, P ^a   Leblond, L ^a   Saifeddine, M ^b   Laniyonu, A ^b   Holienberg, M D ^b  

^a Shire Canada   (Canada)

^b UNIVERSITY OF CALGARY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0345004037     PISSN: 01657208     EISSN: None     Source Type: Book Series    
DOI: 10.1016/S0165-7208(96)80022-5     Document Type: Article

References (122)

1. Kaplan N.M. J Cardiovasc Pharmacol 4 (1982) S187-S189
2. Kerényi T., and Schneider F. In: Machovich R. (Ed). Blood Vessel Wall and Thrombosis (1988), CRC Press, Boca Raton 51-69
3. Shepard L.Y. Trends Biotechnol 11 (1991) 80-85
4. Cook N.S., and Ubben D. Trends Pharmacol Sci 11 (1990) 444-451
5. Sharf R.E., and Harker L.A. Blut 55 (1987) 131-144
6. Furie B., and Furie B.C. Cell 53 (1988) 505-518
7. Altieri D.C. Blood 81 (1993) 569-579
8. Mann K.G., Jenny R.J., and Krishnaswamy S. Ann Rev Biochem 57 (1988) 915-956
9. Machovic R. In: Machovich R. (Ed). Blood vessel wall and Thrombosis (1988), CRC Press, Boca Raton 128-140
10. Andrews R.K., and Fox J. Curr Opinion Cell Biol 2 (1990) 894-901
11. Kunicki T.J. Blut 59 (1989) 30-34
12. Jonasson L., Holm J., Skalli O., Bondjers G., et al. Arteriosclerosis 6 (1986) 131
13. Schwartz S.M., and Gajdusek C.M. Prog Thromb Hemost 6 (1983) 85-112
14. Fitzgerald D.J., and Fitzgerald G.A. Proc Natl Acad Sci USA 86 (1989) 7585-7589
15. Gast A., Tschopp T.B., and Baumgartner H.R. Arterioscler Thromb 14 (1994) 1466-1474
16. Fenton J.W. Ann NY Acad Sci 370 (1981) 468-485
17. Magnusson S. In: Boyer P.D. (Ed). Enzymes (1971), Academic Press, New York 277-321
18. Fenton J.W., Landis B.H., Walz D.A., Bing D.H., et al. In: Bing D.H. (Ed). The Chemistry and Physiology of Human Plasma proteins (1978), Pergamon Press, Oxford 151-183
19. Chang J.Y. Biochem J 240 (1986) 787-802
20. Charles S., Greenberg K., Achyuthan K.E., Hiraglia C.C., et al. Ann NY Acad Sci 485 (1986) 140-143
21. Hemker HC, Beguin S. In: Jolles G, Legrand Y, Nurden A, eds. London: Academic Press, 1986; 219-226.
22. Phillips D.R., Charo I.F., Parise L.V., and Fitzgerald L.A. Blood 71 (1988) 831-843
23. Hynes R.O. Cell 48 (1987) 549-554
24. Nesheim M.E., Hibbard L.S., and Tracy P.B. In: Mann K.G., and Taylor F.B. (Eds). The regulation of coagulation (1980), Elsevier-North Holland, New York 145-159
25. Nawroth P.P., Kisiel W., and Stern D.M. Clin Haematol 14 (1985) 531-546
26. Kroll M.H., and Schafer A.I. Blood 74 (1989) 1181-1195
27. Vu T.K.H., Hung D.T., Wheaton F.I., and Coughlin S.R. Cell 64 (1991) 1057-1068
28. Bahou W.F., Coller B.S., Potter C.L., Norton K.J., et al. J Clin Invest 91 (1993) 1405-1413
29. Rasmussen U.B., Vouret-Craviari V., Jallat S., Schlesinger Y., et al. FEBS Lett 288 (1991) 123-128
30. Hung D.T., Vu T.K.H., Nelken N.A., and Coughlin S.R. J Cell Biol 116 (1992) 827-832
31. Zhong C., Hayzer D.J., Corson M.A., and Runger M.S. J Biol Chem 267 (1992) 16975-16979
32. Howells G.L., Macey M., Curtis M.A., and Stone S.R. Brit J Haematol 84 (1993) 156-160
33. Dihanich M., Kaser M., Reinhard E., Cunningham D., et al. Neuron 6 (1991) 575-581
34. Deschepper C.F., Bigornia V., Berens M.E., and Lapointe M.C. Mol Brain Res 11 (1991) 355-358
35. Weinstein J.R., Gold S.J., Cunningham D.S., and Gall C.M. J Neurosci 15 (1995) 2906-2919
36. Jalink K., and Moolenar W.H. J Cell Biol 118 (1992) 411-419
37. Suiclan H.S., Stone S.R., Hemmings B.A., and Monard D. Neuron 8 (1992) 363-375
38. Smith G.F., Neubauer B.L., Soundboom J.L., Best K.L., et al. Thrombosis Res 50 (1988) 163-174
39. Honn K.V., Tang D.G., and Chen Y.Q. Sem Thromb Haemostas 18 (1992) 392-415
40. Nierodzik M.L., Plotkin A., and Kajumo F. J Clin Invest 87 (1991) 229-236
41. Klepfish A., Greco M.A., and Karpatkin S. Int J Cancer 53 (1993) 978-982
42. Vu T.K.H., Wheaton V.I., Hung D.T., and Coughlin S.R. Nature 353 (1991) 674-677
43. Liu L., Vu T.K.H., Esmon C.T., and Coughlin S.R. J Biol Chem 266 (1991) 19680-19697
44. Rosenberg R.D., and Damus P.S. J Biol Chem 248 (1973) 6490-6505
45. Carrell RW, Boswell DR. In: Barret AJ, Salvesen G, eds. North Holland: Elsevier, 1986; 403-418.
46. Travis J., and Salvesen G.S. Ann Rev Biochem 52 (1983) 655-709
47. Ware J.A., and Salzman E.W. In: Lane D.A., and Lindahl U. (Eds). Heparin Chemical and Biological Properties, Clinical Applications (1989), Edward Arnold, London 475-494
48. Esmon C.T. Science 235 (1987) 1348-1352
49. Sawyer R.T. Biopapers J 10 (1990) 11-13
50. Markwardt F. Methods Enzymol 19 (1970) 925-932
51. Tuszynski G.P., Gasic T.B., and Gasic G.J. J Biol Chem 262 (1987) 9718-9723
52. Connolly T.M., Jacobs J.W., and Condra C. J Biol Chem 267 (1992) 6893-6898
53. Budzynski A.Z., Olexa S.A., and Sawyer R.T. Proc Soc Exp Biol Med 168 (1981) 259-265
54. Keller P., Schultz L.D., Condra C., Karczewski J., et al. J Biol Chem 267 (1992) 6899-6904
55. Dodt J., Machleidt N., Seemuller U., Maschler R., et al. Biol Chem Hoppe-Seyler 367 (1986) 803-811
56. Trippier D. Folia Haematol 115 (1988) 30-35
57. Dodt J., Köhler S., Smitz B., and Wilhelm B. J Biol Chem 265 (1990) 713-718
58. Stone S.R., Braun P.J., and Hofsteenge J. Biochemistry 26 (1987) 4617-4624
59. Noé G., Hofsteenge J., Rovelli G., and Stone S.R. J Biol Chem 263 (1988) 11729-11735
60. Wallace A., Dennis S., Hofsteenge J., and Stone S.R. Biochemistry 28 (1989) 10079-10084
61. Grütter M.G., Priestle J.P., Rahuel J., Grossenbacher H., Bode W., et al. Embo J 9 (1990) 2361-2363
62. Rydel T.J., Ravichandran K.G., Tulinsky A., Bode W., et al. Science 249 (1990) 277-280
63. Braun P.J., Dennis S., Hofsteenge J., and Stone S.R. Biochemistry (1988) 6517-6522
64. Lipowski A.W. Pol J Pharmacol Pharm 39 (1987) 585-596
65. Krstenansky J.L., and Mao J.J.T. FEBS Lett 211 (1987) 10-16
66. Maraganore J.M., Chao B., Joseph M.L., Jablonski J., et al. J Biol Chem 264 (1989) 8692-8698
67. DiMaio J., Gibbs B., Munn D., Lefebvre J., Ni F., et al. J Biol Chem 265 (1990) 21698-21703
68. Bajusz S., Barabas E., Tolnay P., Szell E., et al. Int J Peptide Protein Res 12 (1978) 217-221
69. Maraganore J.M., Bourdon P., Jablonski J., Ramachandran K.L., et al. Biochemistry 29 (1990) 7071-7095
70. DiMaio J., Ni F., Gibbs B., and Konishi Y. FEBS Lett 282 (1991) 47-52
71. DiMaio J., Gibbs B., Lefebvre J., Konishi Y., et al. J Med Chem 35 (1992) 3331-3341
72. Zdanov A., Wu S., DiMaio J., Konishi Y., et al. Proteins Struct Funct Gen 17 (1993) 252-265
73. Hanson S.R., and Harker L.A. Proc Natl Acad Sci USA 85 (1988) 3184-3188
74. Kelly A.B., Marzec U.M., Krupski W., Bass A., et al. Blood 77 (1991) 1006-1012
75. Maraganore J.M. In: Anderson P.S., Kenyon G.L., and Marshall G.R. (Eds). Perspectives in Drug Discovery and Design (1994), Escom, Leiden 461-478
76. Shand R.A., Smith J.R., and Wallis R.B. Thromb Res 36 (1984) 223-232
77. Carone F.A., Peterson D.R., and Flouret G. J Lab Clin Med 100 (1982) 1-14
78. Markwardt F. Cardiovasc Drug Rev 10 (1992) 211-232
79. Kurz K.D., Main B.W., and Sandusky G.E. Thrombosis Res 60 (1990) 269-280
80. Walz D.A., Anderson G.F., Fenton II J.W., and Shuman M.A. Ann NY Acad Sci 485 (1986) 323-334
81. Fenton II J.W. Ann NY Acad Sci 485 (1986) 5-15
82. Shuman M.A. Ann NY Acad Sci 485 (1986) 228-229
83. Bar-Shavit R., Kahn A.J., Mann K.G., and Wilner G.D. Proc Nat Acad Sci 83 (1986) 976-980
84. Bar-Shavit R., Benezra M., Sabbah V., and Bode W. Amer J Resp Cell Mol Biol 6 (1992) 123-130
85. Davey M.G., and Luscher E.F. Nature (Lond) 216 (1967) 857-858
86. Chen L.-B., and Buchanan J.M. Proc Nat Acad Sci 72 (1975) 131-135
87. White R.P., Chapleau C.E., Dugdale M., and Robertson J.T. Stroke 11 (1980) 363-368
88. Cunningham D.D., and Farrell D.H. Ann NY Acad Sci 485 (1986) 240-248
89. Bar-Shavit R., Eldor A., and Vlodavsky I. J Clin Invest 84 (1989) 1096-1104
90. Cuatrecasas P., and Hollenberg M.D. Adv Protein Chem 30 (1976) 251-451
91. Coughlin S.R., Vu T.-K., Hung D.T., and Wheaton V.I. J Clin Invest 89 (1992) 351-355
92. Ishii K., Hein L., Kobilka B., and Coughlin S.R. J Biol Chem 268 (1993) 9780-9786
93. Scarborough R.M., Naughton M.A., Teng W., Hung D.T., et al. J Biol Chem 267 (1992) 13146-13149
94. Vassallo Jr. R.R., Kieber-Emmons T., Cichowski K., and Brass L.F. J Biol Chem 267 (1992) 6081-6085
95. Muramatsu I., Laniyonu A.A., Moore G.J., and Hollenberg M.D. Can J Physiol Pharmacol 70 (1992) 996-1003
96. Yang S.-G., Laniyonu A.A., Saifeddine M., Moore G.J., et al. Life Sciences 51 (1992) 1325-1332
97. DeBlois D., Drapeau G., Petitclerc E., and Marceau F. Brit J Pharmacol 105 (1992) 959-967
98. Antonaccio M.J., Normandin D., Serafino R., and Moreland S. J Pharmacol Exp Ther 266 (1993) 125-132
99. Laniyonu A.A., and Hollenberg M.D. Brit J Pharmacol 114 (1995) 1680-1686
100. Hung D.T., Wong Y.H., Vu T.-K., and Coughlin S.R. J Biol Chem 267 (1992) 20831-20834
101. Vouret-Craviari V., Obberghen-Schilling, Rasmussen U.B., Pavirani A., et al. Mol Biol Cell 3 (1992) 95-102
102. Glen K.C., Frost G.H., Bergmann J.S., and Carney D.H. Pept Res 1 (1988) 65-73
103. Hollenberg M.D., Laniyonu A.A., Saifeddine M., and Moore G.J. Mol Pharmacol 43 (1993) 921-930
104. Chao B.H., Kalkunte S., Maraganore J.M., and Stone S.R. Biochemistry 31 (1992) 6175-6178
105. Hui K.Y., Jakubowski J.A., Wyss V.L., and Angleton E.L. Biochem Biophys Res Comm 184 (1992) 790-796
106. Sabo T., Gurwitz D., Motola L., Brodt P., et al. Biochem Biophys Res Commun 188 (1992) 604-610
107. Hollenberg M.D., Yang S.G., Laniyonu A.A., Moore G.J., et al. Mol Pharmacol 42 (1992) 186-191
108. Natarajan S., Riexinger D., Peluso M., and Seiler S.M. Int J Peptide Protein Res 45 (1995) 145-151
109. Tay-Uyboco J., Poon M.-C., Ahmad S., and Hollenberg M.D. Brit J Pharmacol 115 (1995) 569-578
110. Ahlquist R.P. Am J Physiol 153 (1948) 586-600
111. McIntyre P., Phillips E., Skidmore E., Brown M., et al. Mol Pharmacol 44 (1993) 346-355
112. Kenakin T.P., and Morgan P.H. Mol Pharmacol 35 (1989) 214-222
113. Nystedt S., Emilsson K., Wahlestedt C., and Sundelin J. Proc Natl Acad Sci USA 91 (1994) 9208-9212
114. Nystedt S., Larsson A.-K., Aberg H., and Sundelin J. J Biol Chem 270 (1995) 5950-5955
115. Kinlough-Rathbone R.L., Rand M.L., and Packham M.A. Blood 82 (1993) 103-106
116. Walker R.M., Dai J., and Ku D.D. Faseb J 9 (1995) A57
117. Rasmussen U.B., Gachet C., Schlesinger Y., Hanau D., et al. J. Biol. Chem 268 (1993) 14322-14328
118. Coughlin SR, Scarborough RM. International Patent Application, Publication No WO92/14750, 3 Sept. 1992.
119. Seiler S.M., Peluso M., Michel I.M., Goldenberg H., et al. Biochem Pharmacol 49 (1995) 519-528
120. Tesfamariam B. Am J Physiol 267 (1994) H1962-H1967
121. Ku D.D., Zaleski J.K., and Palgunachari M.N. Faseb J 8 (1994) A328
122. Doorbar J., and Winter G. J Mol Biol 244 (1994) 361-369