Heterocyclic aminopyrrolidine derivatives as melatoninergic agents

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 24, 2003, Pages 4381-4384

  Sun, Li Qiang ^a   Chen, Jie ^a   Mattson, Ronald J ^a   Epperson, James R ^a   Deskus, Jeffrey A ^a   Li, Wen Sen ^a   Takaki, Katherine ^a   Hodges, Donald B ^a   Iben, Lawrence ^a   Mahle, Cathy D ^a,b   Ortiz, Astrid ^a,b   Molstad, David ^a,b   Ryan, Elaine ^a   Yeleswaram, Krishnaswamy ^a,c   Xu, Cen ^a   Luo, Guanglin ^a  

^a BRISTOL MYERS SQUIBB   (United States)

^b BAYER CORPORATION   (United States)

^c Experimental Station   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

HETEROCYCLIC AMINE; HORMONE RECEPTOR STIMULATING AGENT; LIGAND; MELATONIN 1 RECEPTOR; MELATONIN 2 RECEPTOR; MELATONIN DERIVATIVE; MELATONIN RECEPTOR; PYRROLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTERY CONSTRICTION; ARTICLE; BINDING AFFINITY; BOLUS INJECTION; CELL LINE; CHIRALITY; CIRCADIAN RHYTHM; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BINDING; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG BRAIN LEVEL; DRUG CLEARANCE; DRUG EFFECT; DRUG PENETRATION; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG STABILITY; DRUG SYNTHESIS; ENANTIOMER; ENANTIOSELECTIVITY; MOLECULAR CLONING; MOUSE; NONHUMAN; RAT; SLEEP DISORDER; STEREOCHEMISTRY;

EID: 0344496012     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.09.030     Document Type: Article

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