The dipeptide neurokinin-1 receptor antagonist S19752 is a potent and long-acting inhibitor of bronchoconstriction when administered by aerosol to the guinea pig in vivo

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 2, 1997, Pages 203-208

  Fauchère, Jean Luc ^a   Kucharczyk, Nathalie ^a   Jacoby, Edgar ^a   Lonchampt, Michel ^a   Robineau, Pascale ^a   Dacquet, Catherine ^a   Regoli, Domenico ^b   Canet, Emmanuel ^a  

^a INSTITUT DE RECHERCHES SERVIER   (France)

^b NONE

Author keywords

[No Author keywords available]

Indexed keywords

3 (2 METHOXYBENZYLAMINO) 2 PHENYLPIPERIDINE; HISTAMINE; MEPYRAMINE; NEUROKININ 1 RECEPTOR; NEUROKININ 1 RECEPTOR ANTAGONIST; RECEPTOR SUBTYPE; S 19752; SUBSTANCE P; UNCLASSIFIED DRUG;

AEROSOL; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING SITE; BRONCHOSPASM; CHO CELL; DRUG ACTIVITY; DRUG RECEPTOR BINDING; DRUG SOLUBILITY; DRUG SYNTHESIS; GUINEA PIG; HUMAN; HUMAN TISSUE; INHALATIONAL DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN;

EID: 0343907300     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(96)00604-X     Document Type: Article

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