Regioselective alkylations of optically active 4,5-dihydro- 1,2,4- triazin-6(1H)-ones

Tetrahedron Letters

Volumn 41, Issue 5, 2000, Pages 671-674

  Sanière, Laurent ^a   Schmitt, Martine ^a   Bourguignon, Jean Jacques ^a  

^a Laboratoire de Pharmacochimie   (France)

Author keywords

[No Author keywords available]

Indexed keywords

4,5 DIHYDRO 1,2,4 TRIAZIN 6(1H) ONE; TRIAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; FRANCE; MOLECULAR INTERACTION; STEREOCHEMISTRY; SYNTHESIS;

EID: 0343819996     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)02162-0     Document Type: Article

References (10)

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4. Collins, D. J.; Hugues, T. C.; Johnson, W. M. Aust. J. Chem. 1996, 49, 463-468.
5. Chayer, S.; Schneider, M. R.; Bourguignon, J.-J. Submitted for publication.
6. CH-NH=1 Hz, -CH), 5.10-5.20 (m, 1H, NH), 7.40-7.50 (m, 3H, H arom), 7.60-7.75 (m, 2H, H arom).
7. 3,4 and compared with our reaction products in order to ascertain the structure of different regioisomers.
8. Kaji, K.; Kusuya, M. Chem. Pharm. Bull. 1970, 18, 147-156.
9. El-Abdelah, M. M.; Hussein, A. Q.; Thaher, B. A. Heterocycles 1991, 32, 1879-1895.
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