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Volumn 54, Issue 6, 1997, Pages 685-693

Modifying the in vitro accumulation of BMS181321, a technetium-99m-nitroimidazole, with unlabelled nitroaromatics

Author keywords

2 Nitroimidazole; Bioreductive; BMS181321; CHO cells; Diagnosis; Hypoxia

Indexed keywords

ETANIDAZOLE; METRONIDAZOLE; MISONIDAZOLE; NF 167; NITROIMIDAZOLE DERIVATIVE; OXO[3,3,9,9 TETRAMETHYL 1 (2 NITRO 1H IMIDAZOL 1 YL) 4,8 DIAZAUNDECANE 2,10 DIONEDIOXIMATO]TECHNETIUM TC 99M; RP 8979; TINIDAZOLE; UNCLASSIFIED DRUG;

EID: 0343488583     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(97)00222-0     Document Type: Article
Times cited : (12)

References (26)
  • 1
    • 0028632781 scopus 로고
    • Clinical evaluation of nitroimidazoles as modifiers of hypoxia in solid tumors
    • Overgaard J, Clinical evaluation of nitroimidazoles as modifiers of hypoxia in solid tumors. Oncol Res 6: 509-518, 1994.
    • (1994) Oncol Res , vol.6 , pp. 509-518
    • Overgaard, J.1
  • 3
    • 0027141149 scopus 로고
    • Oxygen in human tumors: Correlations between methods of measurement and response to therapy
    • Stone HB, Brown JM, Phillips TL and Sutherland RM, Oxygen in human tumors: Correlations between methods of measurement and response to therapy. Radiat Res 136: 422-434, 1993.
    • (1993) Radiat Res , vol.136 , pp. 422-434
    • Stone, H.B.1    Brown, J.M.2    Phillips, T.L.3    Sutherland, R.M.4
  • 4
    • 0018635742 scopus 로고
    • Hypoxic sensitizers - Implications for radiation therapy
    • Chapman JD, Hypoxic sensitizers - Implications for radiation therapy. N Engl J Med 301: 1429-1432, 1979.
    • (1979) N Engl J Med , vol.301 , pp. 1429-1432
    • Chapman, J.D.1
  • 7
    • 0025870484 scopus 로고
    • Radioiodinated 1-(5-iodo-5-deoxy-β-D-arabinofuranosyl)-2-nitroimidazole (iodoazomycin arabinoside: IAZA): A novel marker of tissue hypoxia
    • Mannan RH, Somayaji VV, Lee J, Mercer JR, Chapman JD and Wiebe LI, Radioiodinated 1-(5-iodo-5-deoxy-β-D-arabinofuranosyl)-2-nitroimidazole (iodoazomycin arabinoside: IAZA): A novel marker of tissue hypoxia. J Nucl Med 32: 1764-1770, 1991.
    • (1991) J Nucl Med , vol.32 , pp. 1764-1770
    • Mannan, R.H.1    Somayaji, V.V.2    Lee, J.3    Mercer, J.R.4    Chapman, J.D.5    Wiebe, L.I.6
  • 8
    • 0028167554 scopus 로고
    • TcO(PnAO-1-(2-nitroimidazole)) [BMS181321], a new technetium-containing nitroimidazole complex for imaging hypoxia: Synthesis, characterization, and xanthine oxidase-catalyzed reduction
    • Linder KE, Chan YW, Cyr JE, Malley MF, Nowotnik DP and Nunn AD, TcO(PnAO-1-(2-nitroimidazole)) [BMS181321], a new technetium-containing nitroimidazole complex for imaging hypoxia: Synthesis, characterization, and xanthine oxidase-catalyzed reduction. J Med Chem 37: 9-17, 1994.
    • (1994) J Med Chem , vol.37 , pp. 9-17
    • Linder, K.E.1    Chan, Y.W.2    Cyr, J.E.3    Malley, M.F.4    Nowotnik, D.P.5    Nunn, A.D.6
  • 9
    • 0028023027 scopus 로고
    • Kinetics of a putative hypoxic tissue marker, technetium-99m-nitroimidazole (BMS181321), in normoxic, hypoxic, ischemic, and stunned myocardium
    • Kusuoka H, Hashimoto K, Fukuchi K and Nishimura T, Kinetics of a putative hypoxic tissue marker, technetium-99m-nitroimidazole (BMS181321), in normoxic, hypoxic, ischemic, and stunned myocardium. J Nucl Med 35: 1371-1376, 1994.
    • (1994) J Nucl Med , vol.35 , pp. 1371-1376
    • Kusuoka, H.1    Hashimoto, K.2    Fukuchi, K.3    Nishimura, T.4
  • 11
    • 0030162585 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of technetium-99m-labelled 2-nitroimidazole (BMS181321) as a marker of tumor hypoxia
    • Ballinger JR, Wan Min Kee J and Rauth AM, In vitro and in vivo evaluation of technetium-99m-labelled 2-nitroimidazole (BMS181321) as a marker of tumor hypoxia. J Nucl Med 37: 1023-1031, 1996.
    • (1996) J Nucl Med , vol.37 , pp. 1023-1031
    • Ballinger, J.R.1    Wan Min Kee, J.2    Rauth, A.M.3
  • 12
    • 0027182896 scopus 로고
    • Bioreductive metabolism of AF-2 [2-(2-furyl)-3-(5-nitro-furyl)acrytamide] combined with 2-nitroimidazoles
    • Koch CJ, Giandomenico AR and Iyengar CWL, Bioreductive metabolism of AF-2 [2-(2-furyl)-3-(5-nitro-furyl)acrytamide] combined with 2-nitroimidazoles. Biochem Pharmacol 46: 1029-1036, 1993.
    • (1993) Biochem Pharmacol , vol.46 , pp. 1029-1036
    • Koch, C.J.1    Giandomenico, A.R.2    Iyengar, C.W.L.3
  • 13
    • 0343047075 scopus 로고
    • The reductive activation of nitroimidazoles; modification by oxygen and other redox-active molecules in cellular systems
    • (Eds. Adams GE, Breccia A, Fielden EM and Wardman P), Plenum Press, New York
    • Koch CJ, The reductive activation of nitroimidazoles; Modification by oxygen and other redox-active molecules in cellular systems. In: Selective Activation of Drugs by Redox Processes (Eds. Adams GE, Breccia A, Fielden EM and Wardman P), pp. 237-247-Plenum Press, New York, 1991.
    • (1991) Selective Activation of Drugs by Redox Processes , pp. 237-247
    • Koch, C.J.1
  • 14
    • 0018945269 scopus 로고
    • An experimental and analytical study of oxygen depletion in stirred cell suspensions
    • Whillans DW and Rauth AM, An experimental and analytical study of oxygen depletion in stirred cell suspensions. Radiat Res 84: 97-114, 1980.
    • (1980) Radiat Res , vol.84 , pp. 97-114
    • Whillans, D.W.1    Rauth, A.M.2
  • 15
    • 0018116095 scopus 로고
    • Differences in the toxicity and metabolism of the 2-nitroimidazole misonidazole (Ro-07-0582) in HeLa and Chinese hamster ovary cells
    • Taylor YC and Rauth AM, Differences in the toxicity and metabolism of the 2-nitroimidazole misonidazole (Ro-07-0582) in HeLa and Chinese hamster ovary cells. Cancer Res 38: 2745-2752, 1978.
    • (1978) Cancer Res , vol.38 , pp. 2745-2752
    • Taylor, Y.C.1    Rauth, A.M.2
  • 16
    • 84872846883 scopus 로고
    • Reduction potentials of one-electron couples involving free radicals in aqueous solutions
    • Wardman P, Reduction potentials of one-electron couples involving free radicals in aqueous solutions. J Physic Chem Ref Data 18: 1637-1755, 1989.
    • (1989) J Physic Chem Ref Data , vol.18 , pp. 1637-1755
    • Wardman, P.1
  • 17
    • 0026016558 scopus 로고
    • The reduction potential of benzyl viologen: An important reference compound for oxidant/radical redox couples
    • Wardman P, The reduction potential of benzyl viologen: An important reference compound for oxidant/radical redox couples. Free Radic Res Commun 14: 57-67, 1991.
    • (1991) Free Radic Res Commun , vol.14 , pp. 57-67
    • Wardman, P.1
  • 18
    • 0016382599 scopus 로고
    • A comparison of the effectiveness of NF-167 and metronidazole as hypoxic cell sensitizers of KHT tumor cells in vitro
    • Thomson JE and Rauth AM, A comparison of the effectiveness of NF-167 and metronidazole as hypoxic cell sensitizers of KHT tumor cells in vitro. Radiat Res 60: 489-500, 1974.
    • (1974) Radiat Res , vol.60 , pp. 489-500
    • Thomson, J.E.1    Rauth, A.M.2
  • 19
    • 0022995459 scopus 로고
    • Measurement of low levels of oxygen and their effect on respiration in cell suspensions maintained in an open system
    • Marshall RS, Koch CJ and Rauth AM, Measurement of low levels of oxygen and their effect on respiration in cell suspensions maintained in an open system. Radiat Res 108: 91-101, 1986.
    • (1986) Radiat Res , vol.108 , pp. 91-101
    • Marshall, R.S.1    Koch, C.J.2    Rauth, A.M.3
  • 20
    • 0006754130 scopus 로고
    • Characterization and subcellular distribution of a novel nitroimidazole complex in the heart
    • Jayatilak PG, Chan YW, Patel BP, Wen M-L and Rumsey WL, Characterization and subcellular distribution of a novel nitroimidazole complex in the heart. J Nucl Med 35: 152P, 1994.
    • (1994) J Nucl Med , vol.35
    • Jayatilak, P.G.1    Chan, Y.W.2    Patel, B.P.3    Wen, M.-L.4    Rumsey, W.L.5
  • 23
    • 0023248351 scopus 로고
    • Enhanced misonidazole binding in the presence of AF-2
    • Olive PL, Enhanced misonidazole binding in the presence of AF-2, Radiat Res 109: 490-499, 1987.
    • (1987) Radiat Res , vol.109 , pp. 490-499
    • Olive, P.L.1
  • 24
    • 0017069834 scopus 로고
    • Oxygen inhibition of nitroreductase: Electron transfer from nitro-radical anions to oxygen
    • Wardman P and Clarke ED, Oxygen inhibition of nitroreductase: Electron transfer from nitro-radical anions to oxygen. Biochem Biophys Res Commun 69: 942-949, 1976.
    • (1976) Biochem Biophys Res Commun , vol.69 , pp. 942-949
    • Wardman, P.1    Clarke, E.D.2
  • 26
    • 0029922596 scopus 로고    scopus 로고
    • Diffusion of nitroimidazoles in V79 multicellular membranes, an in vitro model for the extravascular compartment of tumours
    • Cowan DSM, Hicks KO and Wilson WR, Diffusion of nitroimidazoles in V79 multicellular membranes, an in vitro model for the extravascular compartment of tumours. Br J Cancer 74 (Suppl 27): S28-S31, 1996.
    • (1996) Br J Cancer , vol.74 , Issue.SUPPL. 27
    • Cowan, D.S.M.1    Hicks, K.O.2    Wilson, W.R.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.