Synthesis and analgesic activity of some deaza derivatives of anpirtoline

Archiv der Pharmazie

Volumn 332, Issue 1, 1999, Pages 13-18

  Rádl, Stanislav ^a   Hezky, Petr ^a   Proška, Jan ^a   Krejcí, Ivan ^a  

^a Research Institute of Pharmacy and Biochemistry Prague   (Czech Republic)

Author keywords

4 phenylsulfanyl piperidines; 5 HT(1A) receptor ligands; 5 HT(1B) receptor ligands; Analgesic activity; Anpirtoline analogs

Indexed keywords

ANALGESIC AGENT; ANPIRTOLINE; ANPIRTOLINE DERIVATIVE; FLUPIRTINE; SEROTONIN 1A RECEPTOR; SEROTONIN 1B RECEPTOR; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ARTICLE; BINDING AFFINITY; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ORAL DRUG ADMINISTRATION; PRIORITY JOURNAL; REACTION ANALYSIS;

ANALGESICS, NON-NARCOTIC; ANIMALS; ESCAPE REACTION; HIPPOCAMPUS; MALE; MICE; PAIN MEASUREMENT; PIPERIDINES; PYRIDINES; RADIOLIGAND ASSAY; RATS; REACTION TIME; RECEPTOR, SEROTONIN, 5-HT1B; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN AGONISTS;

EID: 0343413562     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1521-4184(19991)332:1<13::AID-ARDP13>3.0.CO;2-L     Document Type: Article

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