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Volumn 37, Issue 39, 1996, Pages 7155-7158

7-Carbon mimics of D-glucose and L-fucose: Activation of 6R-, and inactivation of 6S-, -6C-methylglucose of glycogen synthase: Inhibition of glucokinase and/or glucose-6-phosphatase

Author keywords

[No Author keywords available]

Indexed keywords

CARBOHYDRATE DERIVATIVE; GLUCOKINASE; GLUCOSE 6 PHOSPHATASE; GLYCOGEN SYNTHASE; GLYCOSIDE;

EID: 0342683712     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4039(96)01565-1     Document Type: Article
Times cited : (20)

References (25)
  • 1
    • 0026654870 scopus 로고
    • 1. Winchester, B., Fleet, G. W. J., Glycobiology, 1992, 2, 199; Jacob, G. S., Bryant, M. L., Prospect. Drug Discovery Des., 1993, 1, 211.
    • (1992) Glycobiology , vol.2 , pp. 199
    • Winchester, B.1    Fleet, G.W.J.2
  • 7
    • 0028360180 scopus 로고
    • 6. Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Orchard, M. G., Fleet, G. W. J., Oikonomakos, N. G., Leonidas, D. D., Kontou, M., Papageoriouo, A., Biochemistry, 1994, 33, 5745; Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Fleet, G. W. J., Oikonomakos, N. G., Kontou, M., Zographos, S. E., Acta Cryst. Sect. D, 1995, 51, 458; Board, M., Bollen, M., Stalmans, W., Kim, Y., Fleet, G. W. J., Johnson, L. N., Biochem. J., 1995, 311, 845; Bichard, C. J. F., Mitchell, E. P., Wormald, M. R., Watson, K. A., Johnson, L. N., Zographos, S. E., Koutra, D. D., Oikonomakos, N. G., Fleet, G. W. J., Tetrahedron Lett., 1995, 36, 2145.
    • (1994) Biochemistry , vol.33 , pp. 5745
    • Watson, K.A.1    Mitchell, E.P.2    Johnson, L.N.3    Son, J.C.4    Bichard, C.J.F.5    Orchard, M.G.6    Fleet, G.W.J.7    Oikonomakos, N.G.8    Leonidas, D.D.9    Kontou, M.10    Papageoriouo, A.11
  • 8
    • 0000119906 scopus 로고
    • 6. Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Orchard, M. G., Fleet, G. W. J., Oikonomakos, N. G., Leonidas, D. D., Kontou, M., Papageoriouo, A., Biochemistry, 1994, 33, 5745; Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Fleet, G. W. J., Oikonomakos, N. G., Kontou, M., Zographos, S. E., Acta Cryst. Sect. D, 1995, 51, 458; Board, M., Bollen, M., Stalmans, W., Kim, Y., Fleet, G. W. J., Johnson, L. N., Biochem. J., 1995, 311, 845; Bichard, C. J. F., Mitchell, E. P., Wormald, M. R., Watson, K. A., Johnson, L. N., Zographos, S. E., Koutra, D. D., Oikonomakos, N. G., Fleet, G. W. J., Tetrahedron Lett., 1995, 36, 2145.
    • (1995) Acta Cryst. Sect. D , vol.51 , pp. 458
    • Watson, K.A.1    Mitchell, E.P.2    Johnson, L.N.3    Son, J.C.4    Bichard, C.J.F.5    Fleet, G.W.J.6    Oikonomakos, N.G.7    Kontou, M.8    Zographos, S.E.9
  • 9
    • 0028805440 scopus 로고
    • 6. Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Orchard, M. G., Fleet, G. W. J., Oikonomakos, N. G., Leonidas, D. D., Kontou, M., Papageoriouo, A., Biochemistry, 1994, 33, 5745; Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Fleet, G. W. J., Oikonomakos, N. G., Kontou, M., Zographos, S. E., Acta Cryst. Sect. D, 1995, 51, 458; Board, M., Bollen, M., Stalmans, W., Kim, Y., Fleet, G. W. J., Johnson, L. N., Biochem. J., 1995, 311, 845; Bichard, C. J. F., Mitchell, E. P., Wormald, M. R., Watson, K. A., Johnson, L. N., Zographos, S. E., Koutra, D. D., Oikonomakos, N. G., Fleet, G. W. J., Tetrahedron Lett., 1995, 36, 2145.
    • (1995) Biochem. J. , vol.311 , pp. 845
    • Board, M.1    Bollen, M.2    Stalmans, W.3    Kim, Y.4    Fleet, G.W.J.5    Johnson, L.N.6
  • 10
    • 0028955885 scopus 로고
    • 6. Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Orchard, M. G., Fleet, G. W. J., Oikonomakos, N. G., Leonidas, D. D., Kontou, M., Papageoriouo, A., Biochemistry, 1994, 33, 5745; Watson, K. A., Mitchell, E. P., Johnson, L. N., Son, J. C., Bichard, C. J. F., Fleet, G. W. J., Oikonomakos, N. G., Kontou, M., Zographos, S. E., Acta Cryst. Sect. D, 1995, 51, 458; Board, M., Bollen, M., Stalmans, W., Kim, Y., Fleet, G. W. J., Johnson, L. N., Biochem. J., 1995, 311, 845; Bichard, C. J. F., Mitchell, E. P., Wormald, M. R., Watson, K. A., Johnson, L. N., Zographos, S. E., Koutra, D. D., Oikonomakos, N. G., Fleet, G. W. J., Tetrahedron Lett., 1995, 36, 2145.
    • (1995) Tetrahedron Lett. , vol.36 , pp. 2145
    • Bichard, C.J.F.1    Mitchell, E.P.2    Wormald, M.R.3    Watson, K.A.4    Johnson, L.N.5    Zographos, S.E.6    Koutra, D.D.7    Oikonomakos, N.G.8    Fleet, G.W.J.9
  • 13
    • 1542728688 scopus 로고
    • 8. Kitihara, T., Ogawa, T., Naganuma, T., Matsui, M., Agr, Biol. Chem., 1974, 38, 2189; Bashyal, B. P., Chow, H.-F., Fleet, G. W. J., Tetrahedron, 1987, 43, 423.
    • (1987) Tetrahedron , vol.43 , pp. 423
    • Bashyal, B.P.1    Chow, H.-F.2    Fleet, G.W.J.3
  • 16
    • 85030274772 scopus 로고    scopus 로고
    • note
    • 2O + dioxan): 19.3 (q, Me), 19.5 (q, Me), 65.0, 65.1, 70.4, 70.6, 72.3, 73.8, 74.0, 75.1, 76.8, 78.5 (10 x d, C-2, C-3, C-4, C-5, C-6 α and β), 92.8 (d, C-1α), 96.9 (d, C-1β).
  • 17
    • 85030273399 scopus 로고    scopus 로고
    • note
    • 11. The details of the crystal structures of 11 and 13 will be presented in the full paper.
  • 18
    • 85030280244 scopus 로고    scopus 로고
    • note
    • 2O + dioxan): 14.7 (q, Me), 14.8 (q, Me), 66.1, 70.5, 70.7, 71.2, 72.8, 72.9, 74.0, 75.7, 77.7 (9 x d, C-2, C-3, C-4, C-5, C-6 α and β), 91.9 (d, C-1α), 96.0 (d, C-1β).
  • 21
    • 0018977855 scopus 로고
    • 15. Assay for glycogen synthase: Dopere, F., Vanstapel, F., Stalmans, W., Eur. J. Biochem., 1980, 104, 137. Assay for Glc-6-P: Lowry, O. H., Passonneau, J. V., A flexible system of enzymatic analysis, Academic Press, New York, pp. 71-77, 1972. Assay for glucokinase: Davidson A. L., Arion, W. J., Arch. Biochem. Biophys., 1987, 253, 156. Assay for Glc-6-Pase: Burchell, A., Hume, R., Burchell, B., Clin. Chim. Acta, 1988, 173, 183.
    • (1980) Eur. J. Biochem. , vol.104 , pp. 137
    • Dopere, F.1    Vanstapel, F.2    Stalmans, W.3
  • 22
    • 0018977855 scopus 로고
    • Academic Press, New York
    • 15. Assay for glycogen synthase: Dopere, F., Vanstapel, F., Stalmans, W., Eur. J. Biochem., 1980, 104, 137. Assay for Glc-6-P: Lowry, O. H., Passonneau, J. V., A flexible system of enzymatic analysis, Academic Press, New York, pp. 71-77, 1972. Assay for glucokinase: Davidson A. L., Arion, W. J., Arch. Biochem. Biophys., 1987, 253, 156. Assay for Glc-6-Pase: Burchell, A., Hume, R., Burchell, B., Clin. Chim. Acta, 1988, 173, 183.
    • (1972) A Flexible System of Enzymatic Analysis , pp. 71-77
    • Lowry, O.H.1    Passonneau, J.V.2
  • 23
    • 0023154010 scopus 로고
    • 15. Assay for glycogen synthase: Dopere, F., Vanstapel, F., Stalmans, W., Eur. J. Biochem., 1980, 104, 137. Assay for Glc-6-P: Lowry, O. H., Passonneau, J. V., A flexible system of enzymatic analysis, Academic Press, New York, pp. 71-77, 1972. Assay for glucokinase: Davidson A. L., Arion, W. J., Arch. Biochem. Biophys., 1987, 253, 156. Assay for Glc-6-Pase: Burchell, A., Hume, R., Burchell, B., Clin. Chim. Acta, 1988, 173, 183.
    • (1987) Arch. Biochem. Biophys. , vol.253 , pp. 156
    • Davidson, A.L.1    Arion, W.J.2
  • 24
    • 0023890340 scopus 로고
    • 15. Assay for glycogen synthase: Dopere, F., Vanstapel, F., Stalmans, W., Eur. J. Biochem., 1980, 104, 137. Assay for Glc-6-P: Lowry, O. H., Passonneau, J. V., A flexible system of enzymatic analysis, Academic Press, New York, pp. 71-77, 1972. Assay for glucokinase: Davidson A. L., Arion, W. J., Arch. Biochem. Biophys., 1987, 253, 156. Assay for Glc-6-Pase: Burchell, A., Hume, R., Burchell, B., Clin. Chim. Acta, 1988, 173, 183.
    • (1988) Clin. Chim. Acta , vol.173 , pp. 183
    • Burchell, A.1    Hume, R.2    Burchell, B.3
  • 25
    • 85030273484 scopus 로고    scopus 로고
    • note
    • 16. Support has been received for a Graduate Studentship from GlaxoWellcome and Post-doctoral fellowships from EPSRC and European Community contract BIO2 CT94 3025


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