A facile preparation of α-amino-β-methoxydiazines through, the lithianation followed by amination

Bulletin of the Korean Chemical Society

Volumn 17, Issue 9, 1996, Pages 868-869

  Lee II, Jung ^a   Cho, Sung Hye ^a  

^a Chung Ang University   (South Korea)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0342620594     PISSN: 02532964     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (13)

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2. Botta, M.; De Angelis, F.; Nicoletti, R. J. Heterocycl. Chem. 1979, 16, 193.
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9. Ple, N.; Turck, A.; Couture, K.; Queguiner, G. Tetrahedron 1994, 50, 10299.
10. Ramadas, K.; Srinivasan, N. Synth. Commun. 1992, 22, 3189.
11. 2,4-Dimethoxypyrimidine (1a) and 4,6-dimethoxypyrimidine (1b) were easily prepared from the corresponding chlorodiazine with sodium methylate: see Mattson, R. J.; Sloan, C. P. J. Org. Chem. 1990, 55, 3410.
12. 3-Methoxypyridazine (2a) and 3,6-dimethoxypyridazine (2 b) were prepared from 3,6-dichloropyridazine: see Coad, P.; Coad, R. A.; Hyepock, J. J. Org. Chem. 1964, 29, 1751.
13. Prystas, M.; Sorm, F. Collect. Czech. Chem. Commun. 1966, 31, 3990.