An Efficient Acid-Catalysed 5-endo-dig Cyclisation Method for Pyrrole Synthesis

Synlett

Volumn , Issue 14, 2003, Pages 2258-2260

  Knight, David W ^a   Sharland, Christopher M ^a  

^a CARDIFF UNIVERSITY   (United Kingdom)

Author keywords

5 endo dig cyclisation; Pyrrole; ynyl hydroxy amino esters

Indexed keywords

ALPHA AMINO ACID; ESTER DERIVATIVE; PYRROLE DERIVATIVE; TIN DERIVATIVE;

ARTICLE; CATALYSIS; CHEMICAL REACTION; CYCLIZATION; ELIMINATION REACTION; OXIDATION; POLYMERIZATION; SYNTHESIS;

EID: 0242659863     PISSN: 09365214     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-2003-42101     Document Type: Article

References (11)

1. Knight, D. W.; Redfern, A. L.; Gilmore, J. J. Chem. Soc., Perkin Trans. 1 2002, 622.
2. For an excellent overview, see: Li, J. J.; Gribble, W. Palladium in Heterocyclic Chemistry, Tetrahedron Organic Chemistry Series, Vol. 20; Pergamon Press: Oxford, 2000.
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7. Gridley, J. J.; Coogan, M. P.; Knight, D. W.; Malik, K. M. A.; Sharland, C. M.; Singkhonrat, J.; Williams, S. M. Chem. Commun. 2003, 2550.
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11. For a review of electrophile-driven 5-endo cyclisation methods, see: Knight, D. W. In Progress in Heterocyclic Chemistry; Gribble, G. W.; Gillchrist, T. L., Eds.; 2002, Vol. 14.