Synthesis and biological evaluation of substituted quinolines: Potential treatment of protozoal and retroviral co-infections

Bioorganic and Medicinal Chemistry

Volumn 11, Issue 23, 2003, Pages 5013-5023

  Fakhfakh, Mohammed A ^a   Fournet, Alain ^a,b   Prina, Eric ^c   Mouscadet, Jean François ^d   Franck, Xavier ^a   Hocquemiller, Reynald ^a   Figadère, Bruno ^a  

^a UNIVERSITÉ PARIS SACLAY   (France)

^b INSTITUT DE RECHERCHE POUR LE DÉVELOPPEMENT   (France)

^c INSTITUT PASTEUR   (France)

^d INSTITUT GUSTAVE ROUSSY   (France)

Author keywords

[No Author keywords available]

Indexed keywords

1 BROMO 2 (2 QUINOLYL)ETHYLENE; 1 QUINOL 2 YLPROPAN 1 OL; 1,1 DIBROMO 2 (2 QUINOLYL)ETHYLENE; 2 ETHYNYLQUINOLINE; 2 TRIMETHYLSILYLETHYNYLQUINOLINE; 2 VINYLQUINOLINE; ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; ANTIPROTOZOAL AGENT; ANTIRETROVIRUS AGENT; MEGLUMINE ANTIMONATE; NIFURTIMOX; QUINOLINE DERIVATIVE; SURAMIN; TUMOR NECROSIS FACTOR ALPHA; UNCLASSIFIED DRUG;

AFRICAN TRYPANOSOMIASIS; ANIMAL CELL; ANIMAL MODEL; ANTIVIRAL ACTIVITY; ARTICLE; BONE MARROW CELL; CHAGAS DISEASE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFICACY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; FEMALE; FEMUR; HAMSTER; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; IC 50; LEISHMANIA; MOUSE; MOUSE STRAIN; NONHUMAN; PERITONEUM MACROPHAGE; PROTOZOAL INFECTION; RETROVIRUS INFECTION; SKIN LEISHMANIASIS; STRUCTURE ACTIVITY RELATION; T CELL LEUKEMIA; TIBIA; VISCERAL LEISHMANIASIS;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0242266523     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2003.09.007     Document Type: Article

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