Synthesis, characterization and in vitro antifungal evaluation of tetrahydropyrazolo[1,5-c]quinazolines

Heterocyclic Communications

Volumn 9, Issue 2, 2003, Pages 153-160

  Insuasty, Braulio ^a   Torres, Harlem ^a   Quiroga, Jairo ^a   Abonía, Rodrigo ^a   Nogueras, Manuel ^b   Sánchez, Adolfo ^b   Sortino, Maximiliano ^c   Zacchino, Susana ^c   Low, John ^d  

^a UNIVERSIDAD DEL VALLE   (Colombia)

^b UNIVERSITY OF JAÉN   (Spain)

^c UNIVERSIDAD NACIONAL DE ROSARIO   (Argentina)

^d UNIVERSITY OF ABERDEEN   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 NITROBENZALDEHYDE; ANTIFUNGAL AGENT; BENZALDEHYDE DERIVATIVE; QUINAZOLINE DERIVATIVE; TETRAHYDROPYRAZOLO[1,5 C]QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; X RAY DIFFRACTION;

EID: 0142025470     PISSN: 07930283     EISSN: None     Source Type: Journal    
DOI: 10.1515/HC.2003.9.2.153     Document Type: Article

References (19)

1. D. W. Fry, A. J. Kraker, A. McMichael, L. A. Ambroso, J. M. Nelson, W. R. Leopold, R. W. Connors, A. L. Bridges, Science, 265, 1093 (1994).
2. a) Dictionary of Natural Products, Buckingham J., ed., Chapman and Hall, London (1994);
3. S. Johne, Pharmazie, 36, 583 (1981).
4. a) G. Daidone, B. Maggio, D. Raffa, S. Plescia, M. L. Bajardi, A. Caruso, V. M. C. Cuttuli, M. Amico-Roxas, Eur. J. Med. Chem., 29, 707 (1994);
5. b) A. A. Backhit, M. A. Khalil, Pharmazie, 53, 539 (1998);
6. c) R. Argarwal, C. Singli, N. S. Mishara, Ind. Drugs, 25, 185 (1988).
7. B. Pramella, E. Rajanarender and A. K. Murty, Ind. J. Heterocyclic Chem., 2, 115 (1992).
8. M. Shyimad, R. Kalsi, K. S. Dixit and J. P. Barthwal, Arzneim-Fosch. Drug Res., 41, 514 (1991).
9. Kh. M. Shakhidoyator, E. O. Eripor, L. M. Yun, M. Yamankulov, Ch. Kadyrov, Fungitsidy, 66 (1980); Chem. Abstr.: 94, 192253 (1981).
10. Kh. M. Shakhidoyator, E. O. Eripor, L. M. Yun, M. Yamankulov, Ch. Kadyrov, Fungitsidy, 66 (1980); Chem. Abstr.: 94, 192253 (1981).
11. a) V. Colotta, D. Catarzi, F. Varano, G. Filacchioni, L. Cecchi, A. Galli, C. Costagli, J. Med. Chem., 39, 2915 (1996);
12. b)F. Varano, D. Catarzi, V. Colotta, G. Filacchioni, A. Galli, C. Costagli, V. Carla, V. J. Med. Chem., 45, 1035 (2002).
13. a) C. Engler, A. Engler, Chem. Ber., 35, 4061 (1902);
14. b) R. P. Barnes, J. H. Graham, M. A. S. Qureshi, J. Org. Chem., 28, 2890 (1963).
15. a) J. N Low, J. Cobo, M. Nogueras, A. Sánchez, H. Torres, B. Insuasty, Acta Cryst., C58, 305 (2002); L. McQuaid, E. Smith, K. South, C. H. Smith, D. Schoepp, R. True, D. Calligaro, P. O'Malley, D. Lodge and P. Ornstein, J. Med. Chem., 35, 3319 (1992).
16. a) J. N Low, J. Cobo, M. Nogueras, A. Sánchez, H. Torres, B. Insuasty, Acta Cryst., C58, 305 (2002); L. McQuaid, E. Smith, K. South, C. H. Smith, D. Schoepp, R. True, D. Calligaro, P. O'Malley, D. Lodge and P. Ornstein, J. Med. Chem., 35, 3319 (1992).
17. L. A. Mitscher, R. P. Leu, M. S. Bathala, W. N. Wu, J. L. Beal, Lloydia, 35, 157 (1972).
18. L. Wright, E. Scott, S. Gorman, J. Antimicrob. Chemother., 12, 317 (1983).
19. S. A. Zacchino, S. N. López, G. Pezzenati, R. L. Furlán, C. B. Santecchia, L. Muñoz, F. A. Giannini, A. M. Rodríguez, R. D. Enriz, J. Nat. Prod., 63, 1353 (1999).