Application of the Thorpe-Ziegler reaction for the synthesis of functionalized thiophenes, thienopyrilnidines, and thienotriazines

Russian Chemical Bulletin

Volumn 51, Issue 5, 2002, Pages 789-793

  Ryndina, S A ^a   Kadushkin, A V ^a   Solov'eva, N P ^b   Granik, V G ^a  

^a Organic Intermediates and Dyes Institute   (Russian Federation)

^b Center for Drug Chemistry   (Russian Federation)

Author keywords

1,2,3 triazines; Enamines; Pyrimidines; The Thorpe Ziegler cyclization; Thiophenes

Indexed keywords

1,2,3 TRIAZINE DERIVATIVE; DICARBOXYLIC ACID DERIVATIVE; PYRIMIDINE DERIVATIVE; THIOPHENE DERIVATIVE;

ARTICLE; CYCLIZATION; SYNTHESIS;

EID: 0141832935     PISSN: 10665285     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1016072414801     Document Type: Article

References (15)

1. F. S. Babichev, Yu. A. Sharanin, V. P. Litvinov, V. K. Promonenkov, and Yu. M. Volovenko, Vnutrimolekulyarnoe vzaimodeistvie nitril'noi i CH-, OH- i SH-grupp [Intramolecular Interactions of a Nitrile Group with CH, OH, and SH Groups], Naukova Dumka, Kiev, 1985, 200 pp. (in Russian).
2. V. G. Granik, A. V. Kadushkin, and J. Liebscher, Adv. Heterocycl. Chem., 1998, 72, 79.
3. S. A. Ryndina, A. V. Kadushkin, N. P. Solov'eva, and V.G. Granik, Khim. Geterotsikl. Soedinenii, 2000, 1643 [Chem. Heterocycl. Compd., 2000, 26, 1409 (Engl. Transl.)].
4. S. A. Ryndina, A. V. Kadushkin, N. P. Solov'eva, and V.G. Granik, Khim. Geterotsikl. Soedinenii, 2000, 1643 [Chem. Heterocycl. Compd., 2000, 26, 1409 (Engl. Transl.)].
5. K. Saito, S. Kambe, A. Sakurai, and H. Midorikawa, Synthesis, 1982, 1056.
6. S. F. Martin and D. R. Moore, Tetrahedron Lett., 1976, 4459.
7. 13C NMR-spectra, Reine Heyden and Son, Ltd, London - New York, 1976, p. 37.
8. A. V. Kadushkin, I. N. Nesterova, T. V. Golovko, I. S. Nikolaeva, T. V. Pushkina, A. N. Fomina, A. S. Sokolova, V. N. Chernov, and V. G. Granik, Khim.-Farm. Zhurn., 1990, 24, 18 [Pharm. Chem. J., 1990, 24, 875 (Engl. Transl.)].
9. A. V. Kadushkin, I. N. Nesterova, T. V. Golovko, I. S. Nikolaeva, T. V. Pushkina, A. N. Fomina, A. S. Sokolova, V. N. Chernov, and V. G. Granik, Khim.-Farm. Zhurn., 1990, 24, 18 [Pharm. Chem. J., 1990, 24, 875 (Engl. Transl.)].
10. V. G. Granik, A. M. Zhidkova, I. S. Zhivotovskaya, N. P. Solov'eva, and M. K. Polievktov, Zhurn. Org. Khim., 1981, 2421 [J. Org. Chem. USSR, 1981, 17, 2163 (Engl. Transl.)].
11. V. G. Granik, A. M. Zhidkova, I. S. Zhivotovskaya, N. P. Solov'eva, and M. K. Polievktov, Zhurn. Org. Khim., 1981, 2421 [J. Org. Chem. USSR, 1981, 17, 2163 (Engl. Transl.)].
12. A. P. Tamiz, S. X. Cai, Z.-L. Zhou, P.-W. Yuen, R. M. Schelkun, E. R. Whittemore, E. Weber, R. M. Woodward, and J. F. W. Keana, J. Med. Chem., 1999, 42, 3412.
13. B. Leonard, J. Am. Chem. Soc., 1950, 72, 2980.
14. T. Whitehead, J. Am. Chem. Soc., 1955, 77, 5867.
15. A. Bellotti, E. Cogni, A. Baruffuni, G. Pagani, and P. Borgna, Farmaco, Ed. Sci., 1968, 23, 591.