Functional identification of rat atypical β-adrenoceptors by the first β3-selective antagonists, aryloxypropanolaminotetralins

British Journal of Pharmacology

Volumn 117, Issue 3, 1996, Pages 435-442

  Manara, Luciano ^a   Badone, Domenico ^a   Baroni, Marco ^a   Boccardi, Giovanni ^a   Cecchi, Roberto ^a   Croci, Tiziano ^a   Giudice, Antonina ^a   Guzzi, Umberto ^a   Landi, Marco ^a   Le Fur, Gérard ^b  

^a Research Centre Sanofi Midy   (Italy)

^b SANOFI   (France)

Author keywords

Aryloxypropanolaminotetralins; Atypical adrenoceptors; Rat BAT thermogenesis; Rat isolated colon; Selective 3 adrenoceptor antagonists; 3 adrenoceptors

Indexed keywords

1 (2 ETHYLPHENOXY) 3 (1,2,3,4 TETRAHYDRO 1 NAPHTHYLAMINO) 2 PROPANOL OXALATE; 4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID; ALPRENOLOL DERIVATIVE; ARTYLOXYPROPANOLAMINOTETRALIN; BETA 3 ADRENERGIC RECEPTOR; BETA 3 ADRENERGIC RECEPTOR BLOCKING AGENT; BETA ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; ISOPRENALINE; SALBUTAMOL; UNCLASSIFIED DRUG; [[7 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO] 5,6,7,8 TETRAHYDRO 2 NAPHTHYL]OXY]ACETIC ACID ETHYL ESTER;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRONCHODILATATION; BROWN ADIPOSE TISSUE; CHEMICAL STRUCTURE; COLON MOTILITY; GUINEA PIG; HEART ATRIUM CONTRACTILITY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SMOOTH MUSCLE RELAXATION; STEREOCHEMISTRY; TACHYCARDIA; THERMOGENESIS; TRACHEA MUSCLE;

EID: 0141799397     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb15209.x     Document Type: Article

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