Conjugation of poor inhibitors with surface binding groups: a strategy to improve inhibition

Chemical Communications

Volumn 3, Issue 18, 2003, Pages 2328-2329

  Roy, Bidhan C ^a   Hegge, Ryan ^a   Rosendahl, Theresa ^a   Jia, Xiao ^a   Lareau, Rachael ^a   Mallik, Sanku ^a   Srivastava, D K ^a  

^a NORTH DAKOTA STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZENESULFONAMIDE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CONJUGATION; ENZYME INHIBITION;

EID: 0141790840     PISSN: 13597345     EISSN: 1364548X     Source Type: Journal    
DOI: 10.1039/b305179j     Document Type: Article

References (19)

1. H. S. Park, Q. Lin, A. D. Hamilton, Proc. Natl. Acad. Sci. USA, 2002, 99, 5105
2. Y. Wei, G. L. McLendon, A. D. Hamilton, M. A. Case, C. B. Purring, H. Park, C. S. Lee, T. Yu, Chem. Commun. 2001, 1580
3. H. Takashima, S. Shinkai, I. Hamachi, Chem. Commun. 1999, 2345
4. L. L. Kissling, J. E. Gestwicki, L. E. Strong, Curr. Opin. Chem. Biol. 2000, 4, 696
5. A. G. Cochran, Chem. Biol. 2000, 7, R85
6. M. A. Fazal, B. C. Roy, S. Sun, S. Mallik, K. A. Rodgers, J. Am. Chem. Soc. 2001, 123, 6283
7. C. T. Supuran, A. Scozzafava, A. Casini, Med. Chem. Res. Rev. 2003, 23, 146
8. E. Kimura, Acc. Chem. Res. 2001, 34, 171
9. A. Scozzafava, C. T. Supuran, Bioorg. Med. Chem. Lett. 2002, 12, 1551
10. A. Scozzafava, C. T. Supuran, J. Med. Chem. 2002, 47, 284
11. A. Scozzafava, L. Menabouni, F. Manicone, C. T. Supuran, J. Med. Chem. 2002, 45, 1466
12. C. A. Blasie, J. M. Berg, Biochemistry, 2002, 41, 15068
13. W. F. DeGrado, L. DiCostanzo, S. Geremia, A. Lombardi, V. Pavone, L. Ranadaccio, Angew. Chem. Int. Ed. 2003, 42, 417
14. Z. Q. Tian, P. A. Bartlett, J. Am. Chem. Soc. 1996, 118, 943
15. A. E. Martell and P. M. Smith, Critical Stability Constants, Plenum Press, New York, 1975, vol. 2, pp. 67-68.
16. V. Gaber-Porekar, V. Menart, J. Biochem. Biophys. Methods, 2001, 49, 335
17. B. C. Roy, S. Mallik, J. Org. Chem. 1999, 64, 2969
18. S. Sun, M. A. Fazal, B. C. Roy, S. Mallik, Org. Lett. 2000, 2, 911
19. N. Shirai, Y. Watanabe, Y. Sato, J. Org. Chem. 1990, 55, 2767