Synthesis and fluorescent properties of 6-(4-biphenylyl)-3,9-dihydro-9-oxo-5H-imidazo[1,2-A]purine analogues of acyclovir and ganciclovir

Nucleosides, Nucleotides and Nucleic Acids

Volumn 22, Issue 5-8, 2003, Pages 911-914

  Goslinski, Tomasz ^a   Wenska, Grazyna ^b   Golankiewicz, Bozenna ^a   Balzarini, Jan ^c   De Clercq, Erik ^c  

^a INSTITUTE OF BIOORGANIC CHEMISTRY   (Poland)

^b ADAM MICKIEWICZ UNIVERSITY   (Poland)

^c REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

Author keywords

Acyclovir; Fluorescent properties; Ganciclovir; Tricyclic analogues

Indexed keywords

6 (4 BIPHENYL) 3,9 DIHYDRO 9 OXO 5H IMIDAZO[1,2 A]PURINE; ACICLOVIR DERIVATIVE; BENZENEBORONIC ACID; BORONIC ACID DERIVATIVE; GANCICLOVIR DERIVATIVE; UNCLASSIFIED DRUG;

ABSORPTION SPECTROSCOPY; ANTIVIRAL ACTIVITY; CARBON NUCLEAR MAGNETIC RESONANCE; CELL STRUCTURE; CONFERENCE PAPER; CONTROLLED STUDY; CYTOMEGALOVIRUS; DRUG SYNTHESIS; FLUORESCENCE SPECTROSCOPY; HERPES SIMPLEX VIRUS 1; HERPES SIMPLEX VIRUS 2; HUMAN; HUMAN CELL; LUNG ALVEOLUS CELL; PROTON NUCLEAR MAGNETIC RESONANCE; VARICELLA ZOSTER VIRUS;

ACYCLOVIR; ANTIVIRAL AGENTS; CELL LINE; GANCICLOVIR; HERPESVIRUS 1, HUMAN; HERPESVIRUS 2, HUMAN; HUMANS; IMIDAZOLES; INDICATORS AND REAGENTS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; SPECTROMETRY, FLUORESCENCE; STRUCTURE-ACTIVITY RELATIONSHIP;

CYTOMEGALOVIRUS; HUMAN HERPESVIRUS 1; HUMAN HERPESVIRUS 2; HUMAN HERPESVIRUS 3; LATEOLABRAX JAPONICUS; SIMPLEXVIRUS; TACARIBE VIRUS;

EID: 0141648314     PISSN: 15257770     EISSN: None     Source Type: Journal    
DOI: 10.1081/NCN-120022684     Document Type: Conference Paper

References (6)

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2. Golankiewicz, B.; Ostrowski, T.; Goslinski, T.; Januszczyk, P.; Zeidler, J.; Baranowski, D.; De Clercq, E. Fluorescent tricyclic analogues of acyclovir and ganciclovir. A structure - antiviral activity study. J. Med. Chem. 2001, 44, 4284-4287.
3. Goslinski, T.; Golankiewicz, B.; De Clercq, E.; Balzarini, J. Synthesis and biological activity of strongly fluorescent tricyclic analogues of acyclovir and ganciclovir. J. Med. Chem. 2002, 45, 5052-5057.
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