(R)-3-(N-Methylpyrrolidin-2-ylmethyl)-5-(1,2,3,6-tetrahydropyridin-4-yl) -1H-indole derivatives as high affinity h5-HT1B/1D ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 20, 2003, Pages 3419-3421

  Egle, Ian ^a   MacLean, Neil ^a   Demchyshyn, Lidia ^a   Edwards, Louise ^a   Slassi, Abdelmalik ^a   Tehim, Ashok ^a,b  

^a NPS Pharmaceuticals Inc   (Canada)

^b Memory Pharmaceuticals Corporation   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

INDOLE DERIVATIVE; LIGAND; SEROTONIN 1B RECEPTOR; SEROTONIN 1D RECEPTOR;

ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HUMAN; PHARMACODYNAMICS; STRUCTURE ACTIVITY RELATION;

EID: 0141628365     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00779-0     Document Type: Article

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