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Volumn 58, Issue 9, 2003, Pages 669-676

N-Homolupinanoyl and N-(ω-lupinylthio)alkanoyl derivatives of some tricyclic systems as ligands for muscarinic M1 and M2 receptor subtypes

Author keywords

Muscarinic receptors ligands; N (Homolupinanoyl)phenothiazines; N (tert Aminoalkanoyl)tricyclic systems; N ( lupinylthio)alkanoyl phenothiazines; Quinolizidine derivatives

Indexed keywords

BENZODIAZEPINE DERIVATIVE; BENZYL DERIVATIVE; MUSCARINIC M1 RECEPTOR; MUSCARINIC M2 RECEPTOR; NANOPARTICLE; PHENOTHIAZINE DERIVATIVE;

EID: 0141453205     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(03)00104-6     Document Type: Article
Times cited : (6)

References (26)
  • 1
    • 0030442725 scopus 로고    scopus 로고
    • Muscarinic receptor subtypes and smooth muscle function
    • Eglen R.M., Hedge S.S., Watson N. Muscarinic receptor subtypes and smooth muscle function. Pharmacol. Rev. 48:1996;531-565.
    • (1996) Pharmacol. Rev. , vol.48 , pp. 531-565
    • Eglen, R.M.1    Hedge, S.S.2    Watson, N.3
  • 2
    • 0034676312 scopus 로고    scopus 로고
    • Therapeutic opportunities for muscarinic receptors in the central nervous system
    • Felder C.C., Bymaster F.P., Ward J., DeLapp N. Therapeutic opportunities for muscarinic receptors in the central nervous system. J. Med. Chem. 43:2000;4333-4353.
    • (2000) J. Med. Chem. , vol.43 , pp. 4333-4353
    • Felder, C.C.1    Bymaster, F.P.2    Ward, J.3    DeLapp, N.4
  • 3
    • 0035424943 scopus 로고    scopus 로고
    • Therapeutic opportunities from muscarinic receptor research
    • Eglen R.M., Choppin A., Watson N. Therapeutic opportunities from muscarinic receptor research. Trends Pharmacol. Sci. 22:2001;409-414.
    • (2001) Trends Pharmacol. Sci. , vol.22 , pp. 409-414
    • Eglen, R.M.1    Choppin, A.2    Watson, N.3
  • 4
    • 0035957582 scopus 로고    scopus 로고
    • Neostriatal muscarinic receptor subtypes involved in the generation of tremulous jaw movements in rodents: Implication for cholinergic involvement in Parkinsonism
    • Salamone J.D., Correa M., Carlson B.B., Wisniecki A., Mayorga A.J., Nisenbaum E., Nisenbaum L., Felder C. Neostriatal muscarinic receptor subtypes involved in the generation of tremulous jaw movements in rodents: implication for cholinergic involvement in Parkinsonism. Life Sci. 68:2001;2579-2584.
    • (2001) Life Sci. , vol.68 , pp. 2579-2584
    • Salamone, J.D.1    Correa, M.2    Carlson, B.B.3    Wisniecki, A.4    Mayorga, A.J.5    Nisenbaum, E.6    Nisenbaum, L.7    Felder, C.8
  • 5
    • 0028927110 scopus 로고
    • 2 antagonists as potential drugs for cognitive disorders
    • 2 antagonists as potential drugs for cognitive disorders. Drugs Fut. 20:1995;157-164.
    • (1995) Drugs Fut. , vol.20 , pp. 157-164
    • Doods, H.N.1
  • 7
    • 0028350706 scopus 로고
    • Preparation and pharmacological activities of 10-homolupinanoyl-2-R-phenothiazines
    • Sparatore A., Sparatore F. Preparation and pharmacological activities of 10-homolupinanoyl-2-R-phenothiazines. Farmaco. 49:1994;5-17.
    • (1994) Farmaco , vol.49 , pp. 5-17
    • Sparatore, A.1    Sparatore, F.2
  • 8
    • 0033581641 scopus 로고    scopus 로고
    • Quinolizidinyl derivatives of 5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one as ligands for muscarinic receptors
    • Novelli F., Sparatore A., Tasso B., Sparatore F. Quinolizidinyl derivatives of 5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one as ligands for muscarinic receptors. Bioorg. Med. Chem. Lett. 9:1999;3031-3034.
    • (1999) Bioorg. Med. Chem. Lett. , vol.9 , pp. 3031-3034
    • Novelli, F.1    Sparatore, A.2    Tasso, B.3    Sparatore, F.4
  • 9
    • 84919292820 scopus 로고
    • Tricyclic compounds as selective muscarinic antagonists: Structure-activity relationships and therapeutic implications
    • P. Angeli, U. Gulini, & W. Quaglia. Amsterdam: Elsevier
    • Eberlein W.G., Engel W.W., Hasselbach K.M., Mayer N., Mihm G., Rudolf K., Doods H. Tricyclic compounds as selective muscarinic antagonists: structure-activity relationships and therapeutic implications. Angeli P., Gulini U., Quaglia W. Trends in Receptor Research. 1992;231-249 Elsevier, Amsterdam.
    • (1992) Trends in Receptor Research , pp. 231-249
    • Eberlein, W.G.1    Engel, W.W.2    Hasselbach, K.M.3    Mayer, N.4    Mihm, G.5    Rudolf, K.6    Doods, H.7
  • 10
    • 0141805133 scopus 로고
    • 10-Aminoacylphenothiazines. I. Aminoacetyl and aminopropionyl derivatives
    • Dahlbom R., Ekstrand T. 10-Aminoacylphenothiazines. I. Aminoacetyl and aminopropionyl derivatives. Acta Chem. Scand. 5:1951;102-114.
    • (1951) Acta Chem. Scand. , vol.5 , pp. 102-114
    • Dahlbom, R.1    Ekstrand, T.2
  • 11
    • 0141693577 scopus 로고
    • 10-Aminoacylphenothiazines. II. Aminobutyryl derivatives
    • Dahlbom R., Ekstrand T. 10-Aminoacylphenothiazines. II. Aminobutyryl derivatives. Acta Chem. Scand. 6:1952;1285-1288.
    • (1952) Acta Chem. Scand. , vol.6 , pp. 1285-1288
    • Dahlbom, R.1    Ekstrand, T.2
  • 12
    • 0141470332 scopus 로고
    • The activity of 10-aminoacylphenothiazine, basically substituted derivatives of phenothiazine-10-carboxylic acid, atropine, papaverine and some other spasmolytic drugs against barium and acetylcholine-induced spasms of guinea pig and rat ileum
    • Dahlbom R., Edlund T., Ekstrand T., Lohi A. The activity of 10-aminoacylphenothiazine, basically substituted derivatives of phenothiazine-10-carboxylic acid, atropine, papaverine and some other spasmolytic drugs against barium and acetylcholine-induced spasms of guinea pig and rat ileum. Acta Pharmacol. Toxicol. 9:1953;168-178.
    • (1953) Acta Pharmacol. Toxicol. , vol.9 , pp. 168-178
    • Dahlbom, R.1    Edlund, T.2    Ekstrand, T.3    Lohi, A.4
  • 13
    • 0141805134 scopus 로고
    • Studies on some phenothiazine derivatives
    • Dahlbom R. Studies on some phenothiazine derivatives. Sci. Repts. Ist. Super Sanit. 2:1962;309-319.
    • (1962) Sci. Repts. Ist. Super Sanit. , vol.2 , pp. 309-319
    • Dahlbom, R.1
  • 14
    • 0141805135 scopus 로고
    • Protective effect of phenothiazine derivatives against poisoning by the irreversible cholinesterase inhibitor dimethylamido-ethoxyphosphoryl cyanide (Tabun)
    • Dahlbom R., Diamant H., Edlund T., Ekstrand T., Holmstedt B. Protective effect of phenothiazine derivatives against poisoning by the irreversible cholinesterase inhibitor dimethylamido-ethoxyphosphoryl cyanide (Tabun). Acta Pharmacol. Toxicol. 9:1953;163-167.
    • (1953) Acta Pharmacol. Toxicol. , vol.9 , pp. 163-167
    • Dahlbom, R.1    Diamant, H.2    Edlund, T.3    Ekstrand, T.4    Holmstedt, B.5
  • 15
    • 0013354882 scopus 로고    scopus 로고
    • K.B. Augustinsson, A titrimetric method for the determination of plasma and red cell cholinesterase activity, Scand. J. Clin. Lab. Invest. 7 (1955) 284-290 [Chem. Abstr. 50 (1956) 11408b].
    • K.B. Augustinsson, A titrimetric method for the determination of plasma and red cell cholinesterase activity, Scand. J. Clin. Lab. Invest. 7 (1955) 284-290 [Chem. Abstr. 50 (1956) 11408b].
  • 16
    • 0023298797 scopus 로고
    • Derivati chinolizidinici ad attività antimicrobica
    • Sparatore A., Veronese M., Sparatore F. Derivati chinolizidinici ad attività antimicrobica. Farmaco Ed. Sci. 42:1987;159-174.
    • (1987) Farmaco Ed. Sci. , vol.42 , pp. 159-174
    • Sparatore, A.1    Veronese, M.2    Sparatore, F.3
  • 17
    • 0027250018 scopus 로고
    • Thiolupinine and some derivatives of pharmacological interest
    • Novelli F., Sparatore F. Thiolupinine and some derivatives of pharmacological interest. Farmaco. 48:1993;1021-1049.
    • (1993) Farmaco , vol.48 , pp. 1021-1049
    • Novelli, F.1    Sparatore, F.2
  • 18
    • 85031081201 scopus 로고    scopus 로고
    • F. Häfliger, W. Schindler, N-Acyl derivatives of iminodibenzyl, US Patent 2,666,051 (1954) [Chem. Abstr. 49 (1955) 9041f].
    • F. Häfliger, W. Schindler, N-Acyl derivatives of iminodibenzyl, US Patent 2,666,051 (1954) [Chem. Abstr. 49 (1955) 9041f].
  • 19
    • 0141805132 scopus 로고
    • Phenothiazine derivatives of pharmacological interest
    • Ekstrand T. Phenothiazine derivatives of pharmacological interest. Acta Chem. Scand. 3:1949;302-303.
    • (1949) Acta Chem. Scand. , vol.3 , pp. 302-303
    • Ekstrand, T.1
  • 20
    • 85031076403 scopus 로고    scopus 로고
    • H.G. Morren, Substituted N-acylphenothiazines, Belg. Patent 586,033 (1960) [Chem. Abstr. 54 (1960) 18561e].
    • H.G. Morren, Substituted N-acylphenothiazines, Belg. Patent 586,033 (1960) [Chem. Abstr. 54 (1960) 18561e].
  • 21
    • 85031067023 scopus 로고    scopus 로고
    • Société des usines chimiques Rhone-Poulenc, Phenothiazine derivatives, Brit. Patent 740,932 (1955) [Chem. Abstr. 51 (1957) 500i].
    • Société des usines chimiques Rhone-Poulenc, Phenothiazine derivatives, Brit. Patent 740,932 (1955) [Chem. Abstr. 51 (1957) 500i].
  • 22
    • 85031078815 scopus 로고    scopus 로고
    • F. Kazutoshi, S. Atsuo, S. Kazuo, O. Kazuo, 10-Chloroacetylphenothiazine, Japan Patent 74,27,191 [Chem. Abstr. 82 (1975) 140161w].
    • F. Kazutoshi, S. Atsuo, S. Kazuo, O. Kazuo, 10-Chloroacetylphenothiazine, Japan Patent 74,27,191 [Chem. Abstr. 82 (1975) 140161w].
  • 23
    • 0141693575 scopus 로고
    • Phenothiazine derivatives. VI. Experiments for the preparation of phenothiazines with selective coronary dilator activity
    • Toldy L., Toth I., Fekete M., Borsy J. Phenothiazine derivatives. VI. Experiments for the preparation of phenothiazines with selective coronary dilator activity. Acta Chim. Acad. Sci. Hung. 44:1965;301-325.
    • (1965) Acta Chim. Acad. Sci. Hung. , vol.44 , pp. 301-325
    • Toldy, L.1    Toth, I.2    Fekete, M.3    Borsy, J.4
  • 24
    • 0141470331 scopus 로고
    • Phenothiazine derivatives. IV. Synthesis of 10-(piperazinoacyl)phenothiazines
    • Hromatka O., Schlager L.H., Sauter F. Phenothiazine derivatives. IV. Synthesis of 10-(piperazinoacyl)phenothiazines. Monatsh. 88:1957;234-241.
    • (1957) Monatsh. , vol.88 , pp. 234-241
    • Hromatka, O.1    Schlager, L.H.2    Sauter, F.3
  • 26
    • 0023821640 scopus 로고
    • 2-receptors mediating opposite effects on neuromuscular transmission in rabbit vas deferens
    • 2-receptors mediating opposite effects on neuromuscular transmission in rabbit vas deferens. Eur. J. Pharmacol. 151:1988;205-221.
    • (1988) Eur. J. Pharmacol. , vol.151 , pp. 205-221
    • Eltze, M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.