Synthesis and antileishmanial activity of new imidazolidin-2-one derivatives

European Journal of Medicinal Chemistry

Volumn 38, Issue 7-8, 2003, Pages 711-718

  Robert, Jean Michel H ^a   Sabourin, Caroline ^a   Alvarez, Nidia ^b   Robert Piessard, Sylvie ^a   Le Baut, Guillaume ^a   Le Pape, Patrice ^b  

^a Laboratoire de Pharmacochimie   (France)

^b UNIVERSITÉ DE NANTES   (France)

Author keywords

Antileishmanial activity; Imidazolidin 2 one; L.mexicana. L infantum; Promastigote

Indexed keywords

1 (3 METHYLISOXAZOL 5 YL) 3 (4 BROMOBENZYL)IMIDAZOLIDIN 2 ONE; 1 (3 METHYLISOXAZOL 5 YL)IMIDAZOLIDIN 2 ONE; 1 (4,6 DIMETHYLPYRIDIN 2 YL) 3 (NAPHTH 2 YLSULFONYL)IMIDAZOLIDIN 2 ONE; 1 (4,6 DIMETHYLPYRIDIN 2 YL)IMIDAZOLIDIN 2 ONE; 1 (5 METHYLTHIAZOL 2 YL) 3 (4 TOLUENESULFONYL)IMIDAZOLIDIN 2 ONE; 1 (5 METHYLTHIAZOL 2 YL)IMIDAZOLIDIN 2 ONE; 3 (3,5 DIFLUOROBENZOYL) 1 (4,6 DIMETHYLPYRIDIN 2 YL)IMIDAZOLIDIN 2 ONE; ANTILEISHMANIAL AGENT; IMIDAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

AMASTIGOTE; ANTIPROTOZOAL ACTIVITY; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; LEISHMANIA INFANTUM; LEISHMANIA MEXICANA; NONHUMAN; PROMASTIGOTE;

EID: 0043158818     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(03)00119-3     Document Type: Article

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