New method for the preparation of solid-phase bound isocyanocarboxylic acids and Ugi reactions therewith

Tetrahedron Letters

Volumn 44, Issue 37, 2003, Pages 7015-7018

  Henkel, Bernd ^a   Sax, Michael ^b   Dömling, Alexander ^a  

^a Morphochem AG   (Germany)

^b UNIVERSITY OF MÜNSTER   (Germany)

Author keywords

Isocyanocarboxylic acid; Multicomponent reaction; Solid phase synthesis; Ugi reaction

Indexed keywords

CARBOXYLIC ACID DERIVATIVE; ISOCYANIC ACID DERIVATIVE; POTASSIUM SALT; RESIN;

ARTICLE; BROMINATION; CHEMICAL REACTION; SOLID; SYNTHESIS;

EID: 0042158218     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(03)01793-3     Document Type: Article

References (13)

1. Arshady R., Ugi I. Polymer. 31:1990;1164-1169.
2. Skorna G., Ugi I. Chem. Ber. 111:1978;3965-3968.
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11. Hoppe I., Schöllkopf U. Chem. Ber. 109:1976;482-487.
12. Patent pending; resin-bound isocyanocarboxylic acids are available from Priaton, Bahnhofstrasse 9-15, D-82327 Tutzing, Germany (www.priaton.de).
13. 3): δ 21.7; 22.6; 25.8; 25.9; 29.1; 36.5; 37.8; 37.9; 38.3; 38.4; 54.8; 67.3; 124.6; 124.7; 126.9; 128.9; 129.0; 129.1; 129.2; 129.6; 129.7; 129.8; 130.0; 131.5; 135.2; 140.1; 140.4; 154.3; 169.3; 170.3; 170.4.